BRPI0818872A2 - Método para prevenir efeitos adversos por glp-1 - Google Patents
Método para prevenir efeitos adversos por glp-1Info
- Publication number
- BRPI0818872A2 BRPI0818872A2 BRPI0818872A BRPI0818872A2 BR PI0818872 A2 BRPI0818872 A2 BR PI0818872A2 BR PI0818872 A BRPI0818872 A BR PI0818872A BR PI0818872 A2 BRPI0818872 A2 BR PI0818872A2
- Authority
- BR
- Brazil
- Prior art keywords
- adverse effects
- glp
- prevent
- prevent glp
- adverse
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/26—Glucagons
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/28—Insulins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61M—DEVICES FOR INTRODUCING MEDIA INTO, OR ONTO, THE BODY; DEVICES FOR TRANSDUCING BODY MEDIA OR FOR TAKING MEDIA FROM THE BODY; DEVICES FOR PRODUCING OR ENDING SLEEP OR STUPOR
- A61M15/00—Inhalators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Gastroenterology & Hepatology (AREA)
- Immunology (AREA)
- Zoology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Hematology (AREA)
- Pulmonology (AREA)
- Heart & Thoracic Surgery (AREA)
- Biomedical Technology (AREA)
- Anesthesiology (AREA)
- Obesity (AREA)
- Emergency Medicine (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US98236807P | 2007-10-24 | 2007-10-24 | |
US98562007P | 2007-11-05 | 2007-11-05 | |
US3374008P | 2008-03-04 | 2008-03-04 | |
US5212708P | 2008-05-09 | 2008-05-09 | |
PCT/US2008/081218 WO2009055740A2 (en) | 2007-10-24 | 2008-10-24 | Method of preventing adverse effects by glp-1 |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0818872A2 true BRPI0818872A2 (pt) | 2015-05-05 |
Family
ID=40546046
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0818872 BRPI0818872A2 (pt) | 2007-10-24 | 2008-10-24 | Método para prevenir efeitos adversos por glp-1 |
Country Status (15)
Country | Link |
---|---|
US (4) | US8377869B2 (pt) |
EP (2) | EP2211842B1 (pt) |
JP (2) | JP2011500850A (pt) |
KR (2) | KR101736535B1 (pt) |
CN (1) | CN101969927A (pt) |
AU (2) | AU2008316634B2 (pt) |
BR (1) | BRPI0818872A2 (pt) |
CA (1) | CA2703338A1 (pt) |
DK (1) | DK2211842T3 (pt) |
ES (1) | ES2547529T3 (pt) |
HU (1) | HUE025485T2 (pt) |
MX (1) | MX2010004510A (pt) |
PL (1) | PL2211842T3 (pt) |
RU (2) | RU2474415C2 (pt) |
WO (1) | WO2009055740A2 (pt) |
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US20080260838A1 (en) * | 2003-08-01 | 2008-10-23 | Mannkind Corporation | Glucagon-like peptide 1 (glp-1) pharmaceutical formulations |
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BR122019022692B1 (pt) | 2004-08-23 | 2023-01-10 | Mannkind Corporation | Composição terapêutica em pó seco contendo dicetopiperazina, pelo menos um tipo de cátion e um agente biologicamente ativo |
HUE028691T2 (en) | 2005-09-14 | 2016-12-28 | Mannkind Corp | A method for formulating a drug based on increasing the affinity of crystalline microparticle surfaces towards active ingredients |
EP1986679B1 (en) | 2006-02-22 | 2017-10-25 | MannKind Corporation | A method for improving the pharmaceutic properties of microparticles comprising diketopiperazine and an active agent |
US8785396B2 (en) * | 2007-10-24 | 2014-07-22 | Mannkind Corporation | Method and composition for treating migraines |
JP2011500850A (ja) | 2007-10-24 | 2011-01-06 | マンカインド コーポレイション | Glp−1による副作用を防止する方法 |
AR072114A1 (es) | 2008-06-13 | 2010-08-04 | Mannkind Corp | Un inhalador de polvo seco y sistema para suministro de farmacos |
US8485180B2 (en) | 2008-06-13 | 2013-07-16 | Mannkind Corporation | Dry powder drug delivery system |
BRPI0914308B8 (pt) | 2008-06-20 | 2021-06-22 | Mannkind Corp | sistema de inalação |
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AU2015203301B2 (en) * | 2009-11-02 | 2017-05-25 | Mannkind Corporation | Reactor for producing pharmaceutical particles in a precipitation process |
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KR101931392B1 (ko) * | 2010-11-09 | 2018-12-20 | 맨카인드 코포레이션 | 세로토닌 수용체 작용제 및 디케토피페라진을 포함하는 편두통 치료용 조성물 |
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JP6018640B2 (ja) | 2011-10-24 | 2016-11-02 | マンカインド コーポレイション | 疼痛を緩和するのに有効な鎮痛組成物並びに当該組成物を含む乾燥粉末及び乾燥粉末薬剤輸送システム |
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US10159644B2 (en) | 2012-10-26 | 2018-12-25 | Mannkind Corporation | Inhalable vaccine compositions and methods |
CN104870009B (zh) | 2012-12-21 | 2021-05-18 | 赛诺菲 | 官能化的毒蜥外泌肽-4衍生物 |
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-
2008
- 2008-10-24 JP JP2010531298A patent/JP2011500850A/ja active Pending
- 2008-10-24 AU AU2008316634A patent/AU2008316634B2/en not_active Ceased
- 2008-10-24 RU RU2010120666/15A patent/RU2474415C2/ru not_active IP Right Cessation
- 2008-10-24 EP EP08841194.7A patent/EP2211842B1/en not_active Not-in-force
- 2008-10-24 US US12/258,340 patent/US8377869B2/en active Active
- 2008-10-24 CN CN2008801226703A patent/CN101969927A/zh active Pending
- 2008-10-24 KR KR1020137027725A patent/KR101736535B1/ko active IP Right Grant
- 2008-10-24 ES ES08841194.7T patent/ES2547529T3/es active Active
- 2008-10-24 MX MX2010004510A patent/MX2010004510A/es active IP Right Grant
- 2008-10-24 WO PCT/US2008/081218 patent/WO2009055740A2/en active Application Filing
- 2008-10-24 KR KR1020107011096A patent/KR101736502B1/ko active IP Right Grant
- 2008-10-24 PL PL08841194T patent/PL2211842T3/pl unknown
- 2008-10-24 BR BRPI0818872 patent/BRPI0818872A2/pt not_active IP Right Cessation
- 2008-10-24 DK DK08841194.7T patent/DK2211842T3/en active
- 2008-10-24 CA CA2703338A patent/CA2703338A1/en not_active Abandoned
- 2008-10-24 HU HUE08841194A patent/HUE025485T2/en unknown
- 2008-10-24 EP EP15178836.1A patent/EP2954893A1/en not_active Withdrawn
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2012
- 2012-10-30 RU RU2012146344/15A patent/RU2012146344A/ru not_active Application Discontinuation
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2013
- 2013-01-02 US US13/732,911 patent/US20130125886A1/en not_active Abandoned
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2014
- 2014-05-20 AU AU2014202731A patent/AU2014202731A1/en not_active Abandoned
- 2014-09-18 JP JP2014190113A patent/JP2015013892A/ja active Pending
-
2020
- 2020-01-14 US US16/742,193 patent/US20200147219A1/en not_active Abandoned
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2022
- 2022-08-15 US US17/887,856 patent/US20220387593A1/en active Pending
Also Published As
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US20200147219A1 (en) | 2020-05-14 |
US8377869B2 (en) | 2013-02-19 |
RU2012146344A (ru) | 2014-05-10 |
AU2008316634A1 (en) | 2009-04-30 |
WO2009055740A3 (en) | 2009-06-11 |
EP2211842A2 (en) | 2010-08-04 |
US20090110647A1 (en) | 2009-04-30 |
CA2703338A1 (en) | 2009-04-30 |
CN101969927A (zh) | 2011-02-09 |
DK2211842T3 (en) | 2015-09-21 |
US20130125886A1 (en) | 2013-05-23 |
RU2474415C2 (ru) | 2013-02-10 |
RU2010120666A (ru) | 2011-11-27 |
EP2211842B1 (en) | 2015-08-12 |
AU2008316634B2 (en) | 2014-02-27 |
EP2954893A1 (en) | 2015-12-16 |
JP2015013892A (ja) | 2015-01-22 |
KR20130123467A (ko) | 2013-11-12 |
WO2009055740A2 (en) | 2009-04-30 |
AU2014202731A1 (en) | 2014-06-12 |
KR101736502B1 (ko) | 2017-05-16 |
MX2010004510A (es) | 2010-07-02 |
US20220387593A1 (en) | 2022-12-08 |
HUE025485T2 (en) | 2016-02-29 |
PL2211842T3 (pl) | 2015-12-31 |
KR101736535B1 (ko) | 2017-05-16 |
ES2547529T3 (es) | 2015-10-07 |
JP2011500850A (ja) | 2011-01-06 |
KR20100093055A (ko) | 2010-08-24 |
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