BRPI0414471A - nova formulação farmacêutica contendo biguanida e um derivado de tiazolidinadiona - Google Patents

nova formulação farmacêutica contendo biguanida e um derivado de tiazolidinadiona

Info

Publication number
BRPI0414471A
BRPI0414471A BRPI0414471-6A BRPI0414471A BRPI0414471A BR PI0414471 A BRPI0414471 A BR PI0414471A BR PI0414471 A BRPI0414471 A BR PI0414471A BR PI0414471 A BRPI0414471 A BR PI0414471A
Authority
BR
Brazil
Prior art keywords
formulation containing
pharmaceutical formulation
new pharmaceutical
thiazolidinedione derivative
containing biguanide
Prior art date
Application number
BRPI0414471-6A
Other languages
English (en)
Inventor
Unchalee Kositprapa
Robert I Goldfarb
John Cardinal
Avinash Nangia
Original Assignee
Andrx Labs Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34520446&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0414471(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Andrx Labs Llc filed Critical Andrx Labs Llc
Publication of BRPI0414471A publication Critical patent/BRPI0414471A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/155Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0004Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/282Organic compounds, e.g. fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

"NOVA FORMULAçãO FARMACêUTICA CONTENDO BIGUANIDA E UM DERIVADO DE TIAZOLIDINADIONA". Uma forma de dosagem farmacêutica compreendendo um componente de liberação controlada compreendendo uma droga antihiperglicêmica em combinação com um segundo componente compreendendo um derivado de tiazolidinadiona é aqui divulgada e descrita.
BRPI0414471-6A 2003-09-19 2004-02-12 nova formulação farmacêutica contendo biguanida e um derivado de tiazolidinadiona BRPI0414471A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10/664,803 US7785627B2 (en) 2002-09-20 2003-09-19 Pharmaceutical formulation containing a biguanide and a thiazolidinedione derivative
PCT/US2004/004112 WO2005039540A1 (en) 2003-09-19 2004-02-12 Novel pharmaceutical formulation containing a biguanide and a thiazolidinedione derivative

Publications (1)

Publication Number Publication Date
BRPI0414471A true BRPI0414471A (pt) 2006-11-14

Family

ID=34520446

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0414471-6A BRPI0414471A (pt) 2003-09-19 2004-02-12 nova formulação farmacêutica contendo biguanida e um derivado de tiazolidinadiona

Country Status (11)

Country Link
US (2) US7785627B2 (pt)
EP (1) EP1663170B1 (pt)
JP (3) JP4718465B2 (pt)
KR (2) KR101249171B1 (pt)
CN (2) CN1852703A (pt)
AU (2) AU2004283059B2 (pt)
BR (1) BRPI0414471A (pt)
CA (1) CA2537665C (pt)
ES (1) ES2541124T3 (pt)
NZ (2) NZ545653A (pt)
WO (1) WO2005039540A1 (pt)

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US9060941B2 (en) * 2002-09-20 2015-06-23 Actavis, Inc. Pharmaceutical formulation containing a biguanide and a thiazolidinedione derivative
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KR20140007247A (ko) * 2010-06-22 2014-01-17 티더블유아이 파머수티컬스, 인코포레이티드 음식물 영향이 감소된 제어 방출 조성물
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KR20130136718A (ko) * 2012-06-05 2013-12-13 한미약품 주식회사 메트포르민 서방성 장용제제 및 이의 제조방법
JPWO2014171542A1 (ja) * 2013-04-19 2017-02-23 武田薬品工業株式会社 放出制御製剤
CN104473894A (zh) * 2014-12-18 2015-04-01 浙江华海药业股份有限公司 一种盐酸吡格列酮载药包衣制剂及其制备方法
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AU2011202162B2 (en) 2013-11-21
NZ545653A (en) 2009-12-24
JP5881962B2 (ja) 2016-03-09
EP1663170A1 (en) 2006-06-07
AU2011202162A1 (en) 2011-06-02
CN101675929A (zh) 2010-03-24
JP2007505903A (ja) 2007-03-15
US7785627B2 (en) 2010-08-31
JP6054909B2 (ja) 2016-12-27
KR20060076299A (ko) 2006-07-04
EP1663170B1 (en) 2015-06-24
KR20110126761A (ko) 2011-11-23
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