BR9713950A - Processo para produção de um composto, e composto. - Google Patents

Processo para produção de um composto, e composto.

Info

Publication number
BR9713950A
BR9713950A BR9713950A BR9713950A BR9713950A BR 9713950 A BR9713950 A BR 9713950A BR 9713950 A BR9713950 A BR 9713950A BR 9713950 A BR9713950 A BR 9713950A BR 9713950 A BR9713950 A BR 9713950A
Authority
BR
Brazil
Prior art keywords
compound
formula
alkyl
producing
independently
Prior art date
Application number
BR9713950A
Other languages
English (en)
Inventor
Alan Richard Harris
Original Assignee
Astra Pharma Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astra Pharma Prod filed Critical Astra Pharma Prod
Publication of BR9713950A publication Critical patent/BR9713950A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00Preparation of carboxylic acid amides
    • C07C231/02Preparation of carboxylic acid amides from carboxylic acids or from esters, anhydrides, or halides thereof by reaction with ammonia or amines
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

O". Esta invenção refere-se a um processo melhorad de fórmula (I): que são úteis como medicamentos, na qual R^ 1^ e R^ 2^ são independentemente selecigênio, C~ 1~-C~ 4~-alquila ou metóxi-carbonila; R^ 4^ é hidrogênio ou metila; que compreende a reação de um composto de fórmula (II): com um composto de fórmula (III): na qual R^ 5^, R^ 6^, R^ 7^, R^ 8^, R^ 9^ e R^ 10^ são independentemente C~ 1~-C~ 6~-alquila, seguida pela desproteção e opcionalmente depois pela formação de um sal farmaceuticamente aceitável.
BR9713950A 1996-12-19 1997-12-12 Processo para produção de um composto, e composto. BR9713950A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9626319.9A GB9626319D0 (en) 1996-12-19 1996-12-19 Synthetic method
PCT/SE1997/002092 WO1998027052A1 (en) 1996-12-19 1997-12-12 Process for the preparation of nmda antagonists

Publications (1)

Publication Number Publication Date
BR9713950A true BR9713950A (pt) 2000-03-21

Family

ID=10804657

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9713950A BR9713950A (pt) 1996-12-19 1997-12-12 Processo para produção de um composto, e composto.

Country Status (33)

Country Link
US (1) US6063962A (pt)
EP (1) EP0946497B1 (pt)
JP (1) JP2002512595A (pt)
KR (1) KR100522337B1 (pt)
CN (1) CN1105098C (pt)
AR (1) AR010366A1 (pt)
AT (1) ATE207053T1 (pt)
AU (1) AU725683B2 (pt)
BR (1) BR9713950A (pt)
CA (1) CA2273286A1 (pt)
CZ (1) CZ296780B6 (pt)
DE (1) DE69707503T2 (pt)
DK (1) DK0946497T3 (pt)
EE (1) EE03762B1 (pt)
EG (1) EG21486A (pt)
ES (1) ES2163806T3 (pt)
GB (1) GB9626319D0 (pt)
HU (1) HUP0000420A3 (pt)
ID (1) ID23994A (pt)
IL (1) IL130425A (pt)
IS (1) IS5059A (pt)
MY (1) MY115259A (pt)
NO (1) NO993065D0 (pt)
NZ (1) NZ335870A (pt)
PL (1) PL191196B1 (pt)
PT (1) PT946497E (pt)
RU (1) RU2190597C2 (pt)
SI (1) SI0946497T1 (pt)
SK (1) SK283033B6 (pt)
TR (1) TR199901394T2 (pt)
TW (1) TW415931B (pt)
WO (1) WO1998027052A1 (pt)
ZA (1) ZA9711057B (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100826497B1 (ko) 2007-01-22 2008-05-02 삼성전자주식회사 전력 소모를 줄이기 위한 반도체 메모리 장치의 입출력센스 앰프 회로

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE955508C (de) * 1954-07-28 1957-01-03 Cilag Ag Verfahren zur Herstellung von antikonvulsivisch wirkenden Carbonsaeureamiden
IL84305A (en) * 1987-02-06 1992-01-15 Fisons Corp 2-aminoacetamide derivatives

Also Published As

Publication number Publication date
GB9626319D0 (en) 1997-02-05
PL191196B1 (pl) 2006-03-31
KR20000069552A (ko) 2000-11-25
KR100522337B1 (ko) 2005-10-19
CZ219899A3 (cs) 1999-11-17
CA2273286A1 (en) 1998-06-25
EE03762B1 (et) 2002-06-17
CZ296780B6 (cs) 2006-06-14
NZ335870A (en) 2001-05-25
RU2190597C2 (ru) 2002-10-10
EP0946497A1 (en) 1999-10-06
ZA9711057B (en) 1998-06-19
NO993065L (no) 1999-06-21
ES2163806T3 (es) 2002-02-01
DK0946497T3 (da) 2001-12-17
MY115259A (en) 2003-04-30
AU5352498A (en) 1998-07-15
CN1105098C (zh) 2003-04-09
EE9900257A (et) 1999-12-15
CN1240420A (zh) 2000-01-05
TW415931B (en) 2000-12-21
IL130425A (en) 2003-02-12
AU725683B2 (en) 2000-10-19
HUP0000420A3 (en) 2000-09-28
EP0946497B1 (en) 2001-10-17
ID23994A (id) 2000-06-14
SI0946497T1 (en) 2002-06-30
DE69707503T2 (de) 2002-05-16
SK283033B6 (sk) 2003-02-04
US6063962A (en) 2000-05-16
NO993065D0 (no) 1999-06-21
PT946497E (pt) 2002-03-28
AR010366A1 (es) 2000-06-07
IL130425A0 (en) 2000-06-01
WO1998027052A1 (en) 1998-06-25
JP2002512595A (ja) 2002-04-23
ATE207053T1 (de) 2001-11-15
TR199901394T2 (xx) 1999-08-23
HUP0000420A2 (hu) 2000-08-28
DE69707503D1 (de) 2001-11-22
EG21486A (en) 2001-11-28
IS5059A (is) 1999-05-28
PL333919A1 (en) 2000-01-31
SK65699A3 (en) 1999-11-08

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Legal Events

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B11B Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements