BR0313178A - Derivados de pirazol e processo para a produção destes - Google Patents

Derivados de pirazol e processo para a produção destes

Info

Publication number
BR0313178A
BR0313178A BR0313178-5A BR0313178A BR0313178A BR 0313178 A BR0313178 A BR 0313178A BR 0313178 A BR0313178 A BR 0313178A BR 0313178 A BR0313178 A BR 0313178A
Authority
BR
Brazil
Prior art keywords
group
haloalkyl
production
derivatives
pyrazole derivatives
Prior art date
Application number
BR0313178-5A
Other languages
English (en)
Other versions
BR0313178B1 (pt
Inventor
Masao Nakatani
Minoru Ito
Masahiro Miyazaki
Original Assignee
Ihara Chemical Ind Co
Kumiai Chemical Industry Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ihara Chemical Ind Co, Kumiai Chemical Industry Co filed Critical Ihara Chemical Ind Co
Publication of BR0313178A publication Critical patent/BR0313178A/pt
Publication of BR0313178B1 publication Critical patent/BR0313178B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5
    • C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms

Abstract

"DERIVADOS DE PIRAZOL E PROCESSO PARA A PRODUçãO DESTES". A presente invenção fornece derivados de pirazol úteis como intermediários de produção para derivados de isoxazolina tendo um excelente efeito herbicida e seletividade entre colheitas e ervas daninhas como processos para produzir os mesmos. Os derivados de pirazol ou sais farmaceuticamente aceitáveis destes que são compostos inventivos são representados pela fórmula geral [1] ou um sal deste: onde R^ 1^ representa um grupo de C1 a C6 alquila, R^ 2^ representa um grupo de C1 a C3 haloalquila, R^ 3^ representa um átomo de hidrogênio, um grupo de C1 a C3 alquila que podem ser substituídos com um ou mais substituintes selecionados do seguinte grupo substituinte <244>, ou um grupo de formila, R^ 4^ representa um átomo de hidrogênio ou um grupo de C1 a C3 haloalquila, contanto que R^ 4^ represente um grupo de C1 a C3 haloalquila no caso em que R^ 3^ é um hidrogênio ou um grupo de formila, e R^ 4^ é um grupo de hidrogênio ou um grupo de C1 a C3 haloalquila no caso em que R^ 3^ é um grupo de C1 a C3 alquila que pode ser substituído com um ou mais substituintes selecionados do seguinte grupo substituinte <244>.
BRPI0313178-5A 2002-08-01 2003-07-31 Derivados de pirazol e processo para a produção destes BR0313178B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2002225083 2002-08-01
JP2002-225083 2002-08-01
PCT/JP2003/009762 WO2004013106A1 (ja) 2002-08-01 2003-07-31 ピラゾール誘導体及びその製造方法

Publications (2)

Publication Number Publication Date
BR0313178A true BR0313178A (pt) 2005-06-14
BR0313178B1 BR0313178B1 (pt) 2014-04-15

Family

ID=31492145

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0313178-5A BR0313178B1 (pt) 2002-08-01 2003-07-31 Derivados de pirazol e processo para a produção destes

Country Status (18)

Country Link
US (2) US7256298B2 (pt)
EP (1) EP1541561B1 (pt)
JP (1) JP4551764B2 (pt)
KR (1) KR101031473B1 (pt)
CN (2) CN100548989C (pt)
AU (1) AU2003252447B2 (pt)
BR (1) BR0313178B1 (pt)
CA (1) CA2494130C (pt)
ES (1) ES2519442T3 (pt)
IL (2) IL166341A (pt)
IN (1) IN2005CH00114A (pt)
MX (1) MX255058B (pt)
PL (1) PL218431B1 (pt)
RS (1) RS53725B1 (pt)
RU (1) RU2315758C2 (pt)
TW (1) TW200409758A (pt)
UA (1) UA79483C2 (pt)
WO (1) WO2004013106A1 (pt)

