BR112012006346A2 - agonista de receptor de acetilcolina, composto, composição farmacêutica, combinação e uso de ativadores de receptor de acetilcolina nicotínico alfa 7 - Google Patents
agonista de receptor de acetilcolina, composto, composição farmacêutica, combinação e uso de ativadores de receptor de acetilcolina nicotínico alfa 7Info
- Publication number
- BR112012006346A2 BR112012006346A2 BR112012006346A BR112012006346A BR112012006346A2 BR 112012006346 A2 BR112012006346 A2 BR 112012006346A2 BR 112012006346 A BR112012006346 A BR 112012006346A BR 112012006346 A BR112012006346 A BR 112012006346A BR 112012006346 A2 BR112012006346 A2 BR 112012006346A2
- Authority
- BR
- Brazil
- Prior art keywords
- acetylcholine receptor
- alpha
- compound
- combination
- pharmaceutical composition
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid, pantothenic acid
- A61K31/198—Alpha-aminoacids, e.g. alanine, edetic acids [EDTA]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
agonista de receptor de acetilcolina, composto, composição farmacêutica, combinação e uso de ativadores de receptor de acetilcolina ninotínico alfa 7 a pres ente invenção se refere ao uso de um ativador de receptor acetilcolina nicotínio alfa 7 para o tratamento, prevenção ou atraso da progressõa da discinesia associada com a terapia com agonista de dopamina na doença de parkinson.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US24465809P | 2009-09-22 | 2009-09-22 | |
PCT/EP2010/063946 WO2011036167A1 (en) | 2009-09-22 | 2010-09-22 | Use of nicotinic acetylcholine receptor alpha 7 activators |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112012006346A2 true BR112012006346A2 (pt) | 2017-05-23 |
Family
ID=42990156
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112012006346A BR112012006346A2 (pt) | 2009-09-22 | 2010-09-22 | agonista de receptor de acetilcolina, composto, composição farmacêutica, combinação e uso de ativadores de receptor de acetilcolina nicotínico alfa 7 |
Country Status (21)
Country | Link |
---|---|
US (3) | US10537539B2 (pt) |
EP (1) | EP2480228B1 (pt) |
JP (2) | JP6178074B2 (pt) |
KR (1) | KR20120068878A (pt) |
CN (2) | CN102573830A (pt) |
AU (1) | AU2010299967B2 (pt) |
BR (1) | BR112012006346A2 (pt) |
CA (1) | CA2774801C (pt) |
CL (1) | CL2012000702A1 (pt) |
EA (1) | EA036742B1 (pt) |
ES (1) | ES2614930T3 (pt) |
IL (1) | IL218299A (pt) |
JO (1) | JO3250B1 (pt) |
MA (1) | MA33590B1 (pt) |
MX (1) | MX359011B (pt) |
NZ (1) | NZ598316A (pt) |
SG (1) | SG178832A1 (pt) |
TN (1) | TN2012000082A1 (pt) |
TW (1) | TWI558398B (pt) |
WO (1) | WO2011036167A1 (pt) |
ZA (1) | ZA201201066B (pt) |
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