BR9811054A - Derivado do grupo a das estreptograminas, processo para preparação de um derivado de estreptogramina, associações , e, composição farmacêutica - Google Patents
Derivado do grupo a das estreptograminas, processo para preparação de um derivado de estreptogramina, associações , e, composição farmacêuticaInfo
- Publication number
- BR9811054A BR9811054A BR9811054-3A BR9811054A BR9811054A BR 9811054 A BR9811054 A BR 9811054A BR 9811054 A BR9811054 A BR 9811054A BR 9811054 A BR9811054 A BR 9811054A
- Authority
- BR
- Brazil
- Prior art keywords
- radical
- group
- derivative
- streptogramin
- alcoholic
- Prior art date
Links
- 108010034396 Streptogramins Proteins 0.000 title abstract 4
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 108010063483 Streptogramin Group A Proteins 0.000 title 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 4
- 230000001476 alcoholic effect Effects 0.000 abstract 3
- -1 ally Chemical group 0.000 abstract 3
- 150000003254 radicals Chemical class 0.000 abstract 3
- 125000004432 carbon atom Chemical group C* 0.000 abstract 2
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 2
- WCYWZMWISLQXQU-UHFFFAOYSA-N methyl Chemical compound [CH3] WCYWZMWISLQXQU-UHFFFAOYSA-N 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 229910052757 nitrogen Inorganic materials 0.000 abstract 2
- 125000002568 propynyl group Chemical group [*]C#CC([H])([H])[H] 0.000 abstract 2
- 229940041030 streptogramins Drugs 0.000 abstract 2
- SLRMQYXOBQWXCR-UHFFFAOYSA-N 2154-56-5 Chemical compound [CH2]C1=CC=CC=C1 SLRMQYXOBQWXCR-UHFFFAOYSA-N 0.000 abstract 1
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 1
- 239000004599 antimicrobial Substances 0.000 abstract 1
- 125000004429 atom Chemical group 0.000 abstract 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- 239000000470 constituent Substances 0.000 abstract 1
- QUPDWYMUPZLYJZ-UHFFFAOYSA-N ethyl Chemical compound C[CH2] QUPDWYMUPZLYJZ-UHFFFAOYSA-N 0.000 abstract 1
- 125000005842 heteroatom Chemical group 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
- IJGRMHOSHXDMSA-UHFFFAOYSA-N nitrogen Substances N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 239000001301 oxygen Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 229920006395 saturated elastomer Polymers 0.000 abstract 1
- 229910052717 sulfur Chemical group 0.000 abstract 1
- 239000011593 sulfur Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
- C07K5/06182—Dipeptides with the first amino acid being heterocyclic and Pristinamycin II; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Oncology (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Veterinary Medicine (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9709557A FR2766489B1 (fr) | 1997-07-28 | 1997-07-28 | Derives de streptogramines, leur preparation et les compositions qui les contiennent |
PCT/FR1998/001639 WO1999005165A1 (fr) | 1997-07-28 | 1998-07-24 | Derives de streptogramines, leur preparation et les compositions qui les contiennent |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9811054A true BR9811054A (pt) | 2000-09-05 |
Family
ID=9509695
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9811054-3A BR9811054A (pt) | 1997-07-28 | 1998-07-24 | Derivado do grupo a das estreptograminas, processo para preparação de um derivado de estreptogramina, associações , e, composição farmacêutica |
Country Status (22)
Country | Link |
---|---|
US (1) | US6815437B1 (es) |
EP (1) | EP0989994B1 (es) |
JP (1) | JP4557419B2 (es) |
KR (1) | KR20010022295A (es) |
CN (1) | CN1265115A (es) |
AT (1) | ATE293635T1 (es) |
AU (1) | AU8867798A (es) |
BR (1) | BR9811054A (es) |
CA (1) | CA2299514A1 (es) |
DE (1) | DE69829849T2 (es) |
DK (1) | DK0989994T3 (es) |
EA (1) | EA200000170A1 (es) |
ES (1) | ES2241158T3 (es) |
FR (1) | FR2766489B1 (es) |
HU (1) | HUP0002827A2 (es) |
IL (1) | IL134194A0 (es) |
NO (1) | NO20000424D0 (es) |
PL (1) | PL338294A1 (es) |
PT (1) | PT989994E (es) |
SK (1) | SK1152000A3 (es) |
WO (1) | WO1999005165A1 (es) |
ZA (1) | ZA986730B (es) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2795733B1 (fr) * | 1999-06-30 | 2001-09-07 | Aventis Pharma Sa | Derives de streptogramines, leur preparation et les compositions qui les contiennent |
FR2818644B1 (fr) * | 2000-12-21 | 2004-10-22 | Aventis Pharma Sa | Derives de streptogramines, leur preparation et les compositions qui les contiennent |
US6562852B2 (en) | 2000-12-21 | 2003-05-13 | Aventis Pharma S.A. | Streptogramin derivatives, their preparation and compositions which contain them |
FR2818645B1 (fr) * | 2000-12-21 | 2003-01-31 | Aventis Pharma Sa | Derives de streptogramines, leur preparation et les compositions qui les contiennent |
AU2018308972A1 (en) * | 2017-08-01 | 2020-02-06 | The Regents Of The University Of California | Methods of making streptogramin compositions and the use thereof |
CA3180078A1 (en) | 2020-05-27 | 2021-12-02 | Universita Degli Studi Di Trento | New therapy for the treatment of tumors |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2549065B1 (fr) * | 1983-07-13 | 1985-10-25 | Rhone Poulenc Sante | Nouveaux derives de synergistines, leur preparation et les compositions pharmaceutiques qui les contiennent |
FR2576022B1 (fr) | 1985-01-11 | 1987-09-11 | Rhone Poulenc Sante | Nouveaux derives de la pristinamycine ii b, leur preparation et les compositions pharmaceutiques qui les contiennent |
FR2599036B1 (fr) | 1986-05-22 | 1988-09-09 | Rhone Poulenc Sante | Nouveaux derives de synergistines, leur preparation et les compositions pharmaceutiques qui les contiennent |
GB8616768D0 (en) | 1986-07-09 | 1986-08-13 | May & Baker Ltd | Process |
GB2206879A (en) * | 1987-07-07 | 1989-01-18 | May & Baker Ltd | Novel pristinamycin IIB derivatives, their preparation and pharmaceutical compositions containing them |
FR2664600B1 (fr) | 1990-07-16 | 1994-09-02 | Rhone Poulenc Sante | Nouveau sel derive de la dialcoylaminoalcoyl-sulfonyl-26 pristinamycine iib. |
FR2696189B1 (fr) | 1992-09-25 | 1994-11-10 | Rhone Poulenc Rorer Sa | Polypeptides impliqués dans la biosynthèse des streptogramines, séquences nucléotidiques codant pour ces polypeptides et leur utilisation. |
IL121821A (en) | 1993-02-17 | 2000-02-17 | Rhone Poulenc Rorer Sa | Process for purifying a group A minority component of streptogramin some such purified components and their uses |
-
1997
- 1997-07-28 FR FR9709557A patent/FR2766489B1/fr not_active Expired - Fee Related
-
1998
- 1998-07-24 BR BR9811054-3A patent/BR9811054A/pt not_active Application Discontinuation
- 1998-07-24 AT AT98940328T patent/ATE293635T1/de active
- 1998-07-24 DK DK98940328T patent/DK0989994T3/da active
- 1998-07-24 SK SK115-2000A patent/SK1152000A3/sk unknown
- 1998-07-24 EP EP98940328A patent/EP0989994B1/fr not_active Expired - Lifetime
- 1998-07-24 KR KR1020007000874A patent/KR20010022295A/ko not_active Application Discontinuation
- 1998-07-24 HU HU0002827A patent/HUP0002827A2/hu unknown
- 1998-07-24 PT PT98940328T patent/PT989994E/pt unknown
- 1998-07-24 ES ES98940328T patent/ES2241158T3/es not_active Expired - Lifetime
- 1998-07-24 CN CN98807630A patent/CN1265115A/zh active Pending
- 1998-07-24 IL IL13419498A patent/IL134194A0/xx unknown
- 1998-07-24 JP JP2000504158A patent/JP4557419B2/ja not_active Expired - Fee Related
- 1998-07-24 AU AU88677/98A patent/AU8867798A/en not_active Abandoned
- 1998-07-24 PL PL98338294A patent/PL338294A1/xx unknown
- 1998-07-24 CA CA002299514A patent/CA2299514A1/fr not_active Abandoned
- 1998-07-24 EA EA200000170A patent/EA200000170A1/ru unknown
- 1998-07-24 WO PCT/FR1998/001639 patent/WO1999005165A1/fr active IP Right Grant
- 1998-07-24 DE DE69829849T patent/DE69829849T2/de not_active Expired - Lifetime
- 1998-07-28 ZA ZA986730A patent/ZA986730B/xx unknown
-
2000
- 2000-01-27 US US09/492,392 patent/US6815437B1/en not_active Expired - Fee Related
- 2000-01-27 NO NO20000424A patent/NO20000424D0/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
PT989994E (pt) | 2005-08-31 |
EA200000170A1 (ru) | 2000-10-30 |