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MY144905A (en) * 2005-03-17 2011-11-30 Basf Ag Herbicidal compositions based on 3-phenyluracils and 3-sulfonylisoxazolines
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EP2065374A1 (de) 2007-11-30 2009-06-03 Bayer CropScience AG 2-(Benzyl- und 1H-pyrazol-4-ylmethyl)sulfinyl-Thiazol-Derivate als Herbizide und Pflanzenwachstumsregulatoren
EP2112143A1 (de) 2008-04-22 2009-10-28 Bayer CropScience AG 2-(Benzylsulfonyl)-Oxazol-Derivate, chirale 2-(Benzylsulfinyl)-Oxazol-Derivate 2-(Benzylsulfanyl-Oxazol Derivate, Verfahren zu deren Herstellung sowie deren Verwendung als Herbizide und Pflanzenwachstumsregulatoren
EP2112149A1 (de) 2008-04-22 2009-10-28 Bayer CropScience Aktiengesellschaft 2-[(1h-Pyrazol-4-ylmethyl)-sulfonyl]-Oxazol-Derivate, 2-[(1H-Pyrazol-4-ylmethyl)-sulfanyl]-Oxazol-Derivate und chirale 2-[(1H-Pyrazol-4-ylmethyl)-sulfinyl]-Oxazol-Derivate, Verfahren zu deren Herstellung sowie deren Verwendung als Herbizide und Pflanzenwachstumsregulatoren
BR112012029363B1 (pt) * 2010-05-20 2018-04-17 Bayer Intellectual Property Gmbh Processo para preparar 1-alquil-3-difluorometil-5 -hidroxipirazóis
CN103145768B (zh) * 2013-03-06 2016-02-10 陕西科技大学 一种制备二茂铁甲醛的方法
BR112017003295A2 (pt) 2014-09-19 2018-01-23 Isagro Spa 1,3,4-tiadiazóis com uma atividade herbicida, suas composições agronômicas e uso relativo
EP3317254B1 (en) * 2015-11-16 2018-10-03 Lonza Ltd Method for preparation of 1-methyl-3-(trifluoromethyl)-1hpyrazol-5-ol
RU2642924C1 (ru) * 2017-03-13 2018-01-30 Федеральное государственное бюджетное учреждение науки Институт органического синтеза им. И.Я. Постовского Уральского отделения Российской академии наук (ИОС УрО РАН) Способ получения 5-фенил-3-(трифторметил)-1н-пиразол-4-амина
CN109796408B (zh) * 2019-01-21 2022-04-15 江苏中旗科技股份有限公司 一种5-二氟甲氧基-3-三氟甲基-1-甲基吡唑的合成方法
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EP4114833A1 (en) 2020-03-05 2023-01-11 Adama Agan Ltd. Process and intermediates for the preparation of pyroxasulfone
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CN112110912B (zh) * 2020-07-31 2022-07-05 绍兴贝斯美化工股份有限公司 一种合成硫醚类中间体的方法
WO2022137370A1 (ja) * 2020-12-23 2022-06-30 クミアイ化学工業株式会社 スルホン誘導体の製造方法
US20240065269A1 (en) * 2021-01-19 2024-02-29 Kumiai Chemical Industry Co., Ltd. Method for controlling weeds
AU2022211738A1 (en) * 2021-01-19 2023-08-24 Kumiai Chemical Industry Co., Ltd. Method for controlling weeds
GB2603771A (en) * 2021-02-11 2022-08-17 Rotam Agrochem Int Co Ltd Novel crystalline form of pyroxa-sulfone, methods for its preparation and use of the same
JP7232567B1 (ja) * 2021-10-29 2023-03-03 クミアイ化学工業株式会社 ジスルフィド化合物、ポリスルフィド化合物及びその用途
WO2023074828A1 (ja) 2021-10-29 2023-05-04 クミアイ化学工業株式会社 ジスルフィド化合物、ポリスルフィド化合物及びその用途
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Also Published As

Publication number Publication date
IL196010A0 (en) 2011-08-01
CN1995021B (zh) 2010-09-08
MX255058B (es) 2008-03-04
EP1541561A1 (en) 2005-06-15
AU2003252447B2 (en) 2008-06-05
CN1995021A (zh) 2007-07-11
IL166341A (en) 2010-12-30
EP1541561A4 (en) 2007-04-25
RU2005105585A (ru) 2005-08-27
US20070249844A1 (en) 2007-10-25
BR0313178B1 (pt) 2014-04-15
EP1541561B1 (en) 2014-07-23
RS20050081A (en) 2007-09-21
CA2494130C (en) 2011-08-23
RS53725B1 (sr) 2015-06-30
IL166341A0 (en) 2006-01-16
UA79483C2 (en) 2007-06-25
RU2315758C2 (ru) 2008-01-27
US7256298B2 (en) 2007-08-14
ES2519442T3 (es) 2014-11-07
JPWO2004013106A1 (ja) 2006-09-21
TWI337997B (pt) 2011-03-01
PL375319A1 (en) 2005-11-28
KR101031473B1 (ko) 2011-04-26
PL218431B1 (pl) 2014-12-31
CN1678588A (zh) 2005-10-05
IN2005CH00114A (pt) 2007-09-07
MXPA05001258A (es) 2005-04-28
WO2004013106A1 (ja) 2004-02-12
AU2003252447A1 (en) 2004-02-23
JP4551764B2 (ja) 2010-09-29
CN100548989C (zh) 2009-10-14
CA2494130A1 (en) 2004-02-12
KR20050026082A (ko) 2005-03-14
US20050215797A1 (en) 2005-09-29
TW200409758A (en) 2004-06-16

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 15/04/2014, OBSERVADAS AS CONDICOES LEGAIS.