BR0210838A - Composto, formulação farmacêutica, uso de um composto, métodos de prevenção e/ou tratamento de condições associadas com glicogênio sintase quinase-3, e de doenças, e medicação contraceptiva, e, processos para a preparação de um composto - Google Patents
Composto, formulação farmacêutica, uso de um composto, métodos de prevenção e/ou tratamento de condições associadas com glicogênio sintase quinase-3, e de doenças, e medicação contraceptiva, e, processos para a preparação de um compostoInfo
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- BR0210838A BR0210838A BR0210838-0A BR0210838A BR0210838A BR 0210838 A BR0210838 A BR 0210838A BR 0210838 A BR0210838 A BR 0210838A BR 0210838 A BR0210838 A BR 0210838A
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/36—Radicals substituted by singly-bound nitrogen atoms
- C07D213/42—Radicals substituted by singly-bound nitrogen atoms having hetero atoms attached to the substituent nitrogen atom
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- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
Abstract
"COMPOSTO, FORMULAçãO FARMACêUTICA, USO DE UM COMPOSTO, MéTODOS DE PREVENçãO E/OU TRATAMENTO DE CONDIçõES ASSOCIADAS COM GLICOGêNIO SINTASE QUINASE-3, E DE DOENçAS, E MEDICAçãO CONTRACEPTIVA, E, PROCESSOS PARA A PREPARAçãO DE UM COMPOSTO". A presente invenção diz respeito a novos compostos da fórmula (1) em que Z, Y, X, P, Q, R, R^ 1^, R^ 2^, R^ 3^, R^ 4^, R^ 5^, R^ 6^, R^ 7^, R^ 8^, R^ 9^, R^ 10^, R^ 11^, R^ 12^, A, m e n são como definidos em qualquer uma das reivindicação de 1 a 3, um processo para sua preparação e novos intermediários preparados neste, composições farmacêuticas contendo os ditos compostos terapeuticamente ativos e ao uso dos ditos compostos ativos na terapia.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE0102439A SE0102439D0 (sv) | 2001-07-05 | 2001-07-05 | New compounds |
PCT/SE2002/001339 WO2003004472A1 (en) | 2001-07-05 | 2002-07-03 | Arylamines for the treatment of conditions associated with gsk-3 |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0210838A true BR0210838A (pt) | 2004-07-13 |
Family
ID=20284777
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0210838-0A BR0210838A (pt) | 2001-07-05 | 2002-07-03 | Composto, formulação farmacêutica, uso de um composto, métodos de prevenção e/ou tratamento de condições associadas com glicogênio sintase quinase-3, e de doenças, e medicação contraceptiva, e, processos para a preparação de um composto |
Country Status (19)
Country | Link |
---|---|
US (1) | US20060052396A1 (pt) |
EP (1) | EP1414801A1 (pt) |
JP (1) | JP2005505515A (pt) |
KR (1) | KR20040013102A (pt) |
CN (1) | CN1551869A (pt) |
AR (1) | AR036132A1 (pt) |
BR (1) | BR0210838A (pt) |
CA (1) | CA2452686A1 (pt) |
CO (1) | CO5540341A2 (pt) |
HU (1) | HUP0500339A2 (pt) |
IL (1) | IL159347A0 (pt) |
IS (1) | IS7095A (pt) |
MX (1) | MXPA03011972A (pt) |
NO (1) | NO20040014L (pt) |
PL (1) | PL367782A1 (pt) |
RU (1) | RU2004102389A (pt) |
SE (1) | SE0102439D0 (pt) |
WO (1) | WO2003004472A1 (pt) |
ZA (1) | ZA200309977B (pt) |
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DE69302168T2 (de) * | 1992-01-28 | 1996-09-05 | Kloeckner Haensel Tevopharm | Verfahren und vorrichtung zur manipulation eines produktstromes |
MA26473A1 (fr) * | 1997-03-01 | 2004-12-20 | Glaxo Group Ltd | Composes pharmacologiquement actifs. |
DZ3293A1 (fr) * | 2000-02-16 | 2001-08-23 | Neurogen Corp | Arylpyrazines substitues |
AR029489A1 (es) * | 2000-03-10 | 2003-07-02 | Euro Celtique Sa | Piridinas, pirimidinas, pirazinas, triazinas sustituidas por arilo, composiciones farmaceuticas y el uso de las mismas para la manufactura de un medicamento |
-
2001
- 2001-07-05 SE SE0102439A patent/SE0102439D0/xx unknown
-
2002
- 2002-07-03 RU RU2004102389/04A patent/RU2004102389A/ru not_active Application Discontinuation
- 2002-07-03 BR BR0210838-0A patent/BR0210838A/pt not_active Application Discontinuation
- 2002-07-03 CA CA002452686A patent/CA2452686A1/en not_active Abandoned
- 2002-07-03 IL IL15934702A patent/IL159347A0/xx unknown
- 2002-07-03 HU HU0500339A patent/HUP0500339A2/hu unknown
- 2002-07-03 CN CNA028135458A patent/CN1551869A/zh active Pending
- 2002-07-03 WO PCT/SE2002/001339 patent/WO2003004472A1/en not_active Application Discontinuation
- 2002-07-03 MX MXPA03011972A patent/MXPA03011972A/es unknown
- 2002-07-03 EP EP02747795A patent/EP1414801A1/en not_active Withdrawn
- 2002-07-03 US US10/481,721 patent/US20060052396A1/en not_active Abandoned
- 2002-07-03 JP JP2003510640A patent/JP2005505515A/ja active Pending
- 2002-07-03 KR KR10-2004-7000080A patent/KR20040013102A/ko not_active Application Discontinuation
- 2002-07-03 PL PL02367782A patent/PL367782A1/xx not_active Application Discontinuation
- 2002-07-05 AR ARP020102533A patent/AR036132A1/es unknown
-
2003
- 2003-12-23 ZA ZA200309977A patent/ZA200309977B/xx unknown
- 2003-12-30 CO CO03113306A patent/CO5540341A2/es not_active Application Discontinuation
- 2003-12-31 IS IS7095A patent/IS7095A/is unknown
-
2004
- 2004-01-02 NO NO20040014A patent/NO20040014L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
IL159347A0 (en) | 2004-06-01 |
AR036132A1 (es) | 2004-08-11 |
EP1414801A1 (en) | 2004-05-06 |
JP2005505515A (ja) | 2005-02-24 |
MXPA03011972A (es) | 2004-03-26 |
HUP0500339A2 (hu) | 2005-07-28 |
CN1551869A (zh) | 2004-12-01 |
PL367782A1 (en) | 2005-03-07 |
NO20040014L (no) | 2004-03-02 |
SE0102439D0 (sv) | 2001-07-05 |
KR20040013102A (ko) | 2004-02-11 |
IS7095A (is) | 2003-12-31 |
WO2003004472A1 (en) | 2003-01-16 |
WO2003004472A8 (en) | 2003-03-13 |
CO5540341A2 (es) | 2005-07-29 |
CA2452686A1 (en) | 2003-01-16 |
US20060052396A1 (en) | 2006-03-09 |
RU2004102389A (ru) | 2005-07-10 |
ZA200309977B (en) | 2005-03-23 |
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