BRPI0510664B8 - derivados de fenol e tiofenol 3 ou 4-monosubstituído, composição farmacêutica, combinação e uso dos compostos para tratamento de doenças relacionadas ao h3, incluindo transtornos do sistema nervoso central e transtornos inflamatórios - Google Patents

derivados de fenol e tiofenol 3 ou 4-monosubstituído, composição farmacêutica, combinação e uso dos compostos para tratamento de doenças relacionadas ao h3, incluindo transtornos do sistema nervoso central e transtornos inflamatórios

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Publication number
BRPI0510664B8
BRPI0510664B8 BRPI0510664A BRPI0510664A BRPI0510664B8 BR PI0510664 B8 BRPI0510664 B8 BR PI0510664B8 BR PI0510664 A BRPI0510664 A BR PI0510664A BR PI0510664 A BRPI0510664 A BR PI0510664A BR PI0510664 B8 BRPI0510664 B8 BR PI0510664B8
Authority
BR
Brazil
Prior art keywords
thiophenol
disorders
monosubstituted
derivatives
compounds
Prior art date
Application number
BRPI0510664A
Other languages
English (en)
Portuguese (pt)
Inventor
Denis Alexis
Michael Cronin Andrew
Serradeil-Civit Delphine
Lorthiois Edwige
Vergne Fabrice
Rousseau Fiona
Jacobelli Henry
Ian Kemp Mark
Bernardelli Patrick
Martin Denton Stephen
Original Assignee
Warner Lambert Co
Ziarco Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP04291187A external-priority patent/EP1593679A1/en
Priority claimed from GB0504564A external-priority patent/GB0504564D0/en
Application filed by Warner Lambert Co, Ziarco Inc filed Critical Warner Lambert Co
Publication of BRPI0510664A publication Critical patent/BRPI0510664A/pt
Publication of BRPI0510664B1 publication Critical patent/BRPI0510664B1/pt
Publication of BRPI0510664B8 publication Critical patent/BRPI0510664B8/pt

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PCT/IB2005/001114 WO2005108384A1 (en) 2004-05-07 2005-04-19 3- or 4-monosubstituted phenol and thiophenol derivatives useful as h3 ligands

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NZ569608A (en) 2006-01-06 2011-09-30 Sepracor Inc Tetralone-based monoamine reuptake inhibitors
CN101421228B (zh) 2006-03-31 2014-05-21 塞普拉柯公司 手性酰胺和胺的制备
AR060404A1 (es) 2006-04-11 2008-06-11 Novartis Ag Compuestos organicos utiles como inhibidores de dipeptidil-peptidasa iv
CN103382174A (zh) 2006-06-23 2013-11-06 雅培制药有限公司 作为组胺h3受体调节物的环丙胺衍生物
US9108948B2 (en) 2006-06-23 2015-08-18 Abbvie Inc. Cyclopropyl amine derivatives
US7884124B2 (en) 2006-06-30 2011-02-08 Sepracor Inc. Fluoro-substituted inhibitors of D-amino acid oxidase
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