MX2022007671A - Compuestos antihelminticos que comprenden una estructura de azaindoles. - Google Patents
Compuestos antihelminticos que comprenden una estructura de azaindoles.Info
- Publication number
- MX2022007671A MX2022007671A MX2022007671A MX2022007671A MX2022007671A MX 2022007671 A MX2022007671 A MX 2022007671A MX 2022007671 A MX2022007671 A MX 2022007671A MX 2022007671 A MX2022007671 A MX 2022007671A MX 2022007671 A MX2022007671 A MX 2022007671A
- Authority
- MX
- Mexico
- Prior art keywords
- azaindoles
- anthelmintic compounds
- compounds
- dirofilaria
- anthelmintic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
- A01P5/00—Nematocides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Wood Science & Technology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Environmental Sciences (AREA)
- Zoology (AREA)
- Plant Pathology (AREA)
- Engineering & Computer Science (AREA)
- Tropical Medicine & Parasitology (AREA)
- Dentistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Agronomy & Crop Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
La presente invención se refiere a nuevos compuestos antihelmínticos. Estos compuestos se pueden usar por ejemplo en el tratamiento del tipo de helmintiasis causados por helmintos tal como Dirofilaria, en particular Dirofilaria immitis.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP19217671 | 2019-12-18 | ||
EP20213299 | 2020-12-11 | ||
PCT/EP2020/086660 WO2021122906A1 (en) | 2019-12-18 | 2020-12-17 | Anthelmintic compounds comprising azaindoles structure |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2022007671A true MX2022007671A (es) | 2022-07-19 |
Family
ID=74106031
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2022007671A MX2022007671A (es) | 2019-12-18 | 2020-12-17 | Compuestos antihelminticos que comprenden una estructura de azaindoles. |
Country Status (9)
Country | Link |
---|---|
US (1) | US20230110397A1 (es) |
EP (1) | EP4077322A1 (es) |
JP (1) | JP2023506303A (es) |
CN (1) | CN114846014A (es) |
AU (1) | AU2020404100A1 (es) |
BR (1) | BR112022012130A2 (es) |
CA (1) | CA3164104A1 (es) |
MX (1) | MX2022007671A (es) |
WO (1) | WO2021122906A1 (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US11560388B2 (en) | 2019-03-19 | 2023-01-24 | Boehringer Ingelheim Vetmedica Gmbh | Anthelmintic aza-benzothiophene and aza-benzofuran compounds |
WO2021242581A1 (en) | 2020-05-29 | 2021-12-02 | Boehringer Ingelheim Animal Health USA Inc. | Anthelmintic heterocyclic compounds |
CA3236894A1 (en) | 2021-11-01 | 2023-05-04 | Boehringer Ingelheim Vetmedica Gmbh | Anthelmintic pyrrolopyridazine compounds |
CN116969976A (zh) * | 2022-04-28 | 2023-10-31 | 杭州普济远成生物医药科技有限公司 | 去泛素化酶抑制剂及其应用 |
Family Cites Families (36)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0539588A1 (en) | 1990-07-05 | 1993-05-05 | Nippon Soda Co., Ltd. | Amine derivative |
US5399582A (en) | 1993-11-01 | 1995-03-21 | Merck & Co., Inc. | Antiparasitic agents |
SK284840B6 (sk) | 1995-03-20 | 2005-12-01 | Merck & Co., Inc. | Deriváty kyseliny nodulisporovej a farmaceutický prostriedok s ich obsahom |
US6221894B1 (en) | 1995-03-20 | 2001-04-24 | Merck & Co., Inc. | Nodulisporic acid derivatives |
US5595991A (en) | 1995-03-20 | 1997-01-21 | Merck & Co., Inc. | Anthelmintic use of nodulisporic acid and analogs thereof |
US5962499A (en) | 1995-03-20 | 1999-10-05 | Merck & Co., Inc. | Nodulisporic acid derivatives |
US5834260A (en) | 1996-08-30 | 1998-11-10 | Merck & Co., Inc. | Antiparasitic agents |
EP1390340B1 (en) | 2001-04-24 | 2017-03-01 | Massachusetts Institute Of Technology | Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds |
WO2005066119A2 (en) | 2003-12-31 | 2005-07-21 | Schering-Plough Ltd. | Antibacterial 1-(4-mono-and di-halomethylsulphonylphenyl)-2-acylamino-3-fluoropropanols and preparation thereof |
NZ548098A (en) | 2003-12-31 | 2010-05-28 | Schering Plough Ltd | Control of parasites in animals by the use of imidazo[1,2-b]pyridazine derivatives |
ES2314724T3 (es) | 2004-09-23 | 2009-03-16 | Schering-Plough Ltd. | Control de parasitos en animales mediante el uso de nuevos derivados de eter de trifluorometanosulfonanilida oxima. |
CA2587495A1 (en) | 2004-11-19 | 2006-05-26 | Schering-Plough Ltd. | Control of parasites in animals by the use of parasiticidal 2-phenyl-3-(1h-pyrrol-2-yl) acrylonitrile derivatives |
MX2007015729A (es) | 2005-06-09 | 2008-02-21 | Schering Plough Ltd | Control de parasitos en animales con derivados de n-[(feniloxi)fenil]-1,1,1-trifluorometansulfonamida y de n[(fenilsulfanil)fenil]-1,1,1-trifluorometansulfonamida. |
DE102006015470A1 (de) | 2006-03-31 | 2007-10-04 | Bayer Cropscience Ag | Substituierte Enaminocarbonylverbindungen |
US8809268B2 (en) | 2008-10-29 | 2014-08-19 | The Regents Of The University Of California | Combination therapy to combat helminth resistance |
US8007761B2 (en) | 2008-12-24 | 2011-08-30 | Praxair Technology, Inc. | Carbon dioxide emission reduction method |
DK3889145T3 (da) | 2015-12-17 | 2024-03-18 | Merck Patent Gmbh | 8-cyano-5-piperidino-quinoliner som TLR7/8-antagonister og anvendelser deraf til behandling af immunsygdomme |
ES2953467T3 (es) | 2016-04-15 | 2023-11-13 | Elanco Animal Health Gmbh | Derivados de pirazolopirimidina |
TWI696615B (zh) | 2016-05-05 | 2020-06-21 | 瑞士商伊蘭科動物健康公司 | 雜芳基-1,2,4-三唑及雜芳基-三唑化合物 |
US20200404919A1 (en) | 2018-03-08 | 2020-12-31 | Bayer Aktiengesellschaft | Use of heteroaryl-triazole and heteroaryl-tetrazole compounds as pesticides in plant protection |
ES2965494T3 (es) | 2018-04-12 | 2024-04-15 | Bayer Ag | Derivados de N-(ciclopropilmetil)-5-(metilsulfonil)-n-{1-[1-(pirimidin-2-il)-1H-1,2,4-triazol-5-il]etil}benzamida y los correspondientes derivados de piridina-carboxamida como plaguicidas |
UY38184A (es) | 2018-04-17 | 2019-10-31 | Bayer Ag | Compuestos heteroarilo-triazol y heteroarilo-tetrazol novedosos como plaguicidas |
DK3919486T3 (da) | 2018-04-25 | 2023-09-04 | Bayer Ag | Hidtil ukendte heteroaryl-triazol- og heteroaryl-tetrazolforbindelser som pesticider |
WO2019215198A1 (en) | 2018-05-08 | 2019-11-14 | Syngenta Crop Protection Ag | Methods of applying one or more certain heteroaryl-1,2,4-triazole and heteroaryl-tetrazole compounds to control damage on plants, propagation material thereof, and plant derived products |
TW202019901A (zh) | 2018-09-13 | 2020-06-01 | 瑞士商先正達合夥公司 | 殺有害生物活性唑-醯胺化合物 |
TW202023386A (zh) | 2018-09-13 | 2020-07-01 | 瑞士商先正達合夥公司 | 殺有害生物活性唑-醯胺化合物 |
JP7485660B2 (ja) | 2018-10-02 | 2024-05-16 | シンジェンタ パーティシペーションズ アーゲー | 殺有害生物性活性ベンゼン-及びアジン-アミド化合物 |
CN112888680A (zh) | 2018-10-19 | 2021-06-01 | 先正达参股股份有限公司 | 杀有害生物活性的唑-酰胺化合物 |
BR112021008675A2 (pt) | 2018-11-05 | 2021-08-10 | Syngenta Participations Ag | compostos de azole-amida pesticidamente ativos |
EP3696175A1 (en) | 2019-02-18 | 2020-08-19 | Syngenta Crop Protection AG | Pesticidally active azole-amide compounds |
CN113597426A (zh) | 2019-03-22 | 2021-11-02 | 先正达农作物保护股份公司 | N-[1-(5-溴-2-嘧啶-2-基-1,2,4-三唑-3-基)乙基]-2-环丙基-6-(三氟甲基)吡啶-4-甲酰胺衍生物及相关的化合物作为杀昆虫剂 |
TW202102489A (zh) | 2019-03-29 | 2021-01-16 | 瑞士商先正達農作物保護公司 | 殺有害生物活性之二𠯤-醯胺化合物 |
CA3131479A1 (en) | 2019-04-05 | 2020-10-08 | Jurgen Harry Schaetzer | Pesticidally active diazine-amide compounds |
MX2021012290A (es) | 2019-04-11 | 2021-11-12 | Syngenta Crop Protection Ag | Compuestos de diazina-amida activos como pesticidas. |
EP3725788A1 (en) | 2019-04-15 | 2020-10-21 | Bayer AG | Novel heteroaryl-substituted aminoalkyl azole compounds as pesticides |
WO2020219871A1 (en) | 2019-04-26 | 2020-10-29 | Celgene Corporation | Heterocyclic compounds and their use for treatment of helminthic infections and diseases |
-
2020
- 2020-12-17 CN CN202080088930.0A patent/CN114846014A/zh active Pending
- 2020-12-17 AU AU2020404100A patent/AU2020404100A1/en active Pending
- 2020-12-17 US US17/785,646 patent/US20230110397A1/en active Pending
- 2020-12-17 JP JP2022537141A patent/JP2023506303A/ja active Pending
- 2020-12-17 CA CA3164104A patent/CA3164104A1/en active Pending
- 2020-12-17 MX MX2022007671A patent/MX2022007671A/es unknown
- 2020-12-17 BR BR112022012130A patent/BR112022012130A2/pt unknown
- 2020-12-17 EP EP20833809.5A patent/EP4077322A1/en active Pending
- 2020-12-17 WO PCT/EP2020/086660 patent/WO2021122906A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
JP2023506303A (ja) | 2023-02-15 |
AU2020404100A1 (en) | 2022-06-09 |
EP4077322A1 (en) | 2022-10-26 |
US20230110397A1 (en) | 2023-04-13 |
BR112022012130A2 (pt) | 2022-08-30 |
CA3164104A1 (en) | 2021-06-24 |
CN114846014A (zh) | 2022-08-02 |
WO2021122906A1 (en) | 2021-06-24 |
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