BR9908195A - Derivado do grupo b das estreptograminas, processo para a preparação do mesmo, composições farmacêuticas, e, associações de derivados de estreptograminas. - Google Patents

Derivado do grupo b das estreptograminas, processo para a preparação do mesmo, composições farmacêuticas, e, associações de derivados de estreptograminas.

Info

Publication number
BR9908195A
BR9908195A BR9908195-4A BR9908195A BR9908195A BR 9908195 A BR9908195 A BR 9908195A BR 9908195 A BR9908195 A BR 9908195A BR 9908195 A BR9908195 A BR 9908195A
Authority
BR
Brazil
Prior art keywords
group
streptogramins
associations
derived
pharmaceutical compositions
Prior art date
Application number
BR9908195-4A
Other languages
English (en)
Inventor
Pascal Desmazeau
Gilles Doerflinger
Yves Ribeill
Eric Bacque
Jean-Claude Barriere
Gilles Dutruc-Rosset
Gerard Puchault
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of BR9908195A publication Critical patent/BR9908195A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/06Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Veterinary Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

"DERIVADO DO GRUPO B DAS ESTREPTOGRAMINAS, PROCESSO PARA A PREPARAçãO DO MESMO, COMPOSIçõES FARMACêUTICAS, E, ASSOCIAçõES DE DERIVADOS DE ESTREPTOGRAMINAS". Derivados de grupo B das estreptograminas de fórmulas gerais (I): em que Ra, Rb, Rc, Rd, R1, R2 e Y são definidos como descrito na descrição. Estes derivados são particularmente interessantes como agentes antimicrobianos, eventualmente associados a pelo menos um derivado de estreptogramina do grupo A.
BR9908195-4A 1998-02-26 1999-02-24 Derivado do grupo b das estreptograminas, processo para a preparação do mesmo, composições farmacêuticas, e, associações de derivados de estreptograminas. BR9908195A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9802316A FR2775288B1 (fr) 1998-02-26 1998-02-26 Derives de streptogramines, leur preparation et les compositons qui les contiennent
PCT/FR1999/000409 WO1999043699A1 (fr) 1998-02-26 1999-02-24 Derives de streptogramines, leur preparation et les compositions qui les contiennent

Publications (1)

Publication Number Publication Date
BR9908195A true BR9908195A (pt) 2000-10-24

Family

ID=9523382

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9908195-4A BR9908195A (pt) 1998-02-26 1999-02-24 Derivado do grupo b das estreptograminas, processo para a preparação do mesmo, composições farmacêuticas, e, associações de derivados de estreptograminas.

Country Status (23)

Country Link
US (2) US6958383B2 (pt)
EP (1) EP1056771B1 (pt)
JP (1) JP4644366B2 (pt)
KR (1) KR20010041325A (pt)
CN (1) CN1290270A (pt)
AT (1) ATE311403T1 (pt)
AU (1) AU2628399A (pt)
BR (1) BR9908195A (pt)
CA (1) CA2321114A1 (pt)
DE (1) DE69928646T2 (pt)
DK (1) DK1056771T3 (pt)
EA (1) EA200000884A1 (pt)
ES (1) ES2252930T3 (pt)
FR (1) FR2775288B1 (pt)
HR (1) HRP20000452A2 (pt)
HU (1) HUP0101098A3 (pt)
IL (1) IL137794A0 (pt)
NO (1) NO20004273L (pt)
PL (1) PL342624A1 (pt)
SK (1) SK12842000A3 (pt)
TR (1) TR200002461T2 (pt)
WO (1) WO1999043699A1 (pt)
ZA (1) ZA991546B (pt)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE60006130D1 (de) * 1999-07-27 2003-11-27 Aventis Pharma Sa Streptograminderivate, ihre herstellung und sie enthaltende zubereitungen
FR2796949B1 (fr) * 1999-07-27 2001-09-21 Aventis Pharma Sa Derives de streptogramines, leur preparation et les compositions qui les contiennent
US7169756B2 (en) * 2004-04-16 2007-01-30 Mcmaster University Streptogramin antibiotics
DE102006007882A1 (de) 2006-02-21 2007-08-30 Bayer Cropscience Ag Cycloalkyl-phenylsubstituierte cyclische Ketoenole
ES2632567T3 (es) 2009-03-11 2017-09-14 Bayer Intellectual Property Gmbh Cetoenoles sustituidos con haloalquilmetilenoxi-fenilo
US8281596B1 (en) 2011-05-16 2012-10-09 General Electric Company Combustor assembly for a turbomachine
JP6042433B2 (ja) 2011-08-11 2016-12-14 バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Intellectual Property GmbH 1,2,4−トリアゾリル置換されたケトエノール類
US8899975B2 (en) 2011-11-04 2014-12-02 General Electric Company Combustor having wake air injection
US9267687B2 (en) 2011-11-04 2016-02-23 General Electric Company Combustion system having a venturi for reducing wakes in an airflow
US9322553B2 (en) 2013-05-08 2016-04-26 General Electric Company Wake manipulating structure for a turbine system
US9739201B2 (en) 2013-05-08 2017-08-22 General Electric Company Wake reducing structure for a turbine system and method of reducing wake
US9435221B2 (en) 2013-08-09 2016-09-06 General Electric Company Turbomachine airfoil positioning
WO2019152977A2 (en) 2018-02-05 2019-08-08 Bio-Rad Laboratories, Inc. Chromatography resin having an anionic exchange-hydrophobic mixed mode ligand

