BR9912138A - Compostos cìclicos úteis no tratamento de dislipidemia, aterosclerose e diabetes, composções farmacêuticas e processo para preparação - Google Patents
Compostos cìclicos úteis no tratamento de dislipidemia, aterosclerose e diabetes, composções farmacêuticas e processo para preparaçãoInfo
- Publication number
- BR9912138A BR9912138A BR9912138-7A BR9912138A BR9912138A BR 9912138 A BR9912138 A BR 9912138A BR 9912138 A BR9912138 A BR 9912138A BR 9912138 A BR9912138 A BR 9912138A
- Authority
- BR
- Brazil
- Prior art keywords
- dyslipidemia
- diabetes
- preparation
- treatment
- atherosclerosis
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D319/04—1,3-Dioxanes; Hydrogenated 1,3-dioxanes
- C07D319/08—1,3-Dioxanes; Hydrogenated 1,3-dioxanes condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D319/04—1,3-Dioxanes; Hydrogenated 1,3-dioxanes
- C07D319/06—1,3-Dioxanes; Hydrogenated 1,3-dioxanes not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
- C07D407/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Emergency Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Steroid Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
- Pyrane Compounds (AREA)
Abstract
Patente de Invenção: <B>"COMPOSTOS CìCLICOS úTEIS NO TRATAMENTO DE DISLIPIDEMIA, ATEROSCLEROSE E DIABETES, COMPOSIçõES FARMACêUTICAS E PROCESSO PARA PREPARAçãO"<D>. A presente invenção refere-se a compostos cíclicos que podem ser usados no tratamento de dislipidemia, aterosclerose e diabetes, a processos para a preparação destes compostos. Os compostos da invenção correspondem a fórmula I em que os radicais X, Y, R, R~ 1~, R~ 2~, R~ 3~, R~ 4~, R~ 5~, R~ 6~, R~ 7~ têm os significados dados na reivindicação 1.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9809164A FR2781222A1 (fr) | 1998-07-17 | 1998-07-17 | Composes cycliques utilisables dans le traitement de dyslipidemies, de l'atherosclerose et du diabete, compositions pharmaceutiques les contenant et procede de preparation |
PCT/EP1999/004831 WO2000004011A1 (en) | 1998-07-17 | 1999-07-09 | Cyclic compounds useful in the treatment of dyslipidaemia, atherosclerosis and diabetes, pharmaceutical compositions and preparation process |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9912138A true BR9912138A (pt) | 2001-04-10 |
Family
ID=9528730
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9912138-7A BR9912138A (pt) | 1998-07-17 | 1999-07-09 | Compostos cìclicos úteis no tratamento de dislipidemia, aterosclerose e diabetes, composções farmacêuticas e processo para preparação |
Country Status (22)
Country | Link |
---|---|
US (1) | US6528538B1 (pt) |
EP (1) | EP1098893B1 (pt) |
JP (1) | JP2002520407A (pt) |
KR (1) | KR20010070966A (pt) |
CN (1) | CN1309655A (pt) |
AT (1) | ATE235485T1 (pt) |
AU (1) | AU753287B2 (pt) |
BR (1) | BR9912138A (pt) |
CA (1) | CA2337481A1 (pt) |
DE (1) | DE69906303T2 (pt) |
DK (1) | DK1098893T3 (pt) |
ES (1) | ES2192853T3 (pt) |
FR (1) | FR2781222A1 (pt) |
HK (1) | HK1039615A1 (pt) |
HU (1) | HUP0103411A3 (pt) |
ID (1) | ID27854A (pt) |
NO (1) | NO20010266D0 (pt) |
PL (1) | PL345397A1 (pt) |
PT (1) | PT1098893E (pt) |
SK (1) | SK482001A3 (pt) |
WO (1) | WO2000004011A1 (pt) |
ZA (1) | ZA200101303B (pt) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TWI311133B (en) | 2001-04-20 | 2009-06-21 | Eisai R&D Man Co Ltd | Carboxylic acid derivativeand the salt thereof |
JPWO2003016265A1 (ja) * | 2001-08-17 | 2004-12-02 | エーザイ株式会社 | 環状化合物およびpparアゴニスト |
PT1622569E (pt) | 2003-04-24 | 2016-03-03 | Incyte Corp | Derivados de aza espiro alcanos como inibidores de metaloproteases |
OA13359A (en) * | 2004-01-09 | 2007-04-13 | Cadila Healthcare Ltd | 1,3-dioxane derivatives and analogues thereof useful in the treatment of i.a. obesity and diabetes. |
CA2577668A1 (en) * | 2004-08-20 | 2006-02-23 | Cadila Healthcare Limited | Novel antidiabetic compounds |
CN100389112C (zh) * | 2004-12-16 | 2008-05-21 | 中国石油化工股份有限公司 | 一类环状缩醛和缩酮化合物及其应用 |
ES2327187T3 (es) * | 2006-02-27 | 2009-10-26 | Cadila Healthcare Limited | Acidos 1,3-dioxano carboxilicos. |
