BR112014017902A2 - Agente terapêutico ou profilático para doenças causadas por distúrbios do metabolismo de glicose - Google Patents

Agente terapêutico ou profilático para doenças causadas por distúrbios do metabolismo de glicose

Info

Publication number
BR112014017902A2
BR112014017902A2 BR112014017902A BR112014017902A BR112014017902A2 BR 112014017902 A2 BR112014017902 A2 BR 112014017902A2 BR 112014017902 A BR112014017902 A BR 112014017902A BR 112014017902 A BR112014017902 A BR 112014017902A BR 112014017902 A2 BR112014017902 A2 BR 112014017902A2
Authority
BR
Brazil
Prior art keywords
glucose metabolism
therapeutic
prophylactic agent
disorders
diseases caused
Prior art date
Application number
BR112014017902A
Other languages
English (en)
Inventor
Hisatome Ichiro
Tsujimoto Shunsuke
Shirakura Takashi
Hiramitsu Shinya
Original Assignee
Teijin Pharma Limited E National Univ Corporation Tottori Univ
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teijin Pharma Limited E National Univ Corporation Tottori Univ filed Critical Teijin Pharma Limited E National Univ Corporation Tottori Univ
Publication of BR112014017902A2 publication Critical patent/BR112014017902A2/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

AGENTE TERAPÊUTICO OU PROFILÁTICO PARA DOENÇAS CAUSADAS POR DISTÚRBIOS DO METABOLISMO DE GLICOSE. O propósito da presente invenção é prover um novo agente terapêutico ou um novo agente profilático para doenças associadas com metabolismo anormal da glicose. A presente invenção é um agente terapêutico ou um agente profilático para doenças associadas com metabolismo anormal da glicose, que compreende um composto de 2-feniltiazol representado pela fórmula (I) ou um sal farmaceuticamente aceitável do mesmo como um ingrediente ativo.
BR112014017902A 2012-01-27 2013-01-25 Agente terapêutico ou profilático para doenças causadas por distúrbios do metabolismo de glicose BR112014017902A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2012015351 2012-01-27
PCT/JP2013/051627 WO2013111870A1 (ja) 2012-01-27 2013-01-25 糖尿病の治療薬

Publications (1)

Publication Number Publication Date
BR112014017902A2 true BR112014017902A2 (pt) 2017-08-22

Family

ID=48873581

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112014017902A BR112014017902A2 (pt) 2012-01-27 2013-01-25 Agente terapêutico ou profilático para doenças causadas por distúrbios do metabolismo de glicose

Country Status (15)

Country Link
US (1) US20150005506A1 (pt)
EP (1) EP2808018B1 (pt)
JP (1) JP5924699B2 (pt)
KR (1) KR20140134266A (pt)
CN (1) CN104066430A (pt)
AR (1) AR089812A1 (pt)
AU (1) AU2013212865A1 (pt)
BR (1) BR112014017902A2 (pt)
CA (1) CA2862602A1 (pt)
HK (1) HK1201209A1 (pt)
IN (1) IN2014DN05972A (pt)
MX (1) MX2014008484A (pt)
RU (1) RU2014134845A (pt)
TW (1) TW201334779A (pt)
WO (1) WO2013111870A1 (pt)

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* Cited by examiner, † Cited by third party
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CN104610188B (zh) * 2015-02-10 2016-07-27 佛山市赛维斯医药科技有限公司 含苯基脒结构的腈基苯噻唑羧酸酰胺类化合物、其制备及用途
CN104628672A (zh) * 2015-02-10 2015-05-20 佛山市赛维斯医药科技有限公司 一类含苯基脒结构的烷氧苯基噻唑羧酸酰胺类化合物及用途
CN104628673A (zh) * 2015-02-10 2015-05-20 佛山市赛维斯医药科技有限公司 一类含叔丁基脒结构的腈基苯噻唑羧酸酰胺类化合物及用途
CN104610190B (zh) * 2015-02-10 2016-08-17 佛山市赛维斯医药科技有限公司 一类含环丙基脒结构的卤代苯基噻唑羧酸酰胺类化合物及用途
CN104628671B (zh) * 2015-02-10 2016-04-13 佛山市赛维斯医药科技有限公司 含苯基脒结构的硝基苯噻唑羧酸酰胺类化合物及用途
KR102473677B1 (ko) * 2015-08-17 2022-12-02 삼성디스플레이 주식회사 액정 표시 장치
JP6732004B2 (ja) 2016-02-19 2020-07-29 国立大学法人鳥取大学 認知症治療薬または予防薬

Family Cites Families (17)

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DE122008000051I1 (de) 1990-11-30 2009-02-05 Teijin Ltd 2-arylthiazolderivat sowie dieses enthaltendes arzneimittel
HUP9902721A2 (hu) * 1997-11-25 1999-12-28 The Procter & Gamble Co. Tömény textillágyító készítmény és ehhez alkalmazható magas telítetlenségű textillágyító vegyület
US20050074442A1 (en) * 2002-03-13 2005-04-07 Natarajan Ranganathan Compositions and methods for augmenting kidney function
EP1778261A4 (en) * 2004-07-21 2010-08-11 Univ Florida COMPOSITIONS AND METHODS FOR TREATMENT AND DIAGNOSIS OF INSULIN RESISTANCE
AU2006276933A1 (en) * 2005-07-21 2007-02-15 University Of Florida Research Foundation, Inc. Compositions and methods for treatment and prevention of hyperuricemia related health consequences
WO2007019153A2 (en) 2005-08-03 2007-02-15 Tap Pharmaceutical Products, Inc. Methods for treating hypertension
CA2630639A1 (en) * 2005-11-21 2007-05-31 Tap Pharmaceutical Products, Inc. Treatment of qt interval prolongation and diseases associated therewith
JP2007210978A (ja) * 2006-02-13 2007-08-23 Hiroshima Univ 耐糖能障害、ii型糖尿病、高脂血症、メタボリックシンドローム、内臓脂肪型肥満、脂肪肝または非アルコール性脂肪性肝炎の予防・治療剤
EP2101761A4 (en) 2006-11-13 2010-01-27 Takeda Pharmaceuticals North A METHODS FOR PRESERVING RENAL FUNCTION USING XANTHINE OXYDOREDUCTASE INHIBITORS
EP2842948A1 (en) * 2007-11-27 2015-03-04 Ardea Biosciences, Inc. Novel compounds and compositions and methods of use
TWI613203B (zh) * 2008-03-31 2018-02-01 C&C新藥研究所 雜環衍生物
KR101613611B1 (ko) * 2008-04-30 2016-04-19 웰스태트 테러퓨틱스 코포레이션 요산 감소용 테트라졸 화합물
JP5820269B2 (ja) * 2008-05-22 2015-11-24 アストラゼネカ・アクチエボラーグAstrazeneca Aktiebolag Sglt2阻害剤を使用する高尿酸血症の治療方法およびsglt2阻害剤を含有する組成物
CN102256488A (zh) * 2008-10-19 2011-11-23 理查德·J·约翰逊 伴随代谢失衡慢性肾病的治疗组合物和治疗方法
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PE20130574A1 (es) * 2010-06-16 2013-06-01 Takeda Pharmaceuticals Usa Inc Nuevas formas de dosificacion de liberacion modificada de un inhibidor de la xantina oxidorreductasa o de inhibidores de xantina oxidasa
CN102958521A (zh) * 2010-06-25 2013-03-06 帝人制药株式会社 缓释性高血压和肾功能不全治疗剂

Also Published As

Publication number Publication date
IN2014DN05972A (pt) 2015-06-26
CA2862602A1 (en) 2013-08-01
EP2808018A1 (en) 2014-12-03
RU2014134845A (ru) 2016-03-20
EP2808018A4 (en) 2015-07-15
EP2808018B1 (en) 2018-03-14
AR089812A1 (es) 2014-09-17
US20150005506A1 (en) 2015-01-01
WO2013111870A1 (ja) 2013-08-01
JPWO2013111870A1 (ja) 2015-05-11
CN104066430A (zh) 2014-09-24
TW201334779A (zh) 2013-09-01
MX2014008484A (es) 2014-10-14
HK1201209A1 (en) 2015-08-28
JP5924699B2 (ja) 2016-05-25
KR20140134266A (ko) 2014-11-21
AU2013212865A1 (en) 2014-08-14

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]
B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]