BR112022012130A2 - Compostos antelmínticos compreendendo uma estrutura azaindólica - Google Patents
Compostos antelmínticos compreendendo uma estrutura azaindólicaInfo
- Publication number
- BR112022012130A2 BR112022012130A2 BR112022012130A BR112022012130A BR112022012130A2 BR 112022012130 A2 BR112022012130 A2 BR 112022012130A2 BR 112022012130 A BR112022012130 A BR 112022012130A BR 112022012130 A BR112022012130 A BR 112022012130A BR 112022012130 A2 BR112022012130 A2 BR 112022012130A2
- Authority
- BR
- Brazil
- Prior art keywords
- compounds
- azaindolic
- antelminthic
- dirofilaria
- helminths
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
- A01P5/00—Nematocides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Abstract
COMPOSTOS ANTELMÍNTICOS COMPREENDENDO UMA ESTRUTURA AZAINDÓLICA. A presente invenção se refere a novos compostos antelmínticos. Estes compostos podem, por exemplo, serem usados no tratamento do tipo doença parasitária causada por helmintos, tais como Dirofilaria, em particular Dirofilaria immitis.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP19217671 | 2019-12-18 | ||
EP20213299 | 2020-12-11 | ||
PCT/EP2020/086660 WO2021122906A1 (en) | 2019-12-18 | 2020-12-17 | Anthelmintic compounds comprising azaindoles structure |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112022012130A2 true BR112022012130A2 (pt) | 2022-08-30 |
Family
ID=74106031
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112022012130A BR112022012130A2 (pt) | 2019-12-18 | 2020-12-17 | Compostos antelmínticos compreendendo uma estrutura azaindólica |
Country Status (9)
Country | Link |
---|---|
US (1) | US20230110397A1 (pt) |
EP (1) | EP4077322A1 (pt) |
JP (1) | JP2023506303A (pt) |
CN (1) | CN114846014A (pt) |
AU (1) | AU2020404100A1 (pt) |
BR (1) | BR112022012130A2 (pt) |
CA (1) | CA3164104A1 (pt) |
MX (1) | MX2022007671A (pt) |
WO (1) | WO2021122906A1 (pt) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PE20220281A1 (es) | 2019-03-19 | 2022-02-25 | Boehringer Ingelheim Animal Health Usa Inc | Compuestos de aza-benzotiofeno y aza-benzofurano como antihelminticos |
IL298596A (en) | 2020-05-29 | 2023-01-01 | Boehringer Ingelheim Animal Health Usa Inc | Heterocyclic anthelmintic compounds |
AR127495A1 (es) | 2021-11-01 | 2024-01-31 | Boehringer Ingelheim Vetmedica Gmbh | Compuestos de pirrolopiridazina como antihelmínticos |
CN116969976A (zh) * | 2022-04-28 | 2023-10-31 | 杭州普济远成生物医药科技有限公司 | 去泛素化酶抑制剂及其应用 |
Family Cites Families (36)
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EP0539588A1 (en) | 1990-07-05 | 1993-05-05 | Nippon Soda Co., Ltd. | Amine derivative |
US5399582A (en) | 1993-11-01 | 1995-03-21 | Merck & Co., Inc. | Antiparasitic agents |
US6221894B1 (en) | 1995-03-20 | 2001-04-24 | Merck & Co., Inc. | Nodulisporic acid derivatives |
US5595991A (en) | 1995-03-20 | 1997-01-21 | Merck & Co., Inc. | Anthelmintic use of nodulisporic acid and analogs thereof |
US5962499A (en) | 1995-03-20 | 1999-10-05 | Merck & Co., Inc. | Nodulisporic acid derivatives |
CZ294699B6 (cs) | 1995-03-20 | 2005-02-16 | Merck And Co., Inc. | Deriváty kyseliny nodulisporové a farmaceutický prostředek s jejich obsahem |
US5834260A (en) | 1996-08-30 | 1998-11-10 | Merck & Co., Inc. | Antiparasitic agents |
DK1390340T3 (en) | 2001-04-24 | 2017-05-15 | Massachusetts Inst Technology | Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds |
US7361689B2 (en) | 2003-12-31 | 2008-04-22 | Schering-Plough Animal Health Corporation | Antibacterial 1-(4-mono- and di-halomethylsulphonylphenyl)-2-acylamino-3-fluoroproponals and preparation thereof |
EP1699799B1 (en) | 2003-12-31 | 2007-05-16 | Schering-Plough Ltd. | Control of parasites in animals by the use of imidazo [1,2-b]pyridazine derivatives |
MX2007003378A (es) | 2004-09-23 | 2007-05-10 | Schering Plough Ltd | Control de parasitos en animales mediante el uso de nuevos derivados de trifluorometansulfonanilida oxima eter. |
WO2006055565A2 (en) | 2004-11-19 | 2006-05-26 | Schering-Plough Ltd. | Control of parasites in animals by the use of parasiticidal 2-phenyl-3-(1h-pyrrol-2-yl) acrylonitrile derivatives |
