BR6908381D0 - Novos derivados de piridil-oxadiasol e processo para a sua preparacao - Google Patents

Novos derivados de piridil-oxadiasol e processo para a sua preparacao

Info

Publication number
BR6908381D0
BR6908381D0 BR208381/69A BR20838169A BR6908381D0 BR 6908381 D0 BR6908381 D0 BR 6908381D0 BR 208381/69 A BR208381/69 A BR 208381/69A BR 20838169 A BR20838169 A BR 20838169A BR 6908381 D0 BR6908381 D0 BR 6908381D0
Authority
BR
Brazil
Prior art keywords
oxadiasol
pyridil
derivatives
preparation
new
Prior art date
Application number
BR208381/69A
Other languages
English (en)
Portuguese (pt)
Inventor
K Harsanvi
C Vertesy
G Leszkovszky
L Tardos
K Takacs
E Bako
J Rener
D Goenczi
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Publication of BR6908381D0 publication Critical patent/BR6908381D0/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/061,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
BR208381/69A 1968-04-26 1969-04-25 Novos derivados de piridil-oxadiasol e processo para a sua preparacao BR6908381D0 (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HUCI000796 1968-04-26

Publications (1)

Publication Number Publication Date
BR6908381D0 true BR6908381D0 (pt) 1973-02-08

Family

ID=10994349

Family Applications (1)

Application Number Title Priority Date Filing Date
BR208381/69A BR6908381D0 (pt) 1968-04-26 1969-04-25 Novos derivados de piridil-oxadiasol e processo para a sua preparacao

Country Status (15)

