BR0113602A - Processo para preparar um composto de imidazopiridina substituìda - Google Patents

Processo para preparar um composto de imidazopiridina substituìda

Info

Publication number
BR0113602A
BR0113602A BR0113602-0A BR0113602A BR0113602A BR 0113602 A BR0113602 A BR 0113602A BR 0113602 A BR0113602 A BR 0113602A BR 0113602 A BR0113602 A BR 0113602A
Authority
BR
Brazil
Prior art keywords
preparing
compound
substituted imidazopyridine
imidazopyridine compound
formula
Prior art date
Application number
BR0113602-0A
Other languages
English (en)
Inventor
Bj Rn Elman
Silke Erback
Eric Thiemermann
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of BR0113602A publication Critical patent/BR0113602A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

"PROCESSO PARA PREPARAR UM COMPOSTO DE IMIDAZOPIRIDINA SUBSTITUìDA". A presente invenção prove um novo processo para a preparação em grande escala de um composto de imidazopiridina substituída da fórmula (I), em que R^ 1^ é um grupo alcóxi C~ 1~-C~ 6~ ou NH~ 2~, que compreende o estágio de reagir um composto da fórmula (2) com um composto de 3-halo-2-butanona em ciclo-hexanona.
BR0113602-0A 2000-09-07 2001-09-05 Processo para preparar um composto de imidazopiridina substituìda BR0113602A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0003186A SE0003186D0 (sv) 2000-09-07 2000-09-07 New process
PCT/SE2001/001897 WO2002020523A1 (en) 2000-09-07 2001-09-05 Process for preparing a substituted imidazopyridine compound

Publications (1)

Publication Number Publication Date
BR0113602A true BR0113602A (pt) 2003-07-15

Family

ID=20280942

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0113602-0A BR0113602A (pt) 2000-09-07 2001-09-05 Processo para preparar um composto de imidazopiridina substituìda

Country Status (27)

Country Link
US (2) US20060063797A1 (pt)
EP (1) EP1317455B9 (pt)
JP (1) JP4157766B2 (pt)
KR (1) KR100770478B1 (pt)
CN (1) CN1255404C (pt)
AT (1) ATE272637T1 (pt)
AU (2) AU8459401A (pt)
BR (1) BR0113602A (pt)
CA (1) CA2419764C (pt)
CZ (1) CZ294957B6 (pt)
DE (1) DE60104704T2 (pt)
EE (1) EE05136B1 (pt)
ES (1) ES2223906T3 (pt)
HK (1) HK1054388B (pt)
HU (1) HU225459B1 (pt)
IL (2) IL154466A0 (pt)
IS (1) IS2084B (pt)
NO (1) NO324252B1 (pt)
NZ (1) NZ524302A (pt)
PL (1) PL360626A1 (pt)
PT (1) PT1317455E (pt)
RU (1) RU2275372C2 (pt)
SE (1) SE0003186D0 (pt)
SK (1) SK286717B6 (pt)
UA (1) UA73788C2 (pt)
WO (1) WO2002020523A1 (pt)
ZA (1) ZA200301171B (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2293068T3 (es) 2002-09-19 2008-03-16 Schering Corporation Imidazopiridinas como inhibidores de quinasas dependientes de ciclina.
SE0303451D0 (sv) * 2003-12-18 2003-12-18 Astrazeneca Ab New compounds
TWI359122B (en) * 2004-04-16 2012-03-01 Smidth As F L Method and apparatus for hydration of a particulat
FI20086158A0 (fi) * 2008-12-03 2008-12-03 Mikael Dahlstroem Imidatsopyridiinijohdannaiset
ES2573148T3 (es) * 2010-08-25 2016-06-06 Neopharm Co., Ltd. Compuestos y composición de 1H-benzo[d]imidazol-5-ilo para el tratamiento de enfermedades inflamatorias
CN104650079A (zh) * 2015-01-31 2015-05-27 山东友帮生化科技有限公司 一种8-甲氧基咪唑并[1,2a]吡啶-3-甲腈的合成方法
KR101777971B1 (ko) * 2016-07-05 2017-09-12 제일약품주식회사 이미다조[1,2-a]피리딘 유도체, 이의 제조방법 및 이의 용도

