BR0315663A - Formulações de depósito de agentes ativos de aril-heterocìclicos na forma de uma suspensão - Google Patents

Formulações de depósito de agentes ativos de aril-heterocìclicos na forma de uma suspensão

Info

Publication number
BR0315663A
BR0315663A BR0315663-0A BR0315663A BR0315663A BR 0315663 A BR0315663 A BR 0315663A BR 0315663 A BR0315663 A BR 0315663A BR 0315663 A BR0315663 A BR 0315663A
Authority
BR
Brazil
Prior art keywords
arylheterocyclic
suspension
active agents
deposit formulations
deposit
Prior art date
Application number
BR0315663-0A
Other languages
English (en)
Inventor
Jaymin Chandrakant Shah
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of BR0315663A publication Critical patent/BR0315663A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/40—Cyclodextrins; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Inorganic Chemistry (AREA)
  • Dermatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Dispersion Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

"FORMULAçõES DE DEPóSITO DE AGENTES ATIVOS DE ARIL-HETEROCìCLICOS NA FORMA DE UMA SUSPENSãO". A presente invenção refere-se a um kit farmacêutico para preparação de uma formulação de depósito injetável de um composto farmacêutico aril-heterocíclico, tal como ziprasidona, e é descrito um método de preparação da referida formulação de depósito.
BR0315663-0A 2002-10-25 2003-10-13 Formulações de depósito de agentes ativos de aril-heterocìclicos na forma de uma suspensão BR0315663A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US42129502P 2002-10-25 2002-10-25
PCT/IB2003/004535 WO2004037224A1 (en) 2002-10-25 2003-10-13 Depot formulations of arylheterocyclic active agents in the form of a suspension

Publications (1)

Publication Number Publication Date
BR0315663A true BR0315663A (pt) 2005-08-30

Family

ID=32176696

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0315663-0A BR0315663A (pt) 2002-10-25 2003-10-13 Formulações de depósito de agentes ativos de aril-heterocìclicos na forma de uma suspensão

Country Status (21)

Country Link
US (1) US20040146562A1 (pt)
EP (1) EP1562546A1 (pt)
JP (2) JP2006505579A (pt)
KR (1) KR20050071611A (pt)
CN (1) CN1703198A (pt)
AR (1) AR041826A1 (pt)
AU (1) AU2003267763A1 (pt)
BR (1) BR0315663A (pt)
CA (1) CA2498276A1 (pt)
GT (1) GT200300227A (pt)
MX (1) MXPA05004299A (pt)
NL (1) NL1024616C (pt)
NO (1) NO20051187L (pt)
PA (1) PA8586301A1 (pt)
PE (1) PE20040471A1 (pt)
PL (1) PL375603A1 (pt)
RU (1) RU2292207C2 (pt)
TW (1) TW200418477A (pt)
UY (1) UY28035A1 (pt)
WO (1) WO2004037224A1 (pt)
ZA (1) ZA200501979B (pt)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20080113025A1 (en) * 1998-11-02 2008-05-15 Elan Pharma International Limited Compositions comprising nanoparticulate naproxen and controlled release hydrocodone
US20040001889A1 (en) 2002-06-25 2004-01-01 Guohua Chen Short duration depot formulations
WO2004017897A2 (en) * 2002-08-20 2004-03-04 Bristol-Myers Squibb Company Aripiprazole complex formulation and method
SI1575569T1 (sl) 2002-12-13 2010-12-31 Durect Corp Oralni sistem dostave zdravila, ki obsega visokoviskozne tekoče nosilne materiale
MXPA05012392A (es) * 2003-05-16 2006-02-02 Pfizer Prod Inc Tratamientos de ansiedad con ziprasidona.
WO2006000913A1 (en) * 2004-06-23 2006-01-05 Pfizer Products Inc. Method for sterile filtration of viscous pharmaceutical compositions
EP2415484B1 (en) 2004-09-17 2014-06-18 Durect Corporation Sustained local anesthetic composition containing SAIB
JP2008531721A (ja) * 2005-03-03 2008-08-14 エラン・ファルマ・インターナショナル・リミテッド 複素環式アミド誘導体のナノ粒子状組成物
US20070027105A1 (en) 2005-07-26 2007-02-01 Alza Corporation Peroxide removal from drug delivery vehicle
CN100391458C (zh) * 2006-02-07 2008-06-04 上海医药工业研究院 齐拉西酮或其盐包合物制备方法
EP2018151A4 (en) * 2006-05-09 2012-07-18 Astrazeneca Ab PARENTERAL FORMULATION COMPRISING AN INHIBITOR OF THE PROTON PUMP STERILIZED IN ITS FINAL CONTAINER BY IONIZING RADIATION
DK2117521T3 (da) 2006-11-03 2012-09-03 Durect Corp Transdermale indgivelsessystemer omfattende bupivacain
CA2706931C (en) * 2007-12-06 2015-05-12 Durect Corporation Oral pharmaceutical dosage forms
US20100260844A1 (en) 2008-11-03 2010-10-14 Scicinski Jan J Oral pharmaceutical dosage forms
EP2983468A4 (en) 2013-03-15 2016-09-07 Durect Corp COMPOSITIONS WITH RHEOLOGY MODIFIER TO REDUCE RESOLUTION VARIABILITY
WO2018153315A1 (zh) * 2017-02-23 2018-08-30 上海华汇拓医药科技有限公司 一种多奈哌齐半帕莫酸盐的粉针剂、包含其的组合物及它们的制备方法
CA3167217A1 (en) 2020-01-13 2021-07-22 Durect Corporation Sustained release drug delivery systems with reduced impurities and related methods

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WO1989002265A1 (en) * 1987-09-07 1989-03-23 Teijin Limited Medicine-containing fat emulsion of the type prepared immediately before use and process for preparing medicine-containing fat emulsion
GB9200247D0 (en) * 1992-01-07 1992-02-26 Erba Carlo Spa Pharmaceutical compositions containing polymer derivative-bound anthracycline glycosides and a method for their preparation
JP3954115B2 (ja) * 1992-07-28 2007-08-08 アストラゼネカ・アクチエボラーグ 注射剤および注射剤キット
US5594141A (en) * 1994-11-23 1997-01-14 Neurogen Corporation Certain aminomethyl biphenyl, aminomethyl phenyl pyridine and aminomethyl phenyl pyrimidine derivatives; novel dopamine receptor subtype selective ligands
US6040295A (en) * 1995-01-13 2000-03-21 Genemedicine, Inc. Formulated nucleic acid compositions and methods of administering the same for gene therapy
UA57734C2 (uk) * 1996-05-07 2003-07-15 Пфайзер Інк. Комплекси включення арилгетероциклічних солей
DK0811386T3 (da) * 1996-05-07 2005-01-03 Pfizer Fremgangsmåde til udvælgelse af et salt til fremstilling af et inklusionskompleks
EP0959873B1 (en) * 1996-12-20 2006-03-01 ALZA Corporation Gel composition and methods
WO1998051348A2 (en) * 1997-05-16 1998-11-19 Amgen Inc. Sustained-release delayed gels
UA72189C2 (uk) * 1997-11-17 2005-02-15 Янссен Фармацевтика Н.В. Фармацевтична композиція, що містить водну суспензію субмікронних ефірів 9-гідроксирисперидон жирних кислот
ES2191618T3 (es) * 1999-05-27 2003-09-16 Pfizer Prod Inc Suspension de ziprasidona.
MY137726A (en) * 2000-11-22 2009-03-31 Nycomed Gmbh Freeze-dried pantoprazole preparation and pantoprazole injection
WO2002074200A1 (en) * 2001-03-20 2002-09-26 Cydex, Inc. Formulations containing propofol and a sulfoalkyl ether cyclodextrin
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AU2002323530B2 (en) * 2001-08-31 2007-09-06 The Rockefeller University Method for classification of anti-psychotic drugs

Also Published As

Publication number Publication date
PA8586301A1 (es) 2004-05-07
JP2006505579A (ja) 2006-02-16
CA2498276A1 (en) 2004-05-06
KR20050071611A (ko) 2005-07-07
AR041826A1 (es) 2005-06-01
WO2004037224A1 (en) 2004-05-06
ZA200501979B (en) 2006-04-26
CN1703198A (zh) 2005-11-30
GT200300227A (es) 2004-06-23
EP1562546A1 (en) 2005-08-17
NL1024616C (nl) 2010-04-19
US20040146562A1 (en) 2004-07-29
NO20051187L (no) 2005-04-11
RU2292207C2 (ru) 2007-01-27
UY28035A1 (es) 2004-05-31
NL1024616A1 (nl) 2004-04-27
AU2003267763A1 (en) 2004-05-13
RU2005112202A (ru) 2005-11-20
TW200418477A (en) 2004-10-01
PL375603A1 (en) 2005-12-12
PE20040471A1 (es) 2004-08-14
MXPA05004299A (es) 2005-08-03
JP2006219501A (ja) 2006-08-24

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 6A,7A E 8A ANUIDADE(S).

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2129 DE 25/10/2011.