BR0113886A - Composição, composição farmacêutica, tratamento de combinação para prevenir ou inibir a geração ou atividade de trombina num paciente, método para inibir ou prevenir a geração ou atividade de trombina num paciente, uso de uma composição ou tratamento de combinação, uso de uma composição, uso e kit - Google Patents

Composição, composição farmacêutica, tratamento de combinação para prevenir ou inibir a geração ou atividade de trombina num paciente, método para inibir ou prevenir a geração ou atividade de trombina num paciente, uso de uma composição ou tratamento de combinação, uso de uma composição, uso e kit

Info

Publication number
BR0113886A
BR0113886A BR0113886-3A BR0113886A BR0113886A BR 0113886 A BR0113886 A BR 0113886A BR 0113886 A BR0113886 A BR 0113886A BR 0113886 A BR0113886 A BR 0113886A
Authority
BR
Brazil
Prior art keywords
composition
activity
preventing
patient
inhibiting
Prior art date
Application number
BR0113886-3A
Other languages
English (en)
Inventor
Jack Hirsh
Kristian Johansen
Jeffery I Weitz
Original Assignee
Hamilton Civic Hospitals Res
Leo Pharma As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hamilton Civic Hospitals Res, Leo Pharma As filed Critical Hamilton Civic Hospitals Res
Publication of BR0113886A publication Critical patent/BR0113886A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/715—Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
    • A61K31/726—Glycosaminoglycans, i.e. mucopolysaccharides
    • A61K31/727—Heparin; Heparan
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/715—Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
    • A61K31/737—Sulfated polysaccharides, e.g. chondroitin sulfate, dermatan sulfate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/55—Protease inhibitors
    • A61K38/57—Protease inhibitors from animals; from humans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Molecular Biology (AREA)
  • Dermatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Zoology (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Materials For Medical Uses (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

"COMPOSIçãO, COMPOSIçãO FARMACêUTICA, TRATAMENTO DE COMBINAçãO PARA PREVENIR OU INIBIR A GERAçãO OU ATIVIDADE DE TROMBINA NUM PACIENTE, MéTODO PARA INIBIR OU PREVENIR A GERAçãO OU ATIVIDADE DE TROMBINA NUM PACIENTE, USO DE UMA COMPOSIçãO OU TRATAMENTO DE COMBINAçãO, USO DE UMA COMPOSIçãO, USO E KIT". A presente invenção refere-se, de forma geral, a composições e métodos para prevenir ou inibir a atividade ou geração de trombina.
BR0113886-3A 2000-09-08 2001-09-07 Composição, composição farmacêutica, tratamento de combinação para prevenir ou inibir a geração ou atividade de trombina num paciente, método para inibir ou prevenir a geração ou atividade de trombina num paciente, uso de uma composição ou tratamento de combinação, uso de uma composição, uso e kit BR0113886A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23142900P 2000-09-08 2000-09-08
PCT/CA2001/001287 WO2002020091A2 (en) 2000-09-08 2001-09-07 Antithrombotic compositions

Publications (1)

Publication Number Publication Date
BR0113886A true BR0113886A (pt) 2003-07-15

Family

ID=22869211

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0113886-3A BR0113886A (pt) 2000-09-08 2001-09-07 Composição, composição farmacêutica, tratamento de combinação para prevenir ou inibir a geração ou atividade de trombina num paciente, método para inibir ou prevenir a geração ou atividade de trombina num paciente, uso de uma composição ou tratamento de combinação, uso de uma composição, uso e kit

Country Status (15)

Country Link
US (1) US20040038932A1 (pt)
EP (1) EP1315539A2 (pt)
JP (1) JP2004507562A (pt)
KR (1) KR20030069990A (pt)
CN (1) CN1473061A (pt)
AU (1) AU2001291549A1 (pt)
BR (1) BR0113886A (pt)
CA (1) CA2420890A1 (pt)
CZ (1) CZ2003961A3 (pt)
HK (1) HK1052315A1 (pt)
HU (1) HUP0300939A2 (pt)
IL (1) IL154771A0 (pt)
MX (1) MXPA03001986A (pt)
PL (1) PL363047A1 (pt)
WO (1) WO2002020091A2 (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003018032A1 (en) * 2001-08-28 2003-03-06 Leo Pharma A/S Antithrombotic compositions comprising low molecular weight heparin and low molecular weight dermatan sulphate
US20040171819A1 (en) 2002-10-10 2004-09-02 Aventis Pharma S.A. Mixtures of polysaccharides derived from heparin, their preparation and pharmaceutical compositions containing them
US20050261241A1 (en) 2004-05-19 2005-11-24 Celsus Biopharmaceuticals, Inc. Use of dermatan sulfates and/or desulfated heparins to treat or prevent heparinoid-induced autoimmune responses
GB2433592A (en) 2005-12-23 2007-06-27 Pentapharm Ag Assay for thrombin inhibitors
CN101724016B (zh) * 2008-10-28 2013-09-25 上海医药工业研究院 一类肽化合物、其制备方法及用途

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Also Published As

Publication number Publication date
CA2420890A1 (en) 2002-03-14
CZ2003961A3 (cs) 2003-10-15
JP2004507562A (ja) 2004-03-11
IL154771A0 (en) 2003-10-31
KR20030069990A (ko) 2003-08-27
WO2002020091A3 (en) 2002-11-21
HK1052315A1 (zh) 2003-09-11
EP1315539A2 (en) 2003-06-04
CN1473061A (zh) 2004-02-04
HUP0300939A2 (hu) 2003-09-29
AU2001291549A1 (en) 2002-03-22
WO2002020091A2 (en) 2002-03-14
PL363047A1 (en) 2004-11-15
US20040038932A1 (en) 2004-02-26
MXPA03001986A (es) 2004-03-19

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Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]
B15K Others concerning applications: alteration of classification

Ipc: A61K 31/727 (2006.01), A61P 7/02 (2006.01), A61K 3