BRPI0510005A - preparação contraceptiva multifase baseada em estrogênio natural com um gestagênio sintético - Google Patents

preparação contraceptiva multifase baseada em estrogênio natural com um gestagênio sintético

Info

Publication number
BRPI0510005A
BRPI0510005A BRPI0510005-4A BRPI0510005A BRPI0510005A BR PI0510005 A BRPI0510005 A BR PI0510005A BR PI0510005 A BRPI0510005 A BR PI0510005A BR PI0510005 A BRPI0510005 A BR PI0510005A
Authority
BR
Brazil
Prior art keywords
preparation
natural estrogen
synthetic
contraceptive
contraceptive preparation
Prior art date
Application number
BRPI0510005-4A
Other languages
English (en)
Inventor
Jan Endrikat
Bernd Duesterberg
Original Assignee
Schering Aktiengellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34979546&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0510005(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Aktiengellschaft filed Critical Schering Aktiengellschaft
Publication of BRPI0510005A publication Critical patent/BRPI0510005A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Endocrinology (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Orthopedics, Nursing, And Contraception (AREA)
  • Steroid Compounds (AREA)
  • Compositions Of Macromolecular Compounds (AREA)

Abstract

PREPARAçãO CONTRACEPTIVA MULTIFASE BASEADA EM ESTROGêNIO NATURAL COM UM GESTAGêNIO SINTéTICO. A presente invenção refere-se a uma preparação contraceptiva multifase que é baseada em um estrogênio natural combinado com um gestagênio sintético. Preparações anovulantes convencionais conhecidas na técnica anterior provaram ser confiáveis e seguras em aplicação em grande escala. O objetivo da invenção é prover uma preparação que ofereça uma segurança contraceptiva maior por toda a duração do ciclo, melhore o comportamento de sangramento cíclico e reduza ou exclua efeitos colaterais, tal como sensibilidade da mama, dores de cabeça, humores depressivos e distúrbios de libido e similares.
BRPI0510005-4A 2004-04-20 2005-04-15 preparação contraceptiva multifase baseada em estrogênio natural com um gestagênio sintético BRPI0510005A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102004019743A DE102004019743B4 (de) 2004-04-20 2004-04-20 Mehrphasenpräparat zur Kontrazeption auf der Basis eines natürlichen Estrogens
PCT/EP2005/004022 WO2005102247A2 (de) 2004-04-20 2005-04-15 Mehrphasenpräparat zur kontrazeption auf der basis eines natürlichen estrogens

Publications (1)

Publication Number Publication Date
BRPI0510005A true BRPI0510005A (pt) 2007-09-18

Family

ID=34979546

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0510005-4A BRPI0510005A (pt) 2004-04-20 2005-04-15 preparação contraceptiva multifase baseada em estrogênio natural com um gestagênio sintético

Country Status (38)

Country Link
US (3) US8071577B2 (pt)
EP (1) EP1740163B2 (pt)
JP (1) JP4908399B2 (pt)
KR (1) KR20060134168A (pt)
CN (1) CN1946383B (pt)
AR (2) AR048830A1 (pt)
AT (1) ATE473734T1 (pt)
AU (1) AU2005235418C1 (pt)
BR (1) BRPI0510005A (pt)
CA (1) CA2561839C (pt)
CR (1) CR8695A (pt)
CY (1) CY1111292T1 (pt)
DE (2) DE102004019743B4 (pt)
DK (1) DK1740163T4 (pt)
EA (1) EA010313B1 (pt)
EC (1) ECSP067000A (pt)
ES (1) ES2348038T5 (pt)
GT (1) GT200500093A (pt)
HK (1) HK1099701A1 (pt)
HR (1) HRP20100513T4 (pt)
IL (2) IL178510A (pt)
ME (1) ME01183B (pt)
MX (1) MXPA06012213A (pt)
MY (1) MY143669A (pt)
NO (1) NO344098B1 (pt)
NZ (1) NZ550417A (pt)
PA (1) PA8630901A1 (pt)
PE (1) PE20060308A1 (pt)
PL (1) PL1740163T5 (pt)
PT (1) PT1740163E (pt)
RS (1) RS51434B2 (pt)
SI (1) SI1740163T2 (pt)
SV (1) SV2006002090A (pt)
TW (1) TWI351960B (pt)
UA (1) UA83915C2 (pt)
UY (1) UY28863A1 (pt)
WO (1) WO2005102247A2 (pt)
ZA (1) ZA200609594B (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102004019743B4 (de) * 2004-04-20 2008-11-27 Bayer Schering Pharma Aktiengesellschaft Mehrphasenpräparat zur Kontrazeption auf der Basis eines natürlichen Estrogens
ATE546144T1 (de) * 2005-10-13 2012-03-15 Bayer Pharma AG Verwendung von estradiolvalerat in kombination mit dienogest zur oralen therapie der dysf unktionellen uterinen blutung in einheit mit einer oralen kontrazeption
ATE424828T1 (de) * 2005-10-13 2009-03-15 Bayer Schering Pharma Ag Verwendung von estradiolvalerat in kombination mit dienogest zur oralen therapie der dysfunktionellen uterinen blutung in einheit mit einer oralen kontrazeption
US8153616B2 (en) 2005-10-17 2012-04-10 Bayer Pharma Aktiengesellschaft Combination preparation for oral contraception and oral therapy of dysfunctional uterine bleeding containing estradiol valerate and dienogest and method of using same
ES2558030T3 (es) 2006-03-02 2016-02-01 Warner Chilcott Company, Llc Método anticonceptivo oral multifásico de ciclo prolongado
DE102006010329A1 (de) * 2006-03-06 2007-09-13 Höltge, Michael, Dipl.-Med. Hormonelles Kontrazeptivum auf der Basis eines Estrogens, eines Gestagens oder einer Kombination von Estrogenen und Gestagenen unter der Zugabe von Testosteron
EP1930010A1 (de) * 2006-10-20 2008-06-11 Bayer Schering Pharma Aktiengesellschaft Verwendung von Estradiolvalerat oder 17ß-Estradiol in Kombination mit Dienogest zur oralen Therapie für den Erhalt und/oder die Steigerung der weiblichen Libido
US20090117183A1 (en) * 2007-11-05 2009-05-07 Sabine Fricke Oral contraceptive containing a gestagen and an estrogen combined with pharmaceutically acceptable auxiliary agents and/or excipients, but not containing lactose, and method of making same
WO2012155091A1 (en) * 2011-05-11 2012-11-15 Kirax Corporation Package for improved treatment of conditions

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DE2431704A1 (de) 1974-07-02 1976-01-22 Asche Ag Stufenkombinationspraeparate per kontrazeption
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DE102004019743B4 (de) 2004-04-20 2008-11-27 Bayer Schering Pharma Aktiengesellschaft Mehrphasenpräparat zur Kontrazeption auf der Basis eines natürlichen Estrogens
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ATE424828T1 (de) 2005-10-13 2009-03-15 Bayer Schering Pharma Ag Verwendung von estradiolvalerat in kombination mit dienogest zur oralen therapie der dysfunktionellen uterinen blutung in einheit mit einer oralen kontrazeption
US8153616B2 (en) 2005-10-17 2012-04-10 Bayer Pharma Aktiengesellschaft Combination preparation for oral contraception and oral therapy of dysfunctional uterine bleeding containing estradiol valerate and dienogest and method of using same
EP1930010A1 (de) 2006-10-20 2008-06-11 Bayer Schering Pharma Aktiengesellschaft Verwendung von Estradiolvalerat oder 17ß-Estradiol in Kombination mit Dienogest zur oralen Therapie für den Erhalt und/oder die Steigerung der weiblichen Libido

Also Published As

Publication number Publication date
SI1740163T1 (sl) 2010-11-30
WO2005102247A3 (de) 2006-01-12
GT200500093A (es) 2006-04-17
PL1740163T5 (pl) 2020-10-05
DE102004019743B4 (de) 2008-11-27
US20100173877A1 (en) 2010-07-08
JP4908399B2 (ja) 2012-04-04
CN1946383B (zh) 2010-06-09
RS51434B2 (sr) 2020-11-30
ES2348038T5 (es) 2020-09-14
ATE473734T1 (de) 2010-07-15
TW200534860A (en) 2005-11-01
ECSP067000A (es) 2006-12-29
EA200601844A1 (ru) 2007-04-27
CY1111292T1 (el) 2015-08-05
DK1740163T4 (da) 2020-04-06
PE20060308A1 (es) 2006-05-25
EP1740163B2 (de) 2020-01-15
HRP20100513T1 (en) 2010-11-30
AU2005235418A1 (en) 2005-11-03
AU2005235418C1 (en) 2015-05-21
KR20060134168A (ko) 2006-12-27
IL178510A0 (en) 2007-02-11
US20110124612A1 (en) 2011-05-26
AR048830A1 (es) 2006-05-31
ZA200609594B (en) 2008-04-30
EP1740163B1 (de) 2010-07-14
AR084229A2 (es) 2013-05-02
ME01183B (me) 2013-03-20
DE102004019743A1 (de) 2005-11-24
DE502005009904D1 (de) 2010-08-26
US20070259840A1 (en) 2007-11-08
UY28863A1 (es) 2005-11-30
HK1099701A1 (en) 2007-08-24
UA83915C2 (ru) 2008-08-26
US8071577B2 (en) 2011-12-06
SI1740163T2 (sl) 2020-04-30
MY143669A (en) 2011-06-30
AU2005235418B2 (en) 2009-08-06
CN1946383A (zh) 2007-04-11
DK1740163T3 (da) 2010-10-18
TWI351960B (en) 2011-11-11
IL178510A (en) 2015-08-31
SV2006002090A (es) 2006-02-15
PT1740163E (pt) 2010-09-28
NO20065292L (no) 2007-01-17
ES2348038T3 (es) 2010-11-29
RS51434B (en) 2011-04-30
WO2005102247A2 (de) 2005-11-03
HRP20100513T4 (hr) 2020-10-02
CA2561839C (en) 2009-09-29
PL1740163T3 (pl) 2010-12-31
NO344098B1 (no) 2019-09-02
JP2007533681A (ja) 2007-11-22
IL239861A0 (en) 2015-08-31
EP1740163A2 (de) 2007-01-10
MXPA06012213A (es) 2007-01-17
NZ550417A (en) 2010-01-29
CR8695A (es) 2008-07-29
EA010313B1 (ru) 2008-08-29
PA8630901A1 (es) 2006-05-16
CA2561839A1 (en) 2005-11-03

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B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
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