BR112016015763B8 - preparação farmacêutica incluindo composto de ácido piridilaminocético, e, uso da mesma - Google Patents

preparação farmacêutica incluindo composto de ácido piridilaminocético, e, uso da mesma

Info

Publication number
BR112016015763B8
BR112016015763B8 BR112016015763A BR112016015763A BR112016015763B8 BR 112016015763 B8 BR112016015763 B8 BR 112016015763B8 BR 112016015763 A BR112016015763 A BR 112016015763A BR 112016015763 A BR112016015763 A BR 112016015763A BR 112016015763 B8 BR112016015763 B8 BR 112016015763B8
Authority
BR
Brazil
Prior art keywords
pharmaceutical preparation
pyridylaminocetic
intraocular pressure
glaucoma
compounds
Prior art date
Application number
BR112016015763A
Other languages
English (en)
Other versions
BR112016015763B1 (pt
Inventor
Kroon Henk-Andre
Kawata Hisashi
Shams Naveed
Kawabata Noriko
Original Assignee
Santen Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=53520400&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR112016015763(B8) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Santen Pharmaceutical Co Ltd filed Critical Santen Pharmaceutical Co Ltd
Publication of BR112016015763B1 publication Critical patent/BR112016015763B1/pt
Publication of BR112016015763B8 publication Critical patent/BR112016015763B8/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0048—Eye, e.g. artificial tears
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Ophthalmology & Optometry (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

preparação farmacêutica, e, método para tratamento ou prevenção de glaucoma ou hipertensão ocular o propósito da presente invenção é descobrir quais compostos dentre o vasto número de compostos de ácido piridilaminocético apresentam uma ação de abaixamento de pressão intraocular notoriamente superior e podem servir como um agente abaixador de pressão intraocular ou como um agente tera-pêutico ou preventivo contra glaucoma ou hipertensão ocular, e descobrir a maneira de administração e/ou de dosagem na qual os compostos desco-bertos concederão um efeito terapêutico ou profilático efetivo quando admi-nistrados aos pacientes (principalmente seres humanos). é fornecida uma preparação farmacêutica para abaixar a pressão intraocular ou para prevenir ou tratar glaucoma ou hipertensão intraocular, a dita preparação farmacêutica contendo 0,0003 a 0,01% (m/v) de (6-{[4-(pirazol-1-il)benzil](piridin-3-ilsulfonil)aminometil}piridin-2-ilamino)acetato de isopropila, ou um sal do mesmo.
BR112016015763A 2014-01-10 2015-01-08 preparação farmacêutica incluindo composto de ácido piridilaminocético, e, uso da mesma BR112016015763B8 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201461925882P 2014-01-10 2014-01-10
US61/925882 2014-01-10
PCT/JP2015/050366 WO2015105144A1 (ja) 2014-01-10 2015-01-08 ピリジルアミノ酢酸化合物を含む医薬製剤

Publications (2)

Publication Number Publication Date
BR112016015763B1 BR112016015763B1 (pt) 2020-09-01
BR112016015763B8 true BR112016015763B8 (pt) 2020-09-15

Family

ID=53520400

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112016015763A BR112016015763B8 (pt) 2014-01-10 2015-01-08 preparação farmacêutica incluindo composto de ácido piridilaminocético, e, uso da mesma

Country Status (26)