Country Link
US (1) US3647809A (https=)
JP (1) JPS4824394B1 (https=)
AT (2) AT292728B (https=)
BE (1) BE732131A (https=)
BR (1) BR6908381D0 (https=)
CA (1) CA954858A (https=)
CH (2) CH542232A (https=)
DE (1) DE1920037A1 (https=)
FR (1) FR2007529B1 (https=)
GB (1) GB1271302A (https=)
IL (1) IL31990A (https=)
NL (1) NL6906401A (https=)
NO (1) NO124253B (https=)
PL (1) PL79435B1 (https=)
SE (1) SE368576B (https=)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3853893A (en) * 1973-04-02 1974-12-10 Squibb & Sons Inc Anthelmintic 5-(pyridyl)-3-(isothiocyanophenyl) oxadiazoles
HU177086B (en) * 1975-06-09 1981-07-28 Eszakmagyar Vegyimuevek Herbicide and fungicide preparation containing substituted 1,2,4-oxadiazolidin-3-one derivatives
JPS58150576A (ja) * 1982-03-03 1983-09-07 Sumitomo Chem Co Ltd 新規な1,2,4−オキサジアゾ−ル誘導体
DE3247118A1 (de) * 1982-12-20 1984-06-20 Cassella Ag, 6000 Frankfurt Neue substituierte 1,4-dihydropyridine, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
KR100875222B1 (ko) * 1999-08-19 2008-12-19 아스트라제네카 아베 헤테로폴리사이클릭 화합물 및 간접 글루타메이트 수용체길항제로서의 그들의 용도
EP1582519A3 (en) * 1999-08-19 2005-12-21 Nps Pharmaceuticals, Inc. Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists
US6660753B2 (en) * 1999-08-19 2003-12-09 Nps Pharmaceuticals, Inc. Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists
MXPA03007513A (es) * 2001-02-21 2004-07-30 Nps Pharma Inc Compuestos heteropoliciclicos y su uso como antagonistas del receptor metabotropico de glutamato.
US7074809B2 (en) 2002-08-09 2006-07-11 Astrazeneca Ab Compounds
US8178570B2 (en) * 2003-04-09 2012-05-15 Exelixis, Inc. Tie-2 modulators and methods of use
AU2004240586A1 (en) * 2003-05-15 2004-12-02 Merck & Co., Inc. 3-(2-amino-1-azacyclyl)-5-aryl-1,2,4-oxadiazoles as S1P receptor agonists
US20060189661A1 (en) * 2003-11-03 2006-08-24 Wagenen Bradford V Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists
WO2005060961A2 (en) * 2003-12-18 2005-07-07 Astrazeneca Ab Treatment of transient lower esophageal sphincter relaxations (tlesrs) and gastro-esophageal reflux disease (gerd)
JP4958560B2 (ja) * 2003-12-24 2012-06-20 プロシディオン・リミテッド Gpcr受容体作動薬としてのヘテロ環誘導体
WO2005077368A2 (en) * 2004-02-03 2005-08-25 Astrazeneca Ab Treatment of gastro-esophageal reflux disease (gerd)
US8017631B2 (en) * 2005-04-26 2011-09-13 Neurosearch A/S Oxadiazole derivatives and their medical use
IL169855A (en) * 2005-07-25 2014-05-28 Elta Systems Ltd A system and method for locating a receiver location
PL1907382T3 (pl) 2005-07-26 2016-01-29 Bial Portela & Ca Sa Pochodne nitrokatecholowe jako inhibitory COMT
EP1845097A1 (en) * 2006-04-10 2007-10-17 Portela & Ca., S.A. Oxadiazole derivatives as COMT inhibitors
PT2069336E (pt) * 2006-09-07 2013-03-07 Actelion Pharmaceuticals Ltd Derivados de piridin-4-ilo como agentes imunomoduladores
PL2069335T3 (pl) * 2006-09-08 2013-05-31 Actelion Pharmaceuticals Ltd Pochodne pirydyn-3-ylu jako środki immunomodulujące
BRPI0721213B1 (pt) * 2007-01-31 2021-11-09 Bial - Portela & Ca, S.A. Uso de nitrocatecóis substituídos, e embalagem
BRPI0808789A2 (pt) * 2007-03-16 2014-08-12 Actelion Pharmaceuticals Ltd Compostos e composição farmacêutica de derivados aminopiridina e uso destes
PT2195311E (pt) * 2007-08-17 2011-05-25 Actelion Pharmaceuticals Ltd Derivados de piridina como moduladores do receptor s1p1/edg1
MX2010009043A (es) * 2008-02-28 2010-10-25 Bial Portela & Ca Sa Composicion farmaceutica para farmacos poco solubles.
EP2262799B1 (en) * 2008-03-06 2012-07-04 Actelion Pharmaceuticals Ltd. Pyridine compounds
WO2009109872A1 (en) * 2008-03-07 2009-09-11 Actelion Pharmaceuticals Ltd Pyridin-2-yl derivatives as immunomodulating agents
WO2009116882A1 (en) 2008-03-17 2009-09-24 Portela & Ca., S.A. Crystal forms of 5- [3- (2, 5-dichloro-4, 6-dimethyl-1-oxy-pyridine-3-yl) [1,2,3] oxadiazol-5-yl] -3-nit robenzene-1, 2-diol
EP3782991A1 (en) 2008-05-14 2021-02-24 The Scripps Research Institute Novel modulators of sphingosine phosphate receptors
CN105418598B (zh) 2009-02-10 2019-05-17 孟山都技术有限公司 用于控制线虫的组合物和方法
PT2413912T (pt) 2009-04-01 2019-06-11 Bial Portela & Ca Sa Formulações farmacêuticas compreendendo derivados de nitrocatecol e métodos para as produzir
BRPI1016132B8 (pt) * 2009-04-01 2021-05-25 Bial Portela & Ca Sa composição, formulação farmacêutica, processo de obtenção de uma formulação farmacêutica estável
CA2767585C (en) 2009-07-16 2017-09-26 Actelion Pharmaceuticals Ltd Pyridin-4-yl derivatives
MA34910B1 (fr) 2011-01-19 2014-02-01 Actelion Pharmaceuticals Ltd Dérivés de 2-methoxy-pyridin-4-yl
US20140045900A1 (en) 2011-02-11 2014-02-13 Bial-Portela & Ca, S.A. Administration regime for nitrocatechols
JP6456143B2 (ja) 2011-12-13 2019-01-23 ノヴィファーマ,エス.アー. カテコール−o−メチル転移酵素阻害剤を調製するための中間体として有用な化学的化合物
US9232800B2 (en) 2013-02-15 2016-01-12 Monsanto Technology Llc 3,5-disubstituted-4,5-dihydro-1,2,4-oxadiazoles and compositions and methods for controlling nematode pests
RU2017120184A (ru) 2014-11-28 2018-12-28 БИАЛ - ПОРТЕЛА ЭНД Ка, С.А. Лекарства для замедления течения болезни паркинсона
PH12017502097B1 (en) 2015-05-20 2023-05-05 Idorsia Pharmaceuticals Ltd Crystalline form of the compound (s)-3-{4-[5-(2-cyclopentyl-6-methoxy-pyridin-4-yl)-[1,2,4]oxadiazol-3-yl]-2-ethyl-6-methyl-phenoxy}-propane-1,2-diol

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL120029C (https=) * 1959-09-29
US3227725A (en) * 1962-04-17 1966-01-04 Union Carbide Corp Certain 3,5-disubstituted 1,2,4-oxadiazole compounds

Also Published As

Publication number Publication date
PL79435B1 (en) 1975-06-30
SE368576B (https=) 1974-07-08
IL31990A0 (en) 1969-06-25
CH540925A (de) 1973-08-31
BE732131A (https=) 1969-10-01
FR2007529B1 (https=) 1973-03-16
NO124253B (https=) 1972-03-27
DE1920037A1 (de) 1970-11-12
AT292728B (de) 1971-09-10
US3647809A (en) 1972-03-07
CH542232A (de) 1973-11-15
AT292727B (de) 1971-09-10
JPS4824394B1 (https=) 1973-07-20
IL31990A (en) 1974-05-16
FR2007529A1 (https=) 1970-01-09
NL6906401A (https=) 1969-10-28
CA954858A (en) 1974-09-17
GB1271302A (en) 1972-04-19

Similar Documents

Publication Publication Date Title
BR6908381D0 (pt) Novos derivados de piridil-oxadiasol e processo para a sua preparacao
BR6677982D0 (pt) Processo para a preparacao de derivados basicos de ftalanas e iso-cromanas
BR6678981D0 (pt) Alcenil-fenoxi-isopropanolaminas e processo para sua preparacao
BR6908638D0 (pt) Processo para a preparacao de organo-silano-penicilinas
BR6909792D0 (pt) Processo para a preparacao de hidro-uracilas halo-substituidas
BR6914562D0 (pt) Processo para obtencao de novos derivados de trepira e oxepira
BR6914375D0 (pt) Processo para a preparacao de benzindenos
BR7019360D0 (pt) Processo para obtencao de novos derivados do diabenzo a e cicloocten-s 11-imina
BR6912232D0 (pt) Processo para a preparacao de derivados de piridoindol
BR6909976D0 (pt) Processo para a preparacao de derivados etenicos
BR6914563D0 (pt) Processo para a obtencao de novos derivados de ozepira
BR6912234D0 (pt) Processo para a preparacao de derivados de piridoindol
BR6911561D0 (pt) Novos derivados de finantridina e processo para sua preparacao
BR6912949D0 (pt) Processo para a preparacao de novos derivados de indano
BR6911905D0 (pt) Processo para a preparacao de imidazopirazinonas
BR6911906D0 (pt) Processo para a preparacao de imidazopirazinonas
BR6913178D0 (pt) Processo para a preparacao de 19-nor-esteroides
BR6907491D0 (pt) Novas cefalosporinas e processo para sua preparacao
BR6911331D0 (pt) Novos derivados de pirrolidina e de processo para a sua preparacao
BR6912482D0 (pt) Processo para a preparacao de cromenopirazol
BR6906644D0 (pt) Processo para a preparacao de cromanois
BR6906559D0 (pt) Derivados de piperazina e processo para sua preparacao
BR6911651D0 (pt) Compostos tendo atividade anti-xistosomose e processo para sua preparacao
BR6911648D0 (pt) Processo para a preparacao de dibenzo-cidohepteno
BR6914629D0 (pt) Fenetilaminas orto-substituidas e processo para a sua obtencao