BR0311343A - Derivados de piridazina - Google Patents
Derivados de piridazinaInfo
- Publication number
- BR0311343A BR0311343A BR0311343-4A BR0311343A BR0311343A BR 0311343 A BR0311343 A BR 0311343A BR 0311343 A BR0311343 A BR 0311343A BR 0311343 A BR0311343 A BR 0311343A
- Authority
- BR
- Brazil
- Prior art keywords
- pyridazine derivatives
- pyridazine
- diseases
- cachexia
- phosphodiesterase
- Prior art date
Links
- 150000004892 pyridazines Chemical class 0.000 title abstract 2
- 208000030507 AIDS Diseases 0.000 abstract 1
- 201000001320 Atherosclerosis Diseases 0.000 abstract 1
- 208000023275 Autoimmune disease Diseases 0.000 abstract 1
- 206010006895 Cachexia Diseases 0.000 abstract 1
- 208000031229 Cardiomyopathies Diseases 0.000 abstract 1
- 206010020751 Hypersensitivity Diseases 0.000 abstract 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 208000001132 Osteoporosis Diseases 0.000 abstract 1
- 229940123932 Phosphodiesterase 4 inhibitor Drugs 0.000 abstract 1
- 230000007815 allergy Effects 0.000 abstract 1
- 208000006673 asthma Diseases 0.000 abstract 1
- 206010012601 diabetes mellitus Diseases 0.000 abstract 1
- 230000004054 inflammatory process Effects 0.000 abstract 1
- 201000006417 multiple sclerosis Diseases 0.000 abstract 1
- 239000002587 phosphodiesterase IV inhibitor Substances 0.000 abstract 1
- PBMFSQRYOILNGV-UHFFFAOYSA-N pyridazine Chemical class C1=CC=NN=C1 PBMFSQRYOILNGV-UHFFFAOYSA-N 0.000 abstract 1
- 206010039073 rheumatoid arthritis Diseases 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
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-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Virology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Oncology (AREA)
- Pulmonology (AREA)
- Communicable Diseases (AREA)
- Physical Education & Sports Medicine (AREA)
- Diabetes (AREA)
- Immunology (AREA)
- Cardiology (AREA)
- Rheumatology (AREA)
- Molecular Biology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Hematology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Dermatology (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Ophthalmology & Optometry (AREA)
- Endocrinology (AREA)
- Hospice & Palliative Care (AREA)
- Psychology (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10224888A DE10224888A1 (de) | 2002-06-05 | 2002-06-05 | Pyridazinderivate |
| PCT/EP2003/004930 WO2003104204A1 (de) | 2002-06-05 | 2003-05-12 | Pyridazinderivate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0311343A true BR0311343A (pt) | 2005-03-22 |
Family
ID=29594275
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0311343-4A BR0311343A (pt) | 2002-06-05 | 2003-05-12 | Derivados de piridazina |
Country Status (17)
| Country | Link |
|---|---|
| US (2) | US7129241B2 (enExample) |
| EP (1) | EP1509506B1 (enExample) |
| JP (1) | JP4511925B2 (enExample) |
| KR (1) | KR20050009735A (enExample) |
| CN (1) | CN1659147A (enExample) |
| AR (1) | AR040141A1 (enExample) |
| AT (1) | ATE438628T1 (enExample) |
| AU (1) | AU2003227746B2 (enExample) |
| BR (1) | BR0311343A (enExample) |
| CA (1) | CA2488372C (enExample) |
| DE (2) | DE10224888A1 (enExample) |
| ES (1) | ES2329670T3 (enExample) |
| MX (1) | MXPA04012009A (enExample) |
| PL (1) | PL371918A1 (enExample) |
| RU (1) | RU2004139032A (enExample) |
| WO (1) | WO2003104204A1 (enExample) |
| ZA (1) | ZA200500071B (enExample) |
Families Citing this family (70)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW200519106A (en) | 2003-05-02 | 2005-06-16 | Novartis Ag | Organic compounds |
| GB0401334D0 (en) | 2004-01-21 | 2004-02-25 | Novartis Ag | Organic compounds |
| GB0411056D0 (en) | 2004-05-18 | 2004-06-23 | Novartis Ag | Organic compounds |
| GT200500281A (es) | 2004-10-22 | 2006-04-24 | Novartis Ag | Compuestos organicos. |
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| DE19632549A1 (de) | 1996-08-13 | 1998-02-19 | Merck Patent Gmbh | Arylalkanoylpyridazine |
| DE19826841A1 (de) * | 1998-06-16 | 1999-12-23 | Merck Patent Gmbh | Arylalkanoylpyridazine |
| DE19915364A1 (de) * | 1999-04-06 | 2000-10-12 | Merck Patent Gmbh | Verwendung von Arylalkanoylpyridazinen |
| WO2001057025A1 (en) * | 2000-01-31 | 2001-08-09 | Pfizer Products Inc. | Pyrimidine carboxamides useful as inhibitors of pde4 isozymes |
-
2002
- 2002-06-05 DE DE10224888A patent/DE10224888A1/de not_active Withdrawn
-
2003
- 2003-05-12 PL PL03371918A patent/PL371918A1/xx unknown
- 2003-05-12 DE DE50311783T patent/DE50311783D1/de not_active Expired - Lifetime
- 2003-05-12 JP JP2004511274A patent/JP4511925B2/ja not_active Expired - Fee Related
- 2003-05-12 BR BR0311343-4A patent/BR0311343A/pt not_active Application Discontinuation
- 2003-05-12 CA CA2488372A patent/CA2488372C/en not_active Expired - Fee Related
- 2003-05-12 MX MXPA04012009A patent/MXPA04012009A/es not_active Application Discontinuation
- 2003-05-12 AU AU2003227746A patent/AU2003227746B2/en not_active Ceased
- 2003-05-12 EP EP03725186A patent/EP1509506B1/de not_active Expired - Lifetime
- 2003-05-12 US US10/516,876 patent/US7129241B2/en not_active Expired - Fee Related
- 2003-05-12 KR KR10-2004-7019787A patent/KR20050009735A/ko not_active Withdrawn
- 2003-05-12 ES ES03725186T patent/ES2329670T3/es not_active Expired - Lifetime
- 2003-05-12 CN CN038128470A patent/CN1659147A/zh active Pending
- 2003-05-12 RU RU2004139032/04A patent/RU2004139032A/ru not_active Application Discontinuation
- 2003-05-12 AT AT03725186T patent/ATE438628T1/de not_active IP Right Cessation
- 2003-05-12 WO PCT/EP2003/004930 patent/WO2003104204A1/de not_active Ceased
- 2003-06-04 AR ARP030101978A patent/AR040141A1/es not_active Application Discontinuation
-
2005
- 2005-01-04 ZA ZA200500071A patent/ZA200500071B/en unknown
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2006
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Also Published As
| Publication number | Publication date |
|---|---|
| ATE438628T1 (de) | 2009-08-15 |
| CA2488372A1 (en) | 2003-12-18 |
| ES2329670T3 (es) | 2009-11-30 |
| AU2003227746B2 (en) | 2009-03-19 |
| AR040141A1 (es) | 2005-03-16 |
| US20060270681A1 (en) | 2006-11-30 |
| US7129241B2 (en) | 2006-10-31 |
| CN1659147A (zh) | 2005-08-24 |
| WO2003104204A1 (de) | 2003-12-18 |
| RU2004139032A (ru) | 2005-08-20 |
| PL371918A1 (en) | 2005-07-11 |
| DE10224888A1 (de) | 2003-12-24 |
| ZA200500071B (en) | 2006-07-26 |
| US7563790B2 (en) | 2009-07-21 |
| JP2005534660A (ja) | 2005-11-17 |
| US20050176714A1 (en) | 2005-08-11 |
| EP1509506A1 (de) | 2005-03-02 |
| KR20050009735A (ko) | 2005-01-25 |
| DE50311783D1 (de) | 2009-09-17 |
| AU2003227746A1 (en) | 2003-12-22 |
| JP4511925B2 (ja) | 2010-07-28 |
| CA2488372C (en) | 2012-02-21 |
| EP1509506B1 (de) | 2009-08-05 |
| MXPA04012009A (es) | 2005-03-07 |
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