BRPI0814825A2 - Composto, processo para a preparação do composto, composição farmacêutica que o compreende, seu uso e métodos para o tratamento ou profilaxia de diabetes, obesidade, distúrbios de alimentação ou dislipimedia e diabetes do tipo ii - Google Patents

Composto, processo para a preparação do composto, composição farmacêutica que o compreende, seu uso e métodos para o tratamento ou profilaxia de diabetes, obesidade, distúrbios de alimentação ou dislipimedia e diabetes do tipo ii

Info

Publication number
BRPI0814825A2
BRPI0814825A2 BRPI0814825-2A2A BRPI0814825A BRPI0814825A2 BR PI0814825 A2 BRPI0814825 A2 BR PI0814825A2 BR PI0814825 A BRPI0814825 A BR PI0814825A BR PI0814825 A2 BRPI0814825 A2 BR PI0814825A2
Authority
BR
Brazil
Prior art keywords
diabetes
compound
dislipimedia
prophylaxy
obesity
Prior art date
Application number
BRPI0814825-2A2A
Other languages
English (en)
Inventor
Paul Gillespie
Kevin Richard Guertin
Lida Qi
Qiang Zhang
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BRPI0814825A2 publication Critical patent/BRPI0814825A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
BRPI0814825-2A2A 2007-07-17 2008-07-07 Composto, processo para a preparação do composto, composição farmacêutica que o compreende, seu uso e métodos para o tratamento ou profilaxia de diabetes, obesidade, distúrbios de alimentação ou dislipimedia e diabetes do tipo ii BRPI0814825A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US95016807P 2007-07-17 2007-07-17
PCT/EP2008/058804 WO2009010416A2 (en) 2007-07-17 2008-07-07 Inhibitors of 11b-hydroxysteroid dehydrogenase

Publications (1)

Publication Number Publication Date
BRPI0814825A2 true BRPI0814825A2 (pt) 2015-02-03

Family

ID=40019292

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0814825-2A2A BRPI0814825A2 (pt) 2007-07-17 2008-07-07 Composto, processo para a preparação do composto, composição farmacêutica que o compreende, seu uso e métodos para o tratamento ou profilaxia de diabetes, obesidade, distúrbios de alimentação ou dislipimedia e diabetes do tipo ii

Country Status (16)

Country Link
US (1) US7790711B2 (pt)
EP (1) EP2178845B1 (pt)
JP (1) JP5189165B2 (pt)
KR (1) KR101158191B1 (pt)
CN (1) CN101743226B (pt)
AR (1) AR067538A1 (pt)
AU (1) AU2008277783B2 (pt)
BR (1) BRPI0814825A2 (pt)
CA (1) CA2693457C (pt)
CL (1) CL2008002052A1 (pt)
ES (1) ES2423181T3 (pt)
PE (1) PE20090813A1 (pt)
RU (1) RU2440989C2 (pt)
TW (1) TWI372623B (pt)
WO (1) WO2009010416A2 (pt)
ZA (1) ZA201000318B (pt)

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Also Published As

Publication number Publication date
JP5189165B2 (ja) 2013-04-24
CA2693457A1 (en) 2009-01-22
WO2009010416A2 (en) 2009-01-22
WO2009010416A3 (en) 2009-03-05
EP2178845B1 (en) 2013-06-19
RU2440989C2 (ru) 2012-01-27
RU2010105299A (ru) 2011-08-27
ES2423181T3 (es) 2013-09-18
TWI372623B (en) 2012-09-21
EP2178845A2 (en) 2010-04-28
PE20090813A1 (es) 2009-06-27
AR067538A1 (es) 2009-10-14
CL2008002052A1 (es) 2009-05-22
CN101743226B (zh) 2012-10-10
JP2010533670A (ja) 2010-10-28
US20090023709A1 (en) 2009-01-22
KR101158191B1 (ko) 2012-06-19
US7790711B2 (en) 2010-09-07
CA2693457C (en) 2012-10-23
AU2008277783B2 (en) 2012-09-20
ZA201000318B (en) 2010-10-27
CN101743226A (zh) 2010-06-16
TW200913992A (en) 2009-04-01
KR20100034763A (ko) 2010-04-01
AU2008277783A1 (en) 2009-01-22

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