CA1113452A - Corticoides hydrosolubles - Google Patents

Corticoides hydrosolubles

Info

Publication number
CA1113452A
CA1113452A CA300,512A CA300512A CA1113452A CA 1113452 A CA1113452 A CA 1113452A CA 300512 A CA300512 A CA 300512A CA 1113452 A CA1113452 A CA 1113452A
Authority
CA
Canada
Prior art keywords
alpha
methyl
beta
delta
pregnadien
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA300,512A
Other languages
English (en)
Inventor
Ulrich Kerb
Rudolf Wiechert
Joachim-Friedrich Kapp
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer Pharma AG
Original Assignee
Schering AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering AG filed Critical Schering AG
Application granted granted Critical
Publication of CA1113452A publication Critical patent/CA1113452A/fr
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J51/00Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J5/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • C07J5/0007Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond not substituted in position 17 alfa
    • C07J5/0023Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond not substituted in position 17 alfa substituted in position 16
    • C07J5/003Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond not substituted in position 17 alfa substituted in position 16 by a saturated or unsaturated hydrocarbon group including 16-alkylidene substitutes
    • C07J5/0038Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond not substituted in position 17 alfa substituted in position 16 by a saturated or unsaturated hydrocarbon group including 16-alkylidene substitutes by an alkyl group

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Saccharide Compounds (AREA)
CA300,512A 1977-04-06 1978-04-05 Corticoides hydrosolubles Expired CA1113452A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DEP2715853.8 1977-04-06
DE19772715853 DE2715853A1 (de) 1977-04-06 1977-04-06 Wasserloesliche kortikoide

Publications (1)

Publication Number Publication Date
CA1113452A true CA1113452A (fr) 1981-12-01

Family

ID=6005979

Family Applications (1)

Application Number Title Priority Date Filing Date
CA300,512A Expired CA1113452A (fr) 1977-04-06 1978-04-05 Corticoides hydrosolubles

Country Status (29)

Country Link
JP (1) JPS53149963A (fr)
AT (1) ATA239978A (fr)
AU (1) AU3481178A (fr)
BE (1) BE865760A (fr)
BG (1) BG28578A3 (fr)
CA (1) CA1113452A (fr)
CH (1) CH638537A5 (fr)
CS (1) CS198295B2 (fr)
DD (1) DD135082A5 (fr)
DE (1) DE2715853A1 (fr)
DK (1) DK153378A (fr)
EG (1) EG13249A (fr)
ES (1) ES468572A1 (fr)
FI (1) FI781053A (fr)
FR (1) FR2386557A1 (fr)
GB (1) GB1602266A (fr)
IE (1) IE46602B1 (fr)
IL (1) IL54443A0 (fr)
IT (1) IT1094296B (fr)
LU (1) LU79375A1 (fr)
NL (1) NL7803188A (fr)
NO (1) NO781200L (fr)
NZ (1) NZ186745A (fr)
PL (1) PL114096B1 (fr)
PT (1) PT67872B (fr)
RO (1) RO81076A2 (fr)
SE (1) SE7803837L (fr)
SU (1) SU668611A3 (fr)
ZA (1) ZA781977B (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4948533A (en) * 1984-03-28 1990-08-14 The Upjohn Company 11a-hydroxy steroid diester

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1169444B (de) * 1961-02-22 1964-05-06 Schering Ag Verfahren zur Herstellung von ?-16ª‡-Methylsteroiden
YU34304B (en) * 1968-08-17 1979-04-30 Schering Ag Process for preparing corticoid-21-mono-phosphates
DK290774A (fr) * 1973-06-08 1975-02-03 Schering Ag

Also Published As

Publication number Publication date
DE2715853A1 (de) 1978-10-19
RO81076B1 (ro) 1983-01-30
NO781200L (no) 1978-10-09
EG13249A (en) 1980-12-31
PL114096B1 (en) 1981-01-31
PT67872A (fr) 1978-05-01
BG28578A3 (bg) 1980-05-15
AU3481178A (en) 1979-10-11
NZ186745A (en) 1980-10-24
GB1602266A (en) 1981-11-11
FR2386557B1 (fr) 1980-02-01
CH638537A5 (en) 1983-09-30
SE7803837L (sv) 1978-10-07
ATA239978A (de) 1981-06-15
LU79375A1 (de) 1978-07-13
IT7821995A0 (it) 1978-04-05
FR2386557A1 (fr) 1978-11-03
BE865760A (fr) 1978-10-06
ES468572A1 (es) 1978-12-01
IT1094296B (it) 1985-07-26
CS198295B2 (en) 1980-05-30
PL205800A1 (pl) 1979-01-29
RO81076A2 (fr) 1983-02-01
NL7803188A (nl) 1978-10-10
IL54443A0 (en) 1978-07-31
DD135082A5 (de) 1979-04-11
ZA781977B (en) 1979-03-28
IE46602B1 (en) 1983-07-27
FI781053A (fi) 1978-10-07
SU668611A3 (ru) 1979-06-15
JPS53149963A (en) 1978-12-27
IE780672L (en) 1978-10-06
DK153378A (da) 1978-10-07
PT67872B (fr) 1979-11-14

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Legal Events

Date Code Title Description
MKEX Expiry