BR112016005601B1 - composto, composição farmacêutica, e usos de um composto - Google Patents

composto, composição farmacêutica, e usos de um composto Download PDF

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Publication number
BR112016005601B1
BR112016005601B1 BR112016005601-9A BR112016005601A BR112016005601B1 BR 112016005601 B1 BR112016005601 B1 BR 112016005601B1 BR 112016005601 A BR112016005601 A BR 112016005601A BR 112016005601 B1 BR112016005601 B1 BR 112016005601B1
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BR
Brazil
Prior art keywords
fibrosis
compound
present
pharmaceutically acceptable
weeks
Prior art date
Application number
BR112016005601-9A
Other languages
English (en)
Portuguese (pt)
Other versions
BR112016005601A8 (pt
Inventor
Karen Annette Duggan
Original Assignee
Vectus Biosystems Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from AU2013903573A external-priority patent/AU2013903573A0/en
Application filed by Vectus Biosystems Limited filed Critical Vectus Biosystems Limited
Publication of BR112016005601A8 publication Critical patent/BR112016005601A8/pt
Publication of BR112016005601B1 publication Critical patent/BR112016005601B1/pt

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/02Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/32Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C07C235/34Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07Optical isomers
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/09Geometrical isomers

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BR112016005601-9A 2013-09-17 2014-09-17 composto, composição farmacêutica, e usos de um composto BR112016005601B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
AU2013903573A AU2013903573A0 (en) 2013-09-17 Compositions for the treatment of hypertension and/or fibrosis
AU2013903573 2013-09-17
PCT/AU2014/000923 WO2015039173A1 (en) 2013-09-17 2014-09-17 Compositions for the treatment of hypertension and/or fibrosis

Publications (2)

Publication Number Publication Date
BR112016005601A8 BR112016005601A8 (pt) 2020-02-18
BR112016005601B1 true BR112016005601B1 (pt) 2021-02-02

Family

ID=52687998

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112016005601-9A BR112016005601B1 (pt) 2013-09-17 2014-09-17 composto, composição farmacêutica, e usos de um composto

Country Status (22)

Country Link
US (1) US9458093B2 (enExample)
EP (1) EP3046901B1 (enExample)
JP (1) JP6122548B2 (enExample)
KR (1) KR101736416B1 (enExample)
CN (1) CN105683152B (enExample)
AP (1) AP2016009079A0 (enExample)
AU (1) AU2014324078B2 (enExample)
BR (1) BR112016005601B1 (enExample)
CA (1) CA2924356C (enExample)
DK (1) DK3046901T3 (enExample)
ES (1) ES2655455T3 (enExample)
IL (1) IL244621A (enExample)
MX (1) MX368865B (enExample)
MY (1) MY172557A (enExample)
NO (1) NO3046901T3 (enExample)
NZ (1) NZ717927A (enExample)
PH (1) PH12016500497B1 (enExample)
PL (1) PL3046901T3 (enExample)
RU (1) RU2635564C2 (enExample)
SG (1) SG11201601642WA (enExample)
UA (1) UA118111C2 (enExample)
WO (1) WO2015039173A1 (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3284981B2 (ja) 1998-11-02 2002-05-27 株式会社デンソー 車両用交流発電機およびそのステータの製造方法
US9956166B2 (en) 2013-09-18 2018-05-01 Sorrento Therapeutics, Inc. Methods for administration and methods for treating cardiovascular diseases with resiniferatoxin
JP6734294B2 (ja) * 2015-03-18 2020-08-05 ヴェクタス バイオシステムズ リミテッド 線維症及び線維症に関連する状態の処置のための組成物
JP6716598B2 (ja) * 2015-03-18 2020-07-01 ヴェクタス バイオシステムズ リミテッド 腎臓及び/又は肝臓疾患を治療するための組成物
WO2017049343A1 (en) 2015-09-22 2017-03-30 Vectus Biosystems Limited Synthesis of terphenyl compounds
CN109562096A (zh) * 2016-04-13 2019-04-02 内布拉斯加大学董事会 施用树脂毒素的方法和用树脂毒素治疗心血管疾病的方法
WO2018018091A1 (en) 2016-07-28 2018-02-01 Vectus Biosystems Limited Compositions for the treatment of pulmonary fibrosis

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2694288B1 (fr) * 1992-06-30 1994-09-09 Rhone Poulenc Agrochimie Phenylbenzamides fongicides et procédés pour les préparer.
MXPA06014462A (es) * 2004-06-11 2007-05-23 Vectus Biosystems Ltd Composiciones y metodos para tratamiento de enfermedades cardiovasculares.
RU2466738C2 (ru) * 2005-12-09 2012-11-20 Вектас Байосистемз Лимитед Фрагменты vip и способы их применения
US20120088737A2 (en) 2009-10-02 2012-04-12 Ajinomoto Co., Inc Novel acyl guanidine derivatives
US9630935B2 (en) * 2013-09-17 2017-04-25 Vectus Biosystems Limited Compositions for the treatment of hypertension and/or fibrosis

Also Published As

Publication number Publication date
AU2014324078A1 (en) 2016-04-07
CA2924356A1 (en) 2015-03-26
EP3046901A1 (en) 2016-07-27
EP3046901B1 (en) 2017-10-18
PH12016500497A1 (en) 2016-06-13
SG11201601642WA (en) 2016-04-28
IL244621A (en) 2017-04-30
AU2014324078B2 (en) 2016-12-15
RU2635564C2 (ru) 2017-11-14
ES2655455T3 (es) 2018-02-20
BR112016005601A8 (pt) 2020-02-18
RU2016112257A (ru) 2017-10-20
UA118111C2 (uk) 2018-11-26
CN105683152A (zh) 2016-06-15
DK3046901T3 (en) 2018-01-02
CN105683152B (zh) 2017-03-22
PL3046901T3 (pl) 2018-03-30
WO2015039173A1 (en) 2015-03-26
JP2016532632A (ja) 2016-10-20
NZ717927A (en) 2018-12-21
JP6122548B2 (ja) 2017-04-26
MX368865B (es) 2019-08-02
KR20160074471A (ko) 2016-06-28
MX2016003371A (es) 2016-10-21
IL244621A0 (en) 2016-04-21
KR101736416B1 (ko) 2017-05-16
US20160221933A1 (en) 2016-08-04
PH12016500497B1 (en) 2017-12-13
EP3046901A4 (en) 2017-04-12
CA2924356C (en) 2018-04-03
NO3046901T3 (enExample) 2018-03-17
US9458093B2 (en) 2016-10-04
AP2016009079A0 (en) 2016-03-31
MY172557A (en) 2019-12-02

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Legal Events

Date Code Title Description
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 17/09/2014, OBSERVADAS AS CONDICOES LEGAIS.