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA81219B (en) * 1980-01-23 1982-01-27 Schering Corp Imidazo (1,2-a) pyridines ,process for their preparation and pharmaceutical compositions containing them
US4444775A (en) * 1981-06-22 1984-04-24 Ciba-Geigy Corporation Substituted imidazo[1,5-A]pyridines
DE3269604D1 (en) * 1981-06-26 1986-04-10 Schering Corp Novel imidazo(1,2-a)pyridines and pyrazines, processes for their preparation and pharmaceutical compositions containing them
FR2525602A1 (fr) * 1982-04-21 1983-10-28 Synthelabo Imidazo(1,2-a)pyridines, leur preparation et leur application en therapeutique
US4725601A (en) * 1985-06-04 1988-02-16 Fujisawa Pharmaceutical Co., Ltd. Certain imidazo[1,2-a]pyridines useful in the treatment of ulcers
EP0228006A1 (en) * 1985-12-16 1987-07-08 Fujisawa Pharmaceutical Co., Ltd. Imidazopyridine compounds and processes for preparation thereof
GB8722488D0 (en) * 1987-09-24 1987-10-28 Fujisawa Pharmaceutical Co Imidazopyridine compound
US5798364A (en) * 1992-03-26 1998-08-25 Merck Patent Gesellschaft Mit Beschrankter Haftung Imidazopyridines
IL108520A (en) * 1993-02-15 1997-09-30 Byk Gulden Lomberg Chem Fab 2, 3, 8-TRISUBSTITUTED IMIDAZO £1, 2-a| PYRIDINE DERIVATIVES, PROCESSES FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
SE512531C2 (sv) * 1997-09-04 2000-03-27 Astacarotene Ab Användning av åtminstone en typ av xantofyller för framställning av ett läkemedel för profylaktisk och/eller terapeutisk förbättring av muskelfunktionsdurationen hos däggdjur och/eller behandling av muskelstörningar eller - sjukdomar hos däggdjur
SE9801526D0 (sv) * 1998-04-29 1998-04-29 Astra Ab New compounds
SE9802794D0 (sv) * 1998-08-21 1998-08-21 Astra Ab New compounds
US6900324B2 (en) * 2000-09-07 2005-05-31 Astrazeneca Ab Process for preparing a substituted imidazopyridine compound

Also Published As

Publication number Publication date
PL360626A1 (en) 2004-09-20
ZA200301171B (en) 2004-03-18
CN1255404C (zh) 2006-05-10
CZ294957B6 (cs) 2005-04-13
SK286717B6 (sk) 2009-04-06
KR20030032011A (ko) 2003-04-23
SE0003186D0 (sv) 2000-09-07
EE200300090A (et) 2004-12-15
IS6728A (is) 2003-02-26
CA2419764C (en) 2009-10-06
US20060063797A1 (en) 2006-03-23
HK1054388A1 (en) 2003-11-28
IL154466A0 (en) 2003-09-17
JP2004508371A (ja) 2004-03-18
IS2084B (is) 2006-02-15
NO20031046D0 (no) 2003-03-06
HK1054388B (zh) 2005-04-08
JP4157766B2 (ja) 2008-10-01
AU2001284594B2 (en) 2005-12-15
US20090247755A1 (en) 2009-10-01
WO2002020523A1 (en) 2002-03-14
ATE272637T1 (de) 2004-08-15
RU2275372C2 (ru) 2006-04-27
NZ524302A (en) 2004-08-27
KR100770478B1 (ko) 2007-10-26
CA2419764A1 (en) 2002-03-14
UA73788C2 (en) 2005-09-15
HUP0302277A2 (hu) 2003-10-28
EP1317455B9 (en) 2004-11-17
DE60104704T2 (de) 2005-08-11
CN1452621A (zh) 2003-10-29
EE05136B1 (et) 2009-02-16
DE60104704D1 (de) 2004-09-09
NO20031046L (no) 2003-05-05
AU8459401A (en) 2002-03-22
EP1317455B1 (en) 2004-08-04
NO324252B1 (no) 2007-09-17
IL154466A (en) 2009-06-15
HU225459B1 (en) 2006-12-28
HUP0302277A3 (en) 2003-12-29
SK2702003A3 (en) 2003-08-05
EP1317455A1 (en) 2003-06-11
ES2223906T3 (es) 2005-03-01
PT1317455E (pt) 2004-11-30

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Legal Events

Date Code Title Description
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B11B Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements