BRPI0615690B8 - compostos heterocíclicos de hidroxamato, seus usos e composição farmacêutica - Google Patents

compostos heterocíclicos de hidroxamato, seus usos e composição farmacêutica

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Publication number
BRPI0615690B8
BRPI0615690B8 BRPI0615690A BRPI0615690A BRPI0615690B8 BR PI0615690 B8 BRPI0615690 B8 BR PI0615690B8 BR PI0615690 A BRPI0615690 A BR PI0615690A BR PI0615690 A BRPI0615690 A BR PI0615690A BR PI0615690 B8 BRPI0615690 B8 BR PI0615690B8
Authority
BR
Brazil
Prior art keywords
pharmaceutical composition
compounds
heterocyclic
hydroxamate compounds
heterocyclic hydroxamate
Prior art date
Application number
BRPI0615690A
Other languages
English (en)
Portuguese (pt)
Inventor
Chen Dizhong
T Sun Eric
Wang Haishan
Chi Lik Lee Ken
Yu Niefang
Ling Lye Pek
Deng Weiping
Original Assignee
Mei Pharma Inc
Sstarbio Pte Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mei Pharma Inc, Sstarbio Pte Ltd filed Critical Mei Pharma Inc
Publication of BRPI0615690A2 publication Critical patent/BRPI0615690A2/pt
Publication of BRPI0615690B1 publication Critical patent/BRPI0615690B1/pt
Publication of BRPI0615690B8 publication Critical patent/BRPI0615690B8/pt

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    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
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    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/08Radicals containing only hydrogen and carbon atoms
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
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    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
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    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/10Radicals substituted by halogen atoms or nitro radicals
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    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
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    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
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    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
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BRPI0615690A 2005-09-08 2006-08-01 compostos heterocíclicos de hidroxamato, seus usos e composição farmacêutica BRPI0615690B8 (pt)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US71482705P 2005-09-08 2005-09-08
US60/714.827 2005-09-08
US78381906P 2006-03-21 2006-03-21
US60/783.819 2006-03-21
PCT/SG2006/000217 WO2007030080A1 (en) 2005-09-08 2006-08-01 Heterocyclic compounds

Publications (3)

Publication Number Publication Date
BRPI0615690A2 BRPI0615690A2 (pt) 2011-05-24
BRPI0615690B1 BRPI0615690B1 (pt) 2020-12-08
BRPI0615690B8 true BRPI0615690B8 (pt) 2021-05-25

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TWI393708B (zh) 2013-04-21
JP5207064B2 (ja) 2013-06-12
CY1111789T1 (el) 2015-10-07
PT1937650E (pt) 2011-09-21
TW200745047A (en) 2007-12-16
JP2009507829A (ja) 2009-02-26
PL1937650T3 (pl) 2011-11-30
HK1123038A1 (en) 2009-06-05
BRPI0615690B1 (pt) 2020-12-08
BRPI0615690A2 (pt) 2011-05-24
US20090048300A1 (en) 2009-02-19
ATE512953T1 (de) 2011-07-15
DK1937650T3 (da) 2011-10-03
US8143282B2 (en) 2012-03-27
EP1937650A1 (en) 2008-07-02
AR055364A1 (es) 2007-08-22
KR101346823B1 (ko) 2014-02-14
MY144970A (en) 2011-11-30
KR20080046219A (ko) 2008-05-26
EP1937650A4 (en) 2010-02-24
WO2007030080A1 (en) 2007-03-15
NZ594108A (en) 2012-12-21

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