MXPA02006029A - Lipopeptidos novedosos como agentes antibacterianos. - Google Patents

Lipopeptidos novedosos como agentes antibacterianos.

Info

Publication number
MXPA02006029A
MXPA02006029A MXPA02006029A MXPA02006029A MXPA02006029A MX PA02006029 A MXPA02006029 A MX PA02006029A MX PA02006029 A MXPA02006029 A MX PA02006029A MX PA02006029 A MXPA02006029 A MX PA02006029A MX PA02006029 A MXPA02006029 A MX PA02006029A
Authority
MX
Mexico
Prior art keywords
compounds
antibacterial agents
novel
novel lipopeptides
relates
Prior art date
Application number
MXPA02006029A
Other languages
English (en)
Inventor
Michael Morytko
Original Assignee
Cubist Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cubist Pharm Inc filed Critical Cubist Pharm Inc
Publication of MXPA02006029A publication Critical patent/MXPA02006029A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Abstract

La presente invencion se relaciona con compuestos lipopeptidicos novedosos. La invencion tambien se relaciona con composiciones farmaceuticas de estos compuestos y los metodos para utilizar estos compuestos como compuestos antibacterianos. La invencion tambien se relaciona con los metodos para producir estos compuestos lipopeptidicos novedosos y los intermediarios utilizados para producir estos compuestos.
MXPA02006029A 1999-12-15 2000-12-15 Lipopeptidos novedosos como agentes antibacterianos. MXPA02006029A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17094399P 1999-12-15 1999-12-15
PCT/US2000/034118 WO2001044272A2 (en) 1999-12-15 2000-12-15 Daptomycin analogs as antibacterial agents

Publications (1)

Publication Number Publication Date
MXPA02006029A true MXPA02006029A (es) 2004-08-23

Family

ID=22621910

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA02006029A MXPA02006029A (es) 1999-12-15 2000-12-15 Lipopeptidos novedosos como agentes antibacterianos.

Country Status (13)

Country Link
US (2) US6911525B2 (es)
EP (4) EP1240181A2 (es)
JP (2) JP4990456B2 (es)
KR (1) KR20020063227A (es)
CN (1) CN1425025A (es)
AU (1) AU784755B2 (es)
BR (1) BR0017026A (es)
CA (1) CA2393907A1 (es)
IL (2) IL150223A0 (es)
MX (1) MXPA02006029A (es)
NO (1) NO20022888L (es)
WO (1) WO2001044272A2 (es)
ZA (1) ZA200205106B (es)

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US20030073647A1 (en) * 2001-08-28 2003-04-17 Chao Robert S. Crystaline clindamycin free base
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WO2003099217A2 (en) * 2002-05-23 2003-12-04 Activbiotics, Inc. Methods of treating bacterial infections and diseases associated therewith
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IL150907A (en) * 2002-07-25 2007-07-04 Stephan Cherkez Process for the preparation of stable amorphous calcium pseudomonate
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US20060004185A1 (en) 2004-07-01 2006-01-05 Leese Richard A Peptide antibiotics and peptide intermediates for their prepartion
US20080051326A1 (en) * 2004-11-12 2008-02-28 Alexander Dylan C Antiinfective Lipopeptides
CA2587848A1 (en) * 2004-11-12 2006-10-19 Cubist Pharmaceuticals, Inc. Antiinfective lipopeptides
WO2006118948A2 (en) * 2005-04-29 2006-11-09 Cubist Pharmaceuticals, Inc. Therapeutic compositions
WO2007127218A2 (en) * 2006-04-26 2007-11-08 Taro Pharmaceuticals U.S.A., Inc. Streptomyces-derived antimicrobial compound and method of using same against antibiotic-resistant bacteria
JP5345532B2 (ja) * 2006-08-02 2013-11-20 ヨハネス・グーテンベルク−ウニヴェルジテート・マインツ Ｌｃｔ中毒に対する医薬品
US8584854B2 (en) * 2007-02-06 2013-11-19 BBK Tobacco & Foods, LLP Reclosable package with magnetic clasp and detachable tray for rolling papers used in smoking articles
US20080185010A1 (en) * 2007-02-06 2008-08-07 Kesselman Joshua D Interleaved Transparent Cellulose Paper with Opaque Adhesive
US8662086B2 (en) 2007-02-06 2014-03-04 BBK Tobacco & Foods, LLP Reclosable package with magnetic clasp for rolling papers used in smoking articles
US20090020443A1 (en) * 2007-05-09 2009-01-22 Kesselman Joshua D Credit Card Carrying Pack for Rolling Papers
US9161572B2 (en) * 2007-06-15 2015-10-20 Bbk Tobacco & Foods, Inc. Structures for creating smoking articles and methods of packaging same
US9072319B2 (en) 2007-06-15 2015-07-07 Joshua D. Kesselman Rolling paper structures for creating smoking articles and gummed, coiled inserts for same
US20090014342A1 (en) * 2007-07-14 2009-01-15 Kesselman Joshua D Rolling papers and methods of packaging same
EP2018864A1 (en) 2007-07-23 2009-01-28 Biomet Deutschland GmbH Pharmaceutical composition, substrate comprising a pharmaceutical composition, and use of a pharmaceutical composition
AU2008343502A1 (en) * 2007-12-26 2009-07-09 Biomarin Pharmaceutical Inc. Novel semi-synthetic glycopeptides as antibacterial agents
US8393332B2 (en) 2008-08-21 2013-03-12 BBK Tobacco & Foods, LLP Packaging for rolling papers for smoking articles
GB2465863A (en) * 2008-12-05 2010-06-09 Lead Therapeutics Inc Semi-synthetic heptapeptidic glycopeptides for the treatment of bacterial infections
EP2379580B1 (en) * 2008-12-22 2013-10-23 Cubist Pharmaceuticals, Inc. Novel antibacterial agents for the treatment of gram positive infections
US8343912B2 (en) 2008-12-23 2013-01-01 Biosource Pharm, Inc. Antibiotic compositions for the treatment of gram negative infections
ES2374779B1 (es) * 2010-03-10 2012-12-27 Universidad De Barcelona Compuestos péptidicos útiles como agentes antibacterianos.
US8415307B1 (en) 2010-06-23 2013-04-09 Biosource Pharm, Inc. Antibiotic compositions for the treatment of gram negative infections
WO2012011917A1 (en) * 2010-07-23 2012-01-26 Activbiotics Pharma, Llc Administration of rifalazil to immunocompromised patients
US10072045B1 (en) 2017-06-26 2018-09-11 Ramapo Pharmaceuticals, Inc. Antibacterial lipopeptides and methods for their preparation and use
US10526343B2 (en) 2018-03-26 2020-01-07 University Of Sharjah Heterocyclic systems and pharmaceutical applications thereof
CN110577581A (zh) * 2018-06-07 2019-12-17 美国蓝博药业公司 一种新型的抑菌脂肽化合物、制备方法及其应用
CN109182563B (zh) * 2018-08-01 2020-07-14 浙江大学 检测20种dfrA类甲氧苄胺嘧啶类药物耐药基因的方法及所用试剂盒
CN113061164B (zh) * 2021-03-29 2023-01-10 四川大学 环脂肽类化合物及其在抗类风湿关节炎药物中的应用

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Also Published As

Publication number Publication date
NO20022888L (no) 2002-08-02
US6911525B2 (en) 2005-06-28
IL150223A0 (en) 2002-12-01
BR0017026A (pt) 2003-01-07
KR20020063227A (ko) 2002-08-01
JP4990456B2 (ja) 2012-08-01
EP1240181A2 (en) 2002-09-18
AU2268201A (en) 2001-06-25
JP2003517004A (ja) 2003-05-20
JP2012140432A (ja) 2012-07-26
NO20022888D0 (no) 2002-06-17
IL150223A (en) 2013-09-30
US7335725B2 (en) 2008-02-26
EP1884520A2 (en) 2008-02-06
ZA200205106B (en) 2003-09-25
WO2001044272A3 (en) 2001-11-29
CA2393907A1 (en) 2001-06-21
EP2295444A2 (en) 2011-03-16
EP2298790A1 (en) 2011-03-23
EP1884520A3 (en) 2008-03-05
CN1425025A (zh) 2003-06-18
AU784755B2 (en) 2006-06-08
US20020025924A1 (en) 2002-02-28
WO2001044272A2 (en) 2001-06-21
US20050203006A1 (en) 2005-09-15
EP2295444A3 (en) 2011-03-23

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