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2722210B1 (fr) * 1994-07-08 1996-08-14 Rhone Poulenc Rorer Sa Nouvelles streptogramines et procede de preparation de streptogramines par mutasynthese
FR2723372B1 (fr) * 1994-08-02 1996-10-04 Rhone Poulenc Rorer Sa Nouveaux derives de streptogramine, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2723373B1 (fr) * 1994-08-02 1996-09-13 Rhone Poulenc Rorer Sa Forme purifiee de streptogramines, sa preparation et les compositions pharmaceutiques qui la contiennent
FR2795733B1 (fr) 1999-06-30 2001-09-07 Aventis Pharma Sa Derives de streptogramines, leur preparation et les compositions qui les contiennent
FR2796949B1 (fr) 1999-07-27 2001-09-21 Aventis Pharma Sa Derives de streptogramines, leur preparation et les compositions qui les contiennent
DE60006130D1 (de) 1999-07-27 2003-11-27 Aventis Pharma Sa Streptograminderivate, ihre herstellung und sie enthaltende zubereitungen

Also Published As

Publication number Publication date
AU2628399A (en) 1999-09-15
ES2252930T3 (es) 2006-05-16
EA200000884A1 (ru) 2001-02-26
WO1999043699A1 (fr) 1999-09-02
KR20010041325A (ko) 2001-05-15
SK12842000A3 (sk) 2001-01-18
HRP20000452A2 (en) 2000-12-31
DE69928646T2 (de) 2006-08-10
IL137794A0 (en) 2001-10-31
ATE311403T1 (de) 2005-12-15
EP1056771A1 (fr) 2000-12-06
TR200002461T2 (tr) 2000-11-21
US7019110B2 (en) 2006-03-28
NO20004273L (no) 2000-10-23
HUP0101098A3 (en) 2001-12-28
US6958383B2 (en) 2005-10-25
PL342624A1 (en) 2001-06-18
DK1056771T3 (da) 2006-04-03
FR2775288A1 (fr) 1999-08-27
CA2321114A1 (fr) 1999-09-02
HUP0101098A1 (hu) 2001-08-28
US20040266667A1 (en) 2004-12-30
ZA991546B (en) 1999-08-25
JP4644366B2 (ja) 2011-03-02
DE69928646D1 (de) 2006-01-05
JP2002504560A (ja) 2002-02-12
FR2775288B1 (fr) 2000-03-31
US20020151676A1 (en) 2002-10-17
EP1056771B1 (fr) 2005-11-30
NO20004273D0 (no) 2000-08-25
CN1290270A (zh) 2001-04-04

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Legal Events

Date Code Title Description
FA10 Dismissal: dismissal - article 33 of industrial property law
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]