PL338294A1 (en) | 2000-10-23 |
KR20010022295A (ko) | 2001-03-15 |
CA2299514A1 (fr) | 1999-02-04 |
CN1265115A (zh) | 2000-08-30 |
WO1999005165A1 (fr) | 1999-02-04 |
NO20000424L (no) | 2000-01-27 |
DE69829849T2 (de) | 2006-02-23 |
NO20000424D0 (no) | 2000-01-27 |
DE69829849D1 (de) | 2005-05-25 |
ES2241158T3 (es) | 2005-10-16 |
IL134194A0 (en) | 2001-04-30 |
SK1152000A3 (en) | 2000-09-12 |
AU8867798A (en) | 1999-02-16 |
ATE293635T1 (de) | 2005-05-15 |
JP2001510849A (ja) | 2001-08-07 |
US6815437B1 (en) | 2004-11-09 |
ZA986730B (en) | 1999-02-02 |
WO1999005165A8 (fr) | 1999-04-29 |
FR2766489B1 (fr) | 1999-08-27 |
JP4557419B2 (ja) | 2010-10-06 |
DK0989994T3 (da) | 2005-08-22 |
EP0989994A1 (fr) | 2000-04-05 |
EP0989994B1 (fr) | 2005-04-20 |
FR2766489A1 (fr) | 1999-01-29 |
HUP0002827A2 (hu) | 2001-01-29 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
KR900007837A (ko) | 퀴누클리딘, 약제로서 이의 용도 및 이의 제조방법 | |
BR9914451A (pt) | Composto de oxazol, processo para sua preparação, composição farmacêutica compreendendo dito composto, uso da composição e métodos de tratamento | |
BRPI9810555A8 (pt) | Derivados epotilona | |
CO4340731A1 (es) | Una combinacion farmaceutica de fluoxetina, venlafaxina, milnacipran o duloxetina, y un componente de alprenolol, way 100135, espiperona, pindolol, (s)-uh-301, penbutolol, pro- pranolol, tertatolol, y una ariloxipropanolamina | |
BRPI0409928A8 (pt) | compostos, enantiômeros, composição farmacêutica, uso de compostos, processo para a fabricação de compostos, e, modificação dos processos | |
BR9811054A (pt) | Derivado do grupo a das estreptograminas, processo para preparação de um derivado de estreptogramina, associações , e, composição farmacêutica | |
NO148672C (no) | Fremgangsmaate til kontinuerlig fremstilling av epoksyderte lavmolekylaere alkener eller deres derivater, hvor alkenkomponenten omsettes med pereddiksyre eller perpropionsyre | |
ATE14439T1 (de) | Veraenderte d-retro cyclische hexapeptide, analoge von somatostatin, verfahren zu deren herstellung und diese enthaltende pharmazeutische zusammensetzungen. | |
KR960010635A (ko) | 약제학적 화합물 | |
KR920021517A (ko) | 중축 신경계에 활성인 신규의 3-아미노피리다진 유도체, 그의 제조방법 및 이들의 존재하는 약제학적 조성물 | |
GT198301599A (es) | 4"-epi-eritromicina a y sus derivados como utiles agentes antibacterianos. | |
BR9713159A (pt) | Composição substancialmente sólida, composto, composição de sal substancialmente sólida, mistura, e, processo para preparar um composto | |
KR900018027A (ko) | 피페리딘 유도체, 그의 제조 방법, 및 그것을 유효성분으로 함유하는 의약용 조성물 | |
BR9908195A (pt) | Derivado do grupo b das estreptograminas, processo para a preparação do mesmo, composições farmacêuticas, e, associações de derivados de estreptograminas. | |
KR920018036A (ko) | 티아졸리디논 및 옥사졸리디논 유도체, 그의 제조방법 및 혈관확장제로서의 용도 | |
KR900700098A (ko) | 발기부전의 치료겸 진단용 플라복세이트 및 그 유도체 | |
ATE3149T1 (de) | Isatinderivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zusammensetzungen. | |
FR2449677B1 (fr) | Nouveaux derives de benzoyl-2 glycylanilides substitues, leur preparation et leur application en tant que medicaments anxiolytiques | |
KR900003142A (ko) | 환형 황을 함유하는 화합물 | |
BRPI0606201A2 (pt) | composto rigidificado para modulação da atividade de heparanase e composição farmacêutica | |
Schwartz | Studies on mechanisms of calcium channel modulators | |
ES2078911T3 (es) | Fenil-heterociclos disustituidos en 3,4 y su utilizacion. | |
DK159112C (da) | Analogifremgangsmaade til fremstilling af n-(1,3-dithiolan-2-yliden)aniliner eller farmaceutisk acceptable syreadditionssalte deraf | |
DE69009604D1 (de) | 2-Alkyliminobenzothiazoline, ihre Herstellung und sie enthaltende Arzneimittel. | |
DK19885A (da) | 3-alkoxy-2-(n-pyrrolidino)-n-pyridyl-n-furyl (eller thienyl)-methyl-propylaminer, fremgangsmaade til fremstilling deraf, samt farmaceutiske midler indeholdende disse |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA10 | Dismissal: dismissal - article 33 of industrial property law | ||
B11Y | Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette] |