BRPI0513083A - oxazolidinonas contendo oxindóis como agentes antibacterianos - Google Patents

oxazolidinonas contendo oxindóis como agentes antibacterianos

Info

Publication number
BRPI0513083A
BRPI0513083A BRPI0513083-2A BRPI0513083A BRPI0513083A BR PI0513083 A BRPI0513083 A BR PI0513083A BR PI0513083 A BRPI0513083 A BR PI0513083A BR PI0513083 A BRPI0513083 A BR PI0513083A
Authority
BR
Brazil
Prior art keywords
antibacterial agents
oxindoles
oxazolidinones containing
oxazolidinones
oxindols
Prior art date
Application number
BRPI0513083-2A
Other languages
English (en)
Inventor
Gary Wayne Luehr
Rama Jain
Adam Robert Renslo
Vara Prasad Venkata Na Josyula
Mikhail Fedorovich Gordeev
Original Assignee
Pharmacia & Upjohn Co Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35079333&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0513083(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacia & Upjohn Co Llc filed Critical Pharmacia & Upjohn Co Llc
Publication of BRPI0513083A publication Critical patent/BRPI0513083A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

OXAZOLIDINONAS CONTENDO OXINDóIS COMO AGENTES ANTIBACTERIANOS. A presente invenção refere-se a novos derivados de oxazolidinonas de oxindóis da fórmula I, ou um sal farmaceuticamente aceitável do mesmo em que Y¬ 1¬ é -CH- ou -CF-; R¬ 1¬ é -C~ 1-4~ alquila, opcionalmente substituída por um átomo de flúor, ou R¬ 1¬ é -C~ 3-5~ cicloalquila; e R¬ 2¬ é -H ou -CH~ 3~. Estes compostos são úteis como agentes anti-bacterianos.
BRPI0513083-2A 2004-08-06 2005-07-19 oxazolidinonas contendo oxindóis como agentes antibacterianos BRPI0513083A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US59982204P 2004-08-06 2004-08-06
PCT/IB2005/002197 WO2006016221A1 (en) 2004-08-06 2005-07-19 Oxazolidinones containing oxindoles as antibacterial agents

Publications (1)

Publication Number Publication Date
BRPI0513083A true BRPI0513083A (pt) 2008-04-22

Family

ID=35079333

Family Applications (2)

Application Number Title Priority Date Filing Date
BRPI0513083-2A BRPI0513083A (pt) 2004-08-06 2005-07-19 oxazolidinonas contendo oxindóis como agentes antibacterianos
BRPI0514020-0A BRPI0514020A (pt) 2004-08-06 2005-07-19 oxindóis oxazolidinonas como agentes antibacterianos

Family Applications After (1)

Application Number Title Priority Date Filing Date
BRPI0514020-0A BRPI0514020A (pt) 2004-08-06 2005-07-19 oxindóis oxazolidinonas como agentes antibacterianos

Country Status (24)

Country Link
US (2) US20080262056A1 (pt)
EP (2) EP1781642A1 (pt)
JP (2) JP2008509126A (pt)
CN (1) CN101001853A (pt)
AP (1) AP2007003904A0 (pt)
AR (1) AR050101A1 (pt)
AU (1) AU2005270951A1 (pt)
BR (2) BRPI0513083A (pt)
CA (2) CA2576041A1 (pt)
EA (1) EA200700322A1 (pt)
GT (1) GT200500204A (pt)
IL (1) IL180957A0 (pt)
MA (1) MA28793B1 (pt)
MX (2) MX2007001568A (pt)
NL (1) NL1029686C2 (pt)
NO (1) NO20071230L (pt)
PA (1) PA8640901A1 (pt)
PE (1) PE20060351A1 (pt)
SV (1) SV2006002180A (pt)
TN (1) TNSN07043A1 (pt)
TW (1) TWI289448B (pt)
UY (1) UY29048A1 (pt)
WO (2) WO2006016221A1 (pt)
ZA (1) ZA200700476B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2006231918A1 (en) * 2005-04-06 2006-10-12 Pharmacia & Upjohn Company Llc An oxindole oxazolidinone as antibacterial agent
AU2006231919A1 (en) 2005-04-06 2006-10-12 Pharmacia & Upjohn Company Llc 7-fluoro-1,3-dihydro-indol-2-one oxazolidinones as antibacterial agents
CN103420995B (zh) * 2013-09-07 2015-07-01 吉首大学 噁唑烷酮-烷胺基-呋喃酮型化合物及其制法和用途
CN103483329B (zh) * 2013-09-07 2015-08-05 吉首大学 呋喃酮-芳基-噁唑烷酮型化合物及其制法和用途
CN111018840B (zh) * 2017-10-25 2022-09-09 西南大学 3-咪唑取代的靛红唑醇类化合物及其制备方法和医药应用

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1990002744A1 (en) * 1988-09-15 1990-03-22 The Upjohn Company In position 3 substituted-5-beta-amidomethyl-oxazolidin-2-ones
US5164510A (en) * 1988-09-15 1992-11-17 The Upjohn Company 5'Indolinyl-5β-amidomethyloxazolidin-2-ones
DE4425612A1 (de) * 1994-07-20 1996-04-04 Bayer Ag 6-gliedrige stickstoffhaltige Heteroaryl-oxazolidinone
WO1996015130A1 (en) * 1994-11-15 1996-05-23 Pharmacia + Upjohn Company Bicyclic oxazine and thiazine oxazolidinone antibacterials
HRP960159A2 (en) * 1995-04-21 1997-08-31 Bayer Ag Benzocyclopentane oxazolidinones containing heteroatoms
BR9610474A (pt) * 1995-09-01 1999-03-02 Upjohn Co Feniloxazolidinonas tendo uma ligação c-c a anéis heterocíclicos com 4-8 membros
DE19601265A1 (de) * 1996-01-16 1997-07-17 Bayer Ag 2-Oxo- und 2-Thio-1,2-dihydrochinolinyl-oxazolidinone
DE19601627A1 (de) * 1996-01-18 1997-07-24 Bayer Ag Heteroatomhaltige Cyclopentanopyridyl-Oxazolidinone
GB9601666D0 (en) * 1996-01-27 1996-03-27 Zeneca Ltd Chemical compounds
GB9702213D0 (en) * 1996-02-24 1997-03-26 Zeneca Ltd Chemical compounds
GB9609919D0 (en) * 1996-05-11 1996-07-17 Zeneca Ltd Chemical compounds
EP0920421B1 (en) * 1996-08-21 2002-11-06 PHARMACIA & UPJOHN COMPANY Isoxazoline derivatives useful as antimicrobials
GB9717804D0 (en) * 1997-08-22 1997-10-29 Zeneca Ltd Chemical compounds
KR20010015910A (ko) * 1998-01-23 2001-02-26 로렌스 티. 마이젠헬더 옥사졸리디논 조합 라이브러리, 조성물 및 제조 방법
GB9812019D0 (en) * 1998-06-05 1998-07-29 Zeneca Ltd Chemical compounds
DE60001807T2 (de) * 1999-02-01 2003-11-06 Upjohn Co VERFAHREN ZU HERSTELLUNG VON o-FLUORIERTEN TETRAHYDROTHIOPYRAN CARBAMATEN
NZ515754A (en) * 1999-05-27 2003-10-31 Upjohn Co Bicyclic oxazolidinone compounds, pharmaceuticals thereof and their use as antibacterial agents
AR038536A1 (es) * 2002-02-25 2005-01-19 Upjohn Co N-aril-2-oxazolidinona-5- carboxamidas y sus derivados
US7012088B2 (en) * 2003-02-24 2006-03-14 Pharmacia & Upjohn Company Indolone oxazolidinones and derivatives thereof
AU2006231919A1 (en) * 2005-04-06 2006-10-12 Pharmacia & Upjohn Company Llc 7-fluoro-1,3-dihydro-indol-2-one oxazolidinones as antibacterial agents

Also Published As

Publication number Publication date
BRPI0514020A (pt) 2008-05-27
NO20071230L (no) 2007-05-04
US20060030609A1 (en) 2006-02-09
EA200700322A1 (ru) 2007-08-31
TWI289448B (en) 2007-11-11
WO2006016221A1 (en) 2006-02-16
CA2576041A1 (en) 2006-02-16
CA2575702A1 (en) 2006-02-16
MA28793B1 (fr) 2007-08-01
CN101001853A (zh) 2007-07-18
PE20060351A1 (es) 2006-05-03
SV2006002180A (es) 2006-06-26
PA8640901A1 (es) 2007-01-17
AR050101A1 (es) 2006-09-27
AP2007003904A0 (en) 2007-02-28
US20080262056A1 (en) 2008-10-23
GT200500204A (es) 2006-03-02
MX2007001568A (es) 2007-04-16
WO2006016220A1 (en) 2006-02-16
JP2008509126A (ja) 2008-03-27
NL1029686A1 (nl) 2006-02-07
NL1029686C2 (nl) 2006-07-18
JP2008509125A (ja) 2008-03-27
MX2007001526A (es) 2007-03-27
ZA200700476B (en) 2008-10-29
UY29048A1 (es) 2006-03-31
IL180957A0 (en) 2007-07-04
EP1781642A1 (en) 2007-05-09
EP1781643A1 (en) 2007-05-09
AU2005270951A1 (en) 2006-02-16
TW200612924A (en) 2006-05-01
TNSN07043A1 (fr) 2008-06-02

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 5A E 6A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2158 DE 15/05/2012.