BR112014017902A2 - Agente terapêutico ou profilático para doenças causadas por distúrbios do metabolismo de glicose - Google Patents
Agente terapêutico ou profilático para doenças causadas por distúrbios do metabolismo de glicoseInfo
- Publication number
- BR112014017902A2 BR112014017902A2 BR112014017902A BR112014017902A BR112014017902A2 BR 112014017902 A2 BR112014017902 A2 BR 112014017902A2 BR 112014017902 A BR112014017902 A BR 112014017902A BR 112014017902 A BR112014017902 A BR 112014017902A BR 112014017902 A2 BR112014017902 A2 BR 112014017902A2
- Authority
- BR
- Brazil
- Prior art keywords
- glucose metabolism
- therapeutic
- prophylactic agent
- disorders
- diseases caused
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
Landscapes
- Health & Medical Sciences (AREA)
- Diabetes (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
AGENTE TERAPÊUTICO OU PROFILÁTICO PARA DOENÇAS CAUSADAS POR DISTÚRBIOS DO METABOLISMO DE GLICOSE. O propósito da presente invenção é prover um novo agente terapêutico ou um novo agente profilático para doenças associadas com metabolismo anormal da glicose. A presente invenção é um agente terapêutico ou um agente profilático para doenças associadas com metabolismo anormal da glicose, que compreende um composto de 2-feniltiazol representado pela fórmula (I) ou um sal farmaceuticamente aceitável do mesmo como um ingrediente ativo.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2012015351 | 2012-01-27 | ||
PCT/JP2013/051627 WO2013111870A1 (ja) | 2012-01-27 | 2013-01-25 | 糖尿病の治療薬 |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112014017902A2 true BR112014017902A2 (pt) | 2017-08-22 |
Family
ID=48873581
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112014017902A BR112014017902A2 (pt) | 2012-01-27 | 2013-01-25 | Agente terapêutico ou profilático para doenças causadas por distúrbios do metabolismo de glicose |
Country Status (15)
Country | Link |
---|---|
US (1) | US20150005506A1 (pt) |
EP (1) | EP2808018B1 (pt) |
JP (1) | JP5924699B2 (pt) |
KR (1) | KR20140134266A (pt) |
CN (1) | CN104066430A (pt) |
AR (1) | AR089812A1 (pt) |
AU (1) | AU2013212865A1 (pt) |
BR (1) | BR112014017902A2 (pt) |
CA (1) | CA2862602A1 (pt) |
HK (1) | HK1201209A1 (pt) |
IN (1) | IN2014DN05972A (pt) |
MX (1) | MX2014008484A (pt) |
RU (1) | RU2014134845A (pt) |
TW (1) | TW201334779A (pt) |
WO (1) | WO2013111870A1 (pt) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN104610188B (zh) * | 2015-02-10 | 2016-07-27 | 佛山市赛维斯医药科技有限公司 | 含苯基脒结构的腈基苯噻唑羧酸酰胺类化合物、其制备及用途 |
CN104628672A (zh) * | 2015-02-10 | 2015-05-20 | 佛山市赛维斯医药科技有限公司 | 一类含苯基脒结构的烷氧苯基噻唑羧酸酰胺类化合物及用途 |
CN104628673A (zh) * | 2015-02-10 | 2015-05-20 | 佛山市赛维斯医药科技有限公司 | 一类含叔丁基脒结构的腈基苯噻唑羧酸酰胺类化合物及用途 |
CN104610190B (zh) * | 2015-02-10 | 2016-08-17 | 佛山市赛维斯医药科技有限公司 | 一类含环丙基脒结构的卤代苯基噻唑羧酸酰胺类化合物及用途 |
CN104628671B (zh) * | 2015-02-10 | 2016-04-13 | 佛山市赛维斯医药科技有限公司 | 含苯基脒结构的硝基苯噻唑羧酸酰胺类化合物及用途 |
KR102473677B1 (ko) * | 2015-08-17 | 2022-12-02 | 삼성디스플레이 주식회사 | 액정 표시 장치 |
JP6732004B2 (ja) | 2016-02-19 | 2020-07-29 | 国立大学法人鳥取大学 | 認知症治療薬または予防薬 |
Family Cites Families (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE122008000051I1 (de) | 1990-11-30 | 2009-02-05 | Teijin Ltd | 2-arylthiazolderivat sowie dieses enthaltendes arzneimittel |
HUP9902721A2 (hu) * | 1997-11-25 | 1999-12-28 | The Procter & Gamble Co. | Tömény textillágyító készítmény és ehhez alkalmazható magas telítetlenségű textillágyító vegyület |
US20050074442A1 (en) * | 2002-03-13 | 2005-04-07 | Natarajan Ranganathan | Compositions and methods for augmenting kidney function |
EP1778261A4 (en) * | 2004-07-21 | 2010-08-11 | Univ Florida | COMPOSITIONS AND METHODS FOR TREATMENT AND DIAGNOSIS OF INSULIN RESISTANCE |
AU2006276933A1 (en) * | 2005-07-21 | 2007-02-15 | University Of Florida Research Foundation, Inc. | Compositions and methods for treatment and prevention of hyperuricemia related health consequences |
WO2007019153A2 (en) | 2005-08-03 | 2007-02-15 | Tap Pharmaceutical Products, Inc. | Methods for treating hypertension |
CA2630639A1 (en) * | 2005-11-21 | 2007-05-31 | Tap Pharmaceutical Products, Inc. | Treatment of qt interval prolongation and diseases associated therewith |
JP2007210978A (ja) * | 2006-02-13 | 2007-08-23 | Hiroshima Univ | 耐糖能障害、ii型糖尿病、高脂血症、メタボリックシンドローム、内臓脂肪型肥満、脂肪肝または非アルコール性脂肪性肝炎の予防・治療剤 |
EP2101761A4 (en) | 2006-11-13 | 2010-01-27 | Takeda Pharmaceuticals North A | METHODS FOR PRESERVING RENAL FUNCTION USING XANTHINE OXYDOREDUCTASE INHIBITORS |
EP2842948A1 (en) * | 2007-11-27 | 2015-03-04 | Ardea Biosciences, Inc. | Novel compounds and compositions and methods of use |
TWI613203B (zh) * | 2008-03-31 | 2018-02-01 | C&C新藥研究所 | 雜環衍生物 |
KR101613611B1 (ko) * | 2008-04-30 | 2016-04-19 | 웰스태트 테러퓨틱스 코포레이션 | 요산 감소용 테트라졸 화합물 |
JP5820269B2 (ja) * | 2008-05-22 | 2015-11-24 | アストラゼネカ・アクチエボラーグAstrazeneca Aktiebolag | Sglt2阻害剤を使用する高尿酸血症の治療方法およびsglt2阻害剤を含有する組成物 |
CN102256488A (zh) * | 2008-10-19 | 2011-11-23 | 理查德·J·约翰逊 | 伴随代谢失衡慢性肾病的治疗组合物和治疗方法 |
EP2470268A4 (en) * | 2009-08-24 | 2012-12-26 | Wound Man Pty Ltd | PURING-ORIENTED DIAGNOSIS AND THERAPY OF WOUNDS |
PE20130574A1 (es) * | 2010-06-16 | 2013-06-01 | Takeda Pharmaceuticals Usa Inc | Nuevas formas de dosificacion de liberacion modificada de un inhibidor de la xantina oxidorreductasa o de inhibidores de xantina oxidasa |
CN102958521A (zh) * | 2010-06-25 | 2013-03-06 | 帝人制药株式会社 | 缓释性高血压和肾功能不全治疗剂 |
-
2013
- 2013-01-25 EP EP13740913.2A patent/EP2808018B1/en not_active Not-in-force
- 2013-01-25 WO PCT/JP2013/051627 patent/WO2013111870A1/ja active Application Filing
- 2013-01-25 AU AU2013212865A patent/AU2013212865A1/en not_active Abandoned
- 2013-01-25 IN IN5972DEN2014 patent/IN2014DN05972A/en unknown
- 2013-01-25 TW TW102102886A patent/TW201334779A/zh unknown
- 2013-01-25 CN CN201380006730.6A patent/CN104066430A/zh active Pending
- 2013-01-25 RU RU2014134845A patent/RU2014134845A/ru not_active Application Discontinuation
- 2013-01-25 AR ARP130100233A patent/AR089812A1/es unknown
- 2013-01-25 MX MX2014008484A patent/MX2014008484A/es unknown
- 2013-01-25 CA CA2862602A patent/CA2862602A1/en not_active Abandoned
- 2013-01-25 KR KR1020147020342A patent/KR20140134266A/ko not_active Application Discontinuation
- 2013-01-25 BR BR112014017902A patent/BR112014017902A2/pt not_active IP Right Cessation
- 2013-01-25 US US14/372,961 patent/US20150005506A1/en not_active Abandoned
- 2013-01-25 JP JP2013555326A patent/JP5924699B2/ja not_active Expired - Fee Related
-
2015
- 2015-02-25 HK HK15101890.2A patent/HK1201209A1/xx unknown
Also Published As
Publication number | Publication date |
---|---|
IN2014DN05972A (pt) | 2015-06-26 |
CA2862602A1 (en) | 2013-08-01 |
EP2808018A1 (en) | 2014-12-03 |
RU2014134845A (ru) | 2016-03-20 |
EP2808018A4 (en) | 2015-07-15 |
EP2808018B1 (en) | 2018-03-14 |
AR089812A1 (es) | 2014-09-17 |
US20150005506A1 (en) | 2015-01-01 |
WO2013111870A1 (ja) | 2013-08-01 |
JPWO2013111870A1 (ja) | 2015-05-11 |
CN104066430A (zh) | 2014-09-24 |
TW201334779A (zh) | 2013-09-01 |
MX2014008484A (es) | 2014-10-14 |
HK1201209A1 (en) | 2015-08-28 |
JP5924699B2 (ja) | 2016-05-25 |
KR20140134266A (ko) | 2014-11-21 |
AU2013212865A1 (en) | 2014-08-14 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] | ||
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |