BR0016467A - Lipopeptìdeos como agentes antibacterianos - Google Patents

Lipopeptìdeos como agentes antibacterianos

Info

Publication number
BR0016467A
BR0016467A BR0016467-4A BR0016467A BR0016467A BR 0016467 A BR0016467 A BR 0016467A BR 0016467 A BR0016467 A BR 0016467A BR 0016467 A BR0016467 A BR 0016467A
Authority
BR
Brazil
Prior art keywords
compounds
antibacterial agents
lipopeptides
relates
methods
Prior art date
Application number
BR0016467-4A
Other languages
English (en)
Inventor
Jason Hill
Ian Parr
Michael Morytko
Jim Siedlecki
Xiang Yang Yu
Jared Silverman
Dennis Keith
John Finn
Dale Christensen
Tsvetelina Lazarova
Alan D Watson
Yan Zhang
Original Assignee
Cubist Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cubist Pharm Inc filed Critical Cubist Pharm Inc
Publication of BR0016467A publication Critical patent/BR0016467A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

"LIPOPEPTìDEOS COMO AGENTES ANTIBACTERIANOS". A presente invenção refere-se a novos compostos de lipopeptídeo. A invenção também refere-se a composições farmacêuticas destes compostos e métodos de empregar estes compostos como compostos anti-bacterianos. A invenção também refere-se a métodos de produzir estes novos compostos de lipopeptídeo e intermediários empregados na produção destes compostos.
BR0016467-4A 1999-12-15 2000-12-15 Lipopeptìdeos como agentes antibacterianos BR0016467A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US17094699P 1999-12-15 1999-12-15
US20822200P 2000-05-30 2000-05-30
PCT/US2000/034205 WO2001044274A1 (en) 1999-12-15 2000-12-15 Lipopeptides as antibacterial agents

Publications (1)

Publication Number Publication Date
BR0016467A true BR0016467A (pt) 2002-08-27

Family

ID=26866577

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0016467-4A BR0016467A (pt) 1999-12-15 2000-12-15 Lipopeptìdeos como agentes antibacterianos

Country Status (12)

Country Link
US (3) US7408025B2 (pt)
EP (1) EP1246838A1 (pt)
JP (1) JP2003517480A (pt)
KR (1) KR20020063228A (pt)
CN (1) CN1423656A (pt)
AU (1) AU784812B2 (pt)
BR (1) BR0016467A (pt)
CA (1) CA2394350A1 (pt)
IL (1) IL150225A0 (pt)
MX (1) MXPA02006030A (pt)
NO (1) NO20022887L (pt)
WO (1) WO2001044274A1 (pt)

Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6696412B1 (en) 2000-01-20 2004-02-24 Cubist Pharmaceuticals, Inc. High purity lipopeptides, Lipopeptide micelles and processes for preparing same
US6511962B1 (en) * 2000-07-17 2003-01-28 Micrologix Biotech Inc. Derivatives of laspartomycin and preparation and use thereof
ES2377931T5 (es) 2000-12-18 2015-11-04 Cubist Pharmaceuticals, Inc. Métodos para preparar lipopéptidos purificados
US20060014674A1 (en) 2000-12-18 2006-01-19 Dennis Keith Methods for preparing purified lipopeptides
EP1423414A4 (en) * 2001-08-06 2005-11-30 Cubist Pharm Inc NEW DEPSIPEPTIDES AND METHOD FOR THE PRODUCTION THEREOF
EP1932853A1 (en) 2001-08-06 2008-06-18 Cubist Pharmaceutical Inc. Novel depsipeptides and process for preparing same
US6767718B2 (en) 2002-05-10 2004-07-27 Biosource Pharm, Inc. Lipodepsipeptide antibiotics and methods of preparation
US7317001B2 (en) 2002-06-06 2008-01-08 Oscient Pharmaceuticals Corporation Use of ramoplanin to treat diseases associated with the use of antibiotics
US7521560B2 (en) * 2004-06-29 2009-04-21 Rigel Pharmaceuticals, Inc. 2-substituted quinoline compounds and their uses
US20060004185A1 (en) 2004-07-01 2006-01-05 Leese Richard A Peptide antibiotics and peptide intermediates for their prepartion
FR2874922A1 (fr) * 2004-07-30 2006-03-10 Palumed Sa Molecules hybrides qa ou q est une aminoquinoleine et a est un residu antibiotique, leur synthese et leurs utilisations en tant qu'agent antibacterien
BRPI0514381A (pt) * 2004-07-30 2008-06-10 Palumed Sa compostos hìbridos de aminoquinolina-antibiótico, composições farmacêuticas, método de preparação e uso destes
CA2587848A1 (en) * 2004-11-12 2006-10-19 Cubist Pharmaceuticals, Inc. Antiinfective lipopeptides
US8968781B2 (en) 2005-04-29 2015-03-03 Cubist Pharmaceuticals, Inc. Therapeutic compositions
US7964729B2 (en) 2006-08-28 2011-06-21 Massachusetts Institute Of Technology Sox-based kinase sensor
US8440835B2 (en) 2007-02-26 2013-05-14 Massachusetts Institute Of Technology Environmentally sensitive fluorophores
EP2018864A1 (en) 2007-07-23 2009-01-28 Biomet Deutschland GmbH Pharmaceutical composition, substrate comprising a pharmaceutical composition, and use of a pharmaceutical composition
PT2379580E (pt) * 2008-12-22 2014-01-20 Cubist Pharm Inc Novos agentes antibacterianos para o tratamento de infecções por bactérias gram positivas
TW201035111A (en) 2008-12-23 2010-10-01 Biosource Pharm Inc Antibiotic compositions for the treatment of gram negative infections
WO2011025546A1 (en) 2009-08-31 2011-03-03 Massachusetts Institute Of Technology 1, 2, 3-triazole containing protein kinase sensors
MX2012005993A (es) 2009-11-23 2012-11-23 Cubist Pharm Inc Composiciones de lipopeptido y metodos relacionados.
US8415307B1 (en) 2010-06-23 2013-04-09 Biosource Pharm, Inc. Antibiotic compositions for the treatment of gram negative infections
WO2012011917A1 (en) * 2010-07-23 2012-01-26 Activbiotics Pharma, Llc Administration of rifalazil to immunocompromised patients
US8609672B2 (en) 2010-08-27 2013-12-17 University Of The Pacific Piperazinylpyrimidine analogues as protein kinase inhibitors
US20120317234A1 (en) * 2011-06-09 2012-12-13 International Business Machines Corporation Managing data access in mobile devices
WO2013059610A1 (en) 2011-10-20 2013-04-25 Trius Therapeutics, Inc. Therapeutic combination of daptomycin and protein synthesis inhibitor antibiotic, and methods of use
US9165332B2 (en) * 2012-01-27 2015-10-20 Microsoft Technology Licensing, Llc Application licensing using multiple forms of licensing
US9348608B2 (en) * 2013-04-24 2016-05-24 QRC, Inc. System and method for registering application and application transforms on a radiofrequency digitization and collection device
EP3004892B1 (en) * 2013-05-24 2018-10-10 Nestec S.A. Method for diagnosing irritable bowel syndrome
CN104322562B (zh) * 2014-09-16 2017-04-26 南京农业大学 一种脂肽‑高岭土复合生防制剂及其制备方法和应用
US10647746B2 (en) * 2016-04-08 2020-05-12 Versitech Limited Antibacterial cyclic lipopeptides
US11667674B2 (en) 2016-04-08 2023-06-06 Versitech Limited Antibacterial cyclic lipopeptides
US20200157144A1 (en) * 2017-08-01 2020-05-21 Agency For Science, Technology And Research Antimicrobial peptidomimetics
CA3170514A1 (en) 2020-03-12 2021-09-16 Baxter International Inc. Daptomycin formulations containing a combination of sorbitol and mannitol

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4399067A (en) * 1982-05-21 1983-08-16 Eli Lilly And Company Derivatives of A-21978C cyclic peptides
US4482487A (en) * 1982-05-21 1984-11-13 Eli Lilly And Company A-21978C cyclic peptides
US4524135A (en) * 1982-05-21 1985-06-18 Eli Lilly And Company A-21978C cyclic peptides
US4537717A (en) * 1982-05-21 1985-08-27 Eli Lilly And Company Derivatives of A-21978C cyclic peptides
IL68700A0 (en) * 1982-05-21 1983-09-30 Lilly Co Eli Improvements relating to a-21978c cyclic peptide derivatives and their production
US4396543A (en) * 1982-05-21 1983-08-02 Eli Lilly And Company Derivatives of A-21978C cyclic peptides
USRE32310E (en) 1982-05-21 1986-12-16 Eli Lilly And Company Derivatives of A-21978C cyclic peptides
USRE32311E (en) 1982-05-21 1986-12-16 Eli Lilly And Company Derivatives of A-21978C cyclic peptides
CN1013120B (zh) 1984-10-09 1991-07-10 伊莱利利公司 A-21978c衍生物生产方法改进
CA1315229C (en) 1987-06-10 1993-03-30 Patrick J. Baker Chromatographic purification process
EP0460882B1 (en) * 1990-06-07 1996-07-24 Eli Lilly And Company Lipopeptide deacylase
DE4411025A1 (de) 1994-03-30 1995-10-05 Hoechst Ag Lipopeptid-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung
KR100545506B1 (ko) 1996-03-08 2006-10-04 아스테라스 세이야쿠 가부시키가이샤 환상 리포펩티드 물질의 탈아실화 방법
DE19807972A1 (de) 1998-02-25 1999-08-26 Hoechst Marion Roussel De Gmbh Lipopeptidantibiotika-Calciumsalze, Verfahren zu ihrer Herstellung und Verwendung
AU784942B2 (en) * 1999-12-15 2006-08-03 Cubist Pharmaceuticals, Inc. Daptomycin analogs and their use as antibacterial agents
KR20020063227A (ko) * 1999-12-15 2002-08-01 큐비스트 파마슈티컬즈 인코포레이티드 항균제로서 신규한 리포펩티드

Also Published As

Publication number Publication date
AU784812B2 (en) 2006-06-29
AU3635701A (en) 2001-06-25
US7408025B2 (en) 2008-08-05
WO2001044274A1 (en) 2001-06-21
IL150225A0 (en) 2002-12-01
US20090011977A1 (en) 2009-01-08
CN1423656A (zh) 2003-06-11
MXPA02006030A (es) 2004-08-23
NO20022887L (no) 2002-08-12
EP1246838A1 (en) 2002-10-09
US20040067878A1 (en) 2004-04-08
NO20022887D0 (no) 2002-06-17
KR20020063228A (ko) 2002-08-01
JP2003517480A (ja) 2003-05-27
CA2394350A1 (en) 2001-06-21
US20080287347A1 (en) 2008-11-20

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 5A, 6A, E 7A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1929 DE 26/12/2007.