AR054380A1 (es) | 2005-06-09 | 2007-06-20 | Schering Plough Ltd | Control de parasitos en animales con derivados de n- ((feniloxi) fenil) -1,1,1-trifluorometansulfonamida y de n-(fenilsulfanil) fenil) -1,1,1-trifluorometansulfonamida |
DE102006015470A1 (de) | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
US8809268B2 (en) | 2008-10-29 | 2014-08-19 | The Regents Of The University Of California | Combination therapy to combat helminth resistance |
US8007761B2 (en) | 2008-12-24 | 2011-08-30 | Praxair Technology, Inc. | Carbon dioxide emission reduction method |
CN113603675A (zh) | 2015-12-17 | 2021-11-05 | 默克专利有限公司 | 多环tlr7/8拮抗剂及其在治疗免疫失调中的用途 |
MX2018012544A (es) | 2016-04-15 | 2019-01-31 | Bayer Animal Health Gmbh | Nuevos derivados de pirazolopirimidina. |
TWI679197B (zh) | 2016-05-05 | 2019-12-11 | 瑞士商伊蘭科動物健康公司 | 雜芳基-1,2,4-三唑及雜芳基-三唑化合物 |
KR20200129128A (ko) | 2018-03-08 | 2020-11-17 | 바이엘 악티엔게젤샤프트 | 식물 보호에서 살충제로서의 헤테로아릴-트리아졸 및 헤테로아릴-테트라졸 화합물의 용도 |
EP3904349B1 (en) | 2018-04-12 | 2023-08-23 | Bayer Aktiengesellschaft | N-(cyclopropylmethyl)-5-(methylsulfonyl)-n-{1-[1-(pyrimidin-2-yl)-1h-1,2,4-triazol-5-yl]ethyl}heterocyclyl amide derivatives and similar compounds as pesticides |
UY38184A (es) | 2018-04-17 | 2019-10-31 | Bayer Ag | Compuestos heteroarilo-triazol y heteroarilo-tetrazol novedosos como plaguicidas |
UA127065C2 (uk) | 2018-04-25 | 2023-03-29 | Баєр Акціенгезельшафт | Нові гетероарил-триазольні та гетероарил-тетразольні сполуки як пестициди |
WO2019215198A1 (en) | 2018-05-08 | 2019-11-14 | Syngenta Crop Protection Ag | Methods of applying one or more certain heteroaryl-1,2,4-triazole and heteroaryl-tetrazole compounds to control damage on plants, propagation material thereof, and plant derived products |
TW202019901A (zh) | 2018-09-13 | 2020-06-01 | 瑞士商先正達合夥公司 | 殺有害生物活性唑-醯胺化合物 |
TW202023386A (zh) | 2018-09-13 | 2020-07-01 | 瑞士商先正達合夥公司 | 殺有害生物活性唑-醯胺化合物 |
UY38394A (es) | 2018-10-02 | 2020-04-30 | Syngenta Participations Ag | Compuestos de benceno y azina-amida activos como plaguicidas |
ES2953567T3 (es) | 2018-10-19 | 2023-11-14 | Syngenta Participations Ag | Compuestos de azol-amida plaguicidamente activos |
CN112955442A (zh) | 2018-11-05 | 2021-06-11 | 先正达参股股份有限公司 | 杀有害生物活性的唑-酰胺化合物 |
EP3696175A1 (en) | 2019-02-18 | 2020-08-19 | Syngenta Crop Protection AG | Pesticidally active azole-amide compounds |
BR112021018822A2 (pt) | 2019-03-22 | 2021-11-23 | Syngenta Crop Prot Ag | Derivados de n-[1-(5-bromo-2-pirimidin-2-il-1,2,4-triazol-3-il)etil]-2-ciclopropil-6-(trifluorometil)piridina-4-carboxamida e compostos relacionados como inseticidas |
UY38623A (es) | 2019-03-29 | 2020-10-30 | Syngenta Crop Protection Ag | Compuestos de diazina-amida activos como pesticidas |
MX2021012162A (es) | 2019-04-05 | 2021-11-03 | Syngenta Crop Protection Ag | Compuestos de diazina-amida activos como pesticidas. |
CN113677672A (zh) | 2019-04-11 | 2021-11-19 | 先正达农作物保护股份公司 | 杀有害生物活性的二嗪-酰胺化合物 |
EP3725788A1 (en) | 2019-04-15 | 2020-10-21 | Bayer AG | Novel heteroaryl-substituted aminoalkyl azole compounds as pesticides |
CN114072395A (zh) | 2019-04-26 | 2022-02-18 | 新基公司 | 杂环化合物及其治疗蠕虫感染和疾病的用途 |
-
2020
- 2020-12-17 CN CN202080088930.0A patent/CN114846014A/zh active Pending
- 2020-12-17 US US17/785,646 patent/US20230110397A1/en active Pending
- 2020-12-17 WO PCT/EP2020/086660 patent/WO2021122906A1/en unknown
- 2020-12-17 AU AU2020404100A patent/AU2020404100A1/en active Pending
- 2020-12-17 BR BR112022012130A patent/BR112022012130A2/pt unknown
- 2020-12-17 EP EP20833809.5A patent/EP4077322A1/en active Pending
- 2020-12-17 MX MX2022007671A patent/MX2022007671A/es unknown
- 2020-12-17 CA CA3164104A patent/CA3164104A1/en active Pending
- 2020-12-17 JP JP2022537141A patent/JP2023506303A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
EP4077322A1 (en) | 2022-10-26 |
AU2020404100A1 (en) | 2022-06-09 |
CN114846014A (zh) | 2022-08-02 |
JP2023506303A (ja) | 2023-02-15 |
WO2021122906A1 (en) | 2021-06-24 |
US20230110397A1 (en) | 2023-04-13 |
CA3164104A1 (en) | 2021-06-24 |
MX2022007671A (es) | 2022-07-19 |
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