Country Link
US (8) US9415038B2 (pt)
EP (3) EP3750541A1 (pt)
JP (6) JP5846338B2 (pt)
KR (1) KR101824829B1 (pt)
CN (2) CN108743587B (pt)
AU (1) AU2015205188B2 (pt)
BR (1) BR112016015763B8 (pt)
CA (1) CA2936026C (pt)
CL (1) CL2016001756A1 (pt)
DK (1) DK3093018T3 (pt)
EA (1) EA031734B1 (pt)
ES (2) ES2711091T3 (pt)
GE (1) GEP20186917B (pt)
HK (1) HK1223036A1 (pt)
HU (1) HUE041653T2 (pt)
IL (1) IL246447B (pt)
MX (1) MX370361B (pt)
MY (1) MY163235A (pt)
PH (1) PH12016501357A1 (pt)
PL (1) PL3093018T3 (pt)
PT (1) PT3093018T (pt)
SG (1) SG11201605653RA (pt)
TR (1) TR201902019T4 (pt)
TW (1) TWI598113B (pt)
UA (1) UA117506C2 (pt)
WO (1) WO2015105144A1 (pt)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101858373B1 (ko) * 2014-01-10 2018-05-15 산텐 세이야꾸 가부시키가이샤 피리딜아미노아세트산 화합물과 폴리옥시에틸렌 피마자유를 함유하는 의약 조성물
EP3750541A1 (en) 2014-01-10 2020-12-16 Santen Pharmaceutical Co., Ltd Pharmaceutical preparation containing pyridylaminoacetic acid compound
AU2015205179B2 (en) 2014-01-10 2019-09-19 Santen Pharmaceutical Co., Ltd. Pharmaceutical composition containing pyridylamino acetic acid compound
MX2017007572A (es) * 2014-12-12 2018-02-09 Kowa Co Composicion acuosa.
AR105215A1 (es) * 2015-07-01 2017-09-13 Santen Pharmaceutical Co Ltd Formulación de depósito que contiene ésteres de ácido cítrico
JP7032134B2 (ja) * 2015-07-09 2022-03-08 参天製薬株式会社 ピリジルアミノ酢酸化合物を含有する予防及び／又は治療剤
WO2018230713A1 (ja) 2017-06-16 2018-12-20 学校法人同志社 カスパーゼ阻害活性を有する化合物、これらの化合物を含む、角膜内皮の症状、障害または疾患を治療または予防するための医薬およびその応用
CA3067332A1 (en) 2017-06-16 2018-12-20 The Doshisha Mtor-inhibitor-containing medicine for treating or preventing ophthalmic symptoms, disorders, or diseases, and application thereof
WO2019065838A1 (ja) 2017-09-29 2019-04-04 参天製薬株式会社 ピリジルアミノ酢酸化合物を含有する医薬
EP3730143A4 (en) 2017-12-21 2021-08-18 Santen Pharmaceutical Co., Ltd. OMIDENEPAG COMBINATION
US11666563B2 (en) 2017-12-28 2023-06-06 Santen Pharmaceutical Co., Ltd. Pharmaceutical preparation containing pyridyl aminoacetic acid compound
WO2019209955A2 (en) * 2018-04-24 2019-10-31 Allergan, Inc. Presbyopia treatments

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2002356420A (ja) * 2001-03-27 2002-12-13 Santen Pharmaceut Co Ltd 安定な水性液剤
DK2264009T3 (en) 2008-03-12 2019-04-15 Ube Industries PYRIDYLAMINE ACEDIC ACID COMPOUND
CA2757291C (en) * 2009-03-30 2017-05-23 Ube Industries, Ltd. Medical composition for treatment or prophylaxis of glaucoma
JP2011057633A (ja) * 2009-09-11 2011-03-24 Ube Industries Ltd ピリジルアミノ酢酸化合物を含有する医薬
US20120202863A1 (en) * 2011-02-03 2012-08-09 Gerald Horn Compositions and methods for treatment of glaucoma
JP2014019650A (ja) * 2012-07-13 2014-02-03 Santen Pharmaceut Co Ltd スルホンアミド化合物とタフルプロストの組み合わせ
US9339496B2 (en) * 2012-07-13 2016-05-17 Santen Pharmaceutical Co., Ltd. Composition for treating or preventing glaucoma comprising a sulfonamide compound, and a beta-receptor antagonist
KR102074020B1 (ko) * 2012-07-13 2020-02-05 산텐 세이야꾸 가부시키가이샤 술폰아미드 화합물의 조합
US20140018350A1 (en) 2012-07-13 2014-01-16 Asahi Glass Co., Ltd. Combination of sulfonamide compound and tafluprost
KR101858373B1 (ko) 2014-01-10 2018-05-15 산텐 세이야꾸 가부시키가이샤 피리딜아미노아세트산 화합물과 폴리옥시에틸렌 피마자유를 함유하는 의약 조성물
EP3750541A1 (en) 2014-01-10 2020-12-16 Santen Pharmaceutical Co., Ltd Pharmaceutical preparation containing pyridylaminoacetic acid compound
AU2015205179B2 (en) * 2014-01-10 2019-09-19 Santen Pharmaceutical Co., Ltd. Pharmaceutical composition containing pyridylamino acetic acid compound

Also Published As

Publication number Publication date
US10702511B2 (en) 2020-07-07
EP3093018A1 (en) 2016-11-16
GEP20186917B (en) 2018-11-12
EP3750541A1 (en) 2020-12-16
TW201609186A (zh) 2016-03-16
JP7087040B2 (ja) 2022-06-20
MX370361B (es) 2019-12-10
IL246447B (en) 2020-06-30
JP6785330B2 (ja) 2020-11-18
NZ721620A (en) 2021-08-27
USRE48183E1 (en) 2020-09-01
EP3093018A4 (en) 2017-09-13
AU2015205188B2 (en) 2019-11-14
PT3093018T (pt) 2019-01-10
KR20160101030A (ko) 2016-08-24
US20200289483A1 (en) 2020-09-17
CN105899209B (zh) 2018-09-11
ES2711091T3 (es) 2019-04-30
IL246447A0 (en) 2016-08-31
TR201902019T4 (tr) 2019-03-21
EA031734B1 (ru) 2019-02-28
US20150196541A1 (en) 2015-07-16
EP3424503B1 (en) 2020-09-02
US9415038B2 (en) 2016-08-16
JP2016027060A (ja) 2016-02-18
US20190105310A1 (en) 2019-04-11
JP7402922B2 (ja) 2023-12-21
HK1223036A1 (zh) 2017-07-21
US10179127B2 (en) 2019-01-15
HUE041653T2 (hu) 2019-05-28
CA2936026A1 (en) 2015-07-16
CA2936026C (en) 2022-04-19
US20180169079A1 (en) 2018-06-21
US9943510B2 (en) 2018-04-17
US20240000763A1 (en) 2024-01-04
EP3093018B1 (en) 2018-11-28
UA117506C2 (uk) 2018-08-10
BR112016015763B1 (pt) 2020-09-01
ES2834334T3 (es) 2021-06-17
JP2024019479A (ja) 2024-02-09
AU2015205188A1 (en) 2016-07-14
JP2019108363A (ja) 2019-07-04
JP2022111280A (ja) 2022-07-29
CN105899209A (zh) 2016-08-24
CN108743587B (zh) 2021-04-30
PH12016501357B1 (en) 2016-08-15
SG11201605653RA (en) 2016-08-30
US20220054466A1 (en) 2022-02-24
DK3093018T3 (en) 2019-02-04
CL2016001756A1 (es) 2017-05-12
PL3093018T3 (pl) 2019-05-31
JP2021006593A (ja) 2021-01-21
US11793798B2 (en) 2023-10-24
KR101824829B1 (ko) 2018-02-01
JPWO2015105144A1 (ja) 2017-03-23
MY163235A (en) 2017-08-30
US20160324838A1 (en) 2016-11-10
US11197849B2 (en) 2021-12-14
CN108743587A (zh) 2018-11-06
JP6491588B2 (ja) 2019-03-27
MX2016009063A (es) 2016-09-28
JP5846338B2 (ja) 2016-01-20
PH12016501357A1 (en) 2016-08-15
TWI598113B (zh) 2017-09-11
WO2015105144A1 (ja) 2015-07-16
EA201691402A1 (ru) 2016-10-31
EP3424503A1 (en) 2019-01-09

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 08/01/2015, OBSERVADAS AS CONDICOES LEGAIS.

B16C Correction of notification of the grant [chapter 16.3 patent gazette]

Free format text: REF. RPI 2591 DE 01/09/2020 QUANTO AO TITULO.