AU2007253929B2 (en) * | 2006-05-18 | 2011-07-21 | Wellstat Therapeutics Corporation | Compounds for the treatment of metabolic disorders |
US7910108B2 (en) * | 2006-06-05 | 2011-03-22 | Incyte Corporation | Sheddase inhibitors combined with CD30-binding immunotherapeutics for the treatment of CD30 positive diseases |
WO2016056031A1 (en) | 2014-10-08 | 2016-04-14 | Council Of Scientific & Industrial Research | Novel diol compounds synthesis and its use for formal synthesis of (2r, 3 s)-3-hydroxypipecolic acid |
US9637575B2 (en) * | 2014-12-31 | 2017-05-02 | W. R. Grace & Co. -Conn. | Catalyst system, olefin polymerization catalyst components comprising at least an internal electron donor compound, and methods of making and using the same |
US20230050418A1 (en) * | 2019-12-13 | 2023-02-16 | Rhodia Operations | Production of benzene derivatives |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4032536A (en) * | 1976-07-22 | 1977-06-28 | Janssen Pharmaceutica N.V. | (1h-benzimidazol-2-yl)carbamates |
US5179216A (en) * | 1990-08-16 | 1993-01-12 | American Home Products Corporation | N,n', n'-trisubstituted-5-bisaminomethylene-1,3-dioxane-4,6-dione inhibitors of acyl-coa:cholesterol-acyl transferase |
TW209868B (pt) * | 1991-04-04 | 1993-07-21 | Yoshitomi Pharmaceutical | |
DE19637840A1 (de) * | 1996-09-17 | 1998-03-19 | Henkel Kgaa | Verwendung von geminalen Dialkoxyalkansäureestern zur Herstellung von desodorierenden Körperpflegemitteln |
-
1998
- 1998-07-17 FR FR9809164A patent/FR2781222A1/fr not_active Withdrawn
-
1999
- 1999-07-09 WO PCT/EP1999/004831 patent/WO2000004011A1/en not_active Application Discontinuation
- 1999-07-09 ES ES99934643T patent/ES2192853T3/es not_active Expired - Lifetime
- 1999-07-09 ID IDW20010261A patent/ID27854A/id unknown
- 1999-07-09 CA CA002337481A patent/CA2337481A1/en not_active Abandoned
- 1999-07-09 PL PL99345397A patent/PL345397A1/xx unknown
- 1999-07-09 EP EP99934643A patent/EP1098893B1/en not_active Expired - Lifetime
- 1999-07-09 DE DE69906303T patent/DE69906303T2/de not_active Expired - Fee Related
- 1999-07-09 BR BR9912138-7A patent/BR9912138A/pt not_active IP Right Cessation
- 1999-07-09 AU AU50347/99A patent/AU753287B2/en not_active Ceased
- 1999-07-09 US US09/743,759 patent/US6528538B1/en not_active Expired - Fee Related
- 1999-07-09 HU HU0103411A patent/HUP0103411A3/hu unknown
- 1999-07-09 JP JP2000560117A patent/JP2002520407A/ja active Pending
- 1999-07-09 DK DK99934643T patent/DK1098893T3/da active
- 1999-07-09 KR KR1020017000647A patent/KR20010070966A/ko not_active Application Discontinuation
- 1999-07-09 CN CN99808783A patent/CN1309655A/zh active Pending
- 1999-07-09 PT PT99934643T patent/PT1098893E/pt unknown
- 1999-07-09 AT AT99934643T patent/ATE235485T1/de not_active IP Right Cessation
- 1999-07-09 SK SK48-2001A patent/SK482001A3/sk unknown
-
2001
- 2001-01-16 NO NO20010266A patent/NO20010266D0/no not_active Application Discontinuation
- 2001-02-15 ZA ZA200101303A patent/ZA200101303B/en unknown
-
2002
- 2002-02-07 HK HK02100966.8A patent/HK1039615A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
AU5034799A (en) | 2000-02-07 |
DE69906303D1 (de) | 2003-04-30 |
ATE235485T1 (de) | 2003-04-15 |
SK482001A3 (en) | 2001-09-11 |
CN1309655A (zh) | 2001-08-22 |
NO20010266L (no) | 2001-01-16 |
HUP0103411A2 (hu) | 2002-04-29 |
NO20010266D0 (no) | 2001-01-16 |
EP1098893B1 (en) | 2003-03-26 |
KR20010070966A (ko) | 2001-07-28 |
PT1098893E (pt) | 2003-08-29 |
AU753287B2 (en) | 2002-10-17 |
ID27854A (id) | 2001-04-26 |
HK1039615A1 (zh) | 2002-05-03 |
ES2192853T3 (es) | 2003-10-16 |
PL345397A1 (en) | 2001-12-17 |
DE69906303T2 (de) | 2003-12-11 |
CA2337481A1 (en) | 2000-01-27 |
JP2002520407A (ja) | 2002-07-09 |
FR2781222A1 (fr) | 2000-01-21 |
US6528538B1 (en) | 2003-03-04 |
WO2000004011A1 (en) | 2000-01-27 |
ZA200101303B (en) | 2002-05-15 |
HUP0103411A3 (en) | 2002-08-28 |
EP1098893A1 (en) | 2001-05-16 |
DK1098893T3 (da) | 2003-07-07 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 6A, 7A E 8A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1911 DE 21/08/2007. |