BR0013090A - Inibidores de triptase - Google Patents

Inibidores de triptase

Info

Publication number
BR0013090A
BR0013090A BR0013090-7A BR0013090A BR0013090A BR 0013090 A BR0013090 A BR 0013090A BR 0013090 A BR0013090 A BR 0013090A BR 0013090 A BR0013090 A BR 0013090A
Authority
BR
Brazil
Prior art keywords
tryptase inhibitors
inhibitors
tryptase
compound
novel effective
Prior art date
Application number
BR0013090-7A
Other languages
English (en)
Inventor
Thomas Baer
Thomas Martin
Josef Stadlwieser
Andreas Dominik
Daniela Bundschuh
Karl Zech
Original Assignee
Byk Gulden Lomberg Chem Fab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Byk Gulden Lomberg Chem Fab filed Critical Byk Gulden Lomberg Chem Fab
Publication of BR0013090A publication Critical patent/BR0013090A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D245/00—Heterocyclic compounds containing rings of more than seven members having two nitrogen atoms as the only ring hetero atoms
    • C07D245/02—Heterocyclic compounds containing rings of more than seven members having two nitrogen atoms as the only ring hetero atoms not condensed with other rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Patente de Invenção: "INIBIDORES DE TRIPTASE". A invenção refere-se a compostos de fórmula 1 em que M, A1, A2, A3, A4, A5, A6, B1, B2, B3, B4, BS, B6, K1 e K2 têm os significados como fornecidos na descrição, compostos estes que são novos inibidores de triptase eficazes.
BR0013090-7A 1999-08-10 2000-08-09 Inibidores de triptase BR0013090A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP99115737 1999-08-10
PCT/EP2000/007720 WO2001010848A2 (en) 1999-08-10 2000-08-09 Diazocin-dione derivatives and their use s tryptase inhibitors

Publications (1)

Publication Number Publication Date
BR0013090A true BR0013090A (pt) 2002-04-30

Family

ID=8238754

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0013090-7A BR0013090A (pt) 1999-08-10 2000-08-09 Inibidores de triptase

Country Status (19)

Country Link
US (1) US6673786B1 (pt)
EP (1) EP1208089B1 (pt)
JP (1) JP2003506442A (pt)
KR (1) KR20020016942A (pt)
CN (1) CN1378538A (pt)
AT (1) ATE279398T1 (pt)
AU (1) AU777026B2 (pt)
BR (1) BR0013090A (pt)
CA (1) CA2381919A1 (pt)
DE (1) DE60014932T2 (pt)
DK (1) DK1208089T3 (pt)
ES (1) ES2230155T3 (pt)
IL (1) IL147649A0 (pt)
MX (1) MXPA02001426A (pt)
PL (1) PL356170A1 (pt)
PT (1) PT1208089E (pt)
SI (1) SI1208089T1 (pt)
WO (1) WO2001010848A2 (pt)
ZA (1) ZA200201112B (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TR200402164T4 (tr) 1999-12-20 2004-10-21 Altana Pharma Ag Triptaz inhibitörler
US7015325B2 (en) 1999-12-20 2006-03-21 Altana Pharma Ag Tryptase inhibitors
CA2438594A1 (en) 2001-01-31 2002-08-08 Altana Pharma Ag Diazocine derivatives and their use as tryptase inhibitors
CA2438685A1 (en) 2001-02-21 2002-08-29 Altana Pharma Ag Tryptase inhibitors
WO2002066420A2 (en) 2001-02-21 2002-08-29 Altana Pharma Ag Tryptase inhibitors
ATE348803T1 (de) 2001-06-19 2007-01-15 Altana Pharma Ag Tryptase-inhibitoren
WO2006044133A1 (en) * 2004-09-24 2006-04-27 Axys Pharmaceuticals, Inc. Active ketone inhibitors of tryptase

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0782571A1 (en) 1994-09-23 1997-07-09 Arris Pharmaceutical Corporation Compositions and methods for treating mast-cell inflammatory condition
KR20000029679A (ko) * 1996-07-30 2000-05-25 헤이즈 더블유.그쉬웬드 다니엘 에이치.페트리 트립타아제활성관련질병을치료하기위한화합물및조성물
JP2002502850A (ja) 1998-02-06 2002-01-29 マックス−プランク−ゲゼルシャフト・ツア・フェルデルング・デア・ヴィッセンシャフテン・エー・ファオ トリプターゼ阻害物質

Also Published As

Publication number Publication date
EP1208089B1 (en) 2004-10-13
AU777026B2 (en) 2004-09-30
JP2003506442A (ja) 2003-02-18
PL356170A1 (en) 2004-06-14
AU7273700A (en) 2001-03-05
EP1208089A2 (en) 2002-05-29
DE60014932T2 (de) 2005-10-13
ATE279398T1 (de) 2004-10-15
DK1208089T3 (da) 2005-02-14
SI1208089T1 (en) 2005-04-30
US6673786B1 (en) 2004-01-06
WO2001010848A2 (en) 2001-02-15
ZA200201112B (en) 2002-11-27
CN1378538A (zh) 2002-11-06
WO2001010848A3 (en) 2001-12-06
ES2230155T3 (es) 2005-05-01
KR20020016942A (ko) 2002-03-06
IL147649A0 (en) 2002-08-14
CA2381919A1 (en) 2001-02-15
DE60014932D1 (de) 2004-11-18
MXPA02001426A (es) 2002-08-12
PT1208089E (pt) 2005-02-28

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Legal Events

Date Code Title Description
B25D Requested change of name of applicant approved
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]