BG60533B2 - Заместени имидазолидини,метод за получаването ими приложението им като лекарствено средство и състави,които ги съдържат - Google Patents

Заместени имидазолидини,метод за получаването ими приложението им като лекарствено средство и състави,които ги съдържат Download PDF

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Publication number
BG60533B2
BG60533B2 BG98507A BG9850794A BG60533B2 BG 60533 B2 BG60533 B2 BG 60533B2 BG 98507 A BG98507 A BG 98507A BG 9850794 A BG9850794 A BG 9850794A BG 60533 B2 BG60533 B2 BG 60533B2
Authority
BG
Bulgaria
Prior art keywords
trifluoromethyl
nitrophenyl
dimethyl
compound
dimethylimidazoline
Prior art date
Application number
BG98507A
Other languages
Bulgarian (bg)
English (en)
Inventor
Claude Bonne
Pierre Girault
Jacques Perronnet
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of BG60533B2 publication Critical patent/BG60533B2/bg

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/72—Two oxygen atoms, e.g. hydantoin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/88—Nitrogen atoms, e.g. allantoin

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Electromechanical Clocks (AREA)
BG98507A 1975-10-29 1994-02-22 Заместени имидазолидини,метод за получаването ими приложението им като лекарствено средство и състави,които ги съдържат BG60533B2 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7533084A FR2329276A1 (fr) 1975-10-29 1975-10-29 Nouvelles imidazolidines substituees, procede de preparation, application comme medicament et compositions les renfermant

Publications (1)

Publication Number Publication Date
BG60533B2 true BG60533B2 (bg) 1995-07-28

Family

ID=9161795

Family Applications (1)

Application Number Title Priority Date Filing Date
BG98507A BG60533B2 (bg) 1975-10-29 1994-02-22 Заместени имидазолидини,метод за получаването ими приложението им като лекарствено средство и състави,които ги съдържат

Country Status (18)

Country Link
US (1) US4097578A (US07655688-20100202-C00086.png)
JP (1) JPS6011701B2 (US07655688-20100202-C00086.png)
AU (1) AU500542B2 (US07655688-20100202-C00086.png)
BE (1) BE847742A (US07655688-20100202-C00086.png)
BG (1) BG60533B2 (US07655688-20100202-C00086.png)
CA (1) CA1086751A (US07655688-20100202-C00086.png)
CH (1) CH599164A5 (US07655688-20100202-C00086.png)
DE (1) DE2649925C2 (US07655688-20100202-C00086.png)
DK (1) DK152125C (US07655688-20100202-C00086.png)
ES (1) ES452746A1 (US07655688-20100202-C00086.png)
FR (1) FR2329276A1 (US07655688-20100202-C00086.png)
GB (1) GB1518444A (US07655688-20100202-C00086.png)
GE (1) GEP19970948B (US07655688-20100202-C00086.png)
IE (1) IE43875B1 (US07655688-20100202-C00086.png)
LU (2) LU76085A1 (US07655688-20100202-C00086.png)
NL (2) NL187102C (US07655688-20100202-C00086.png)
SE (1) SE430502B (US07655688-20100202-C00086.png)
SU (1) SU596165A3 (US07655688-20100202-C00086.png)

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FR2671348B1 (fr) * 1991-01-09 1993-03-26 Roussel Uclaf Nouvelles phenylimidazolidines, leur procede de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant.
US5411981A (en) * 1991-01-09 1995-05-02 Roussel Uclaf Phenylimidazolidines having antiandrogenic activity
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FR2685328B1 (fr) * 1991-12-20 1995-12-01 Rhone Poulenc Agrochimie Derives de 2-imidazoline-5-ones et 2-imidazoline-5-thiones fongicides.
US6002016A (en) * 1991-12-20 1999-12-14 Rhone-Poulenc Agrochimie Fungicidal 2-imidazolin-5-ones and 2-imidazoline-5-thiones
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TW521073B (en) * 1994-01-05 2003-02-21 Hoechst Marion Roussel Inc New optionally substituted phenylimidazolidines, their preparation process, their use as anti-androgenic agent and the pharmaceutical compositions containing them
FR2724169B1 (fr) * 1994-09-06 1997-01-03 Roussel Uclaf Nouvelles phenylimidazolidines eventuellement substituees, leur procede et des intermediaires de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant
FR2715402B1 (fr) * 1994-01-05 1996-10-04 Roussel Uclaf Nouvelles phénylimidazolines éventuellement substituées, leur procédé et des intermédiaires de préparation, leur application comme médicaments et les compositions pharmaceutiques les renfermant.
FR2725206B1 (fr) * 1994-09-29 1996-12-06 Roussel Uclaf Nouvelles imidazolidines substituees par un heterocycle, leur procede et des intermediaires de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant
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Also Published As

Publication number Publication date
LU88282I2 (fr) 1994-05-04
ES452746A1 (es) 1977-10-01
CA1086751A (fr) 1980-09-30
DK152125C (da) 1988-06-20
JPS6011701B2 (ja) 1985-03-27
AU1909576A (en) 1978-05-04
SE7610859L (sv) 1977-04-30
DK487476A (da) 1977-04-30
FR2329276B1 (US07655688-20100202-C00086.png) 1979-09-14
NL930079I2 (nl) 1993-10-01
BE847742A (fr) 1977-04-28
AU500542B2 (en) 1979-05-24
SE430502B (sv) 1983-11-21
NL187102B (nl) 1991-01-02
GB1518444A (en) 1978-07-19
IE43875L (en) 1977-04-29
FR2329276A1 (fr) 1977-05-27
IE43875B1 (en) 1981-06-17
DE2649925A1 (de) 1977-05-12
JPS5257176A (en) 1977-05-11
NL187102C (nl) 1991-06-03
CH599164A5 (US07655688-20100202-C00086.png) 1978-05-12
DE2649925C2 (de) 1986-08-28
LU76085A1 (US07655688-20100202-C00086.png) 1977-05-31
NL930079I1 (nl) 1993-09-16
US4097578A (en) 1978-06-27
DK152125B (da) 1988-02-01
NL7611576A (nl) 1977-05-03
SU596165A3 (ru) 1978-02-28
GEP19970948B (en) 1997-04-18

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