IT1214735B - Impiego di 1-(3'-trifluorometil 4'nitrofenil) 4,4-dimetilimidazolin2,5-dione per il trattamento di cancri ormonodipendenti diverso da quello della prostata - Google Patents

Impiego di 1-(3'-trifluorometil 4'nitrofenil) 4,4-dimetilimidazolin2,5-dione per il trattamento di cancri ormonodipendenti diverso da quello della prostata

Info

Publication number
IT1214735B
IT1214735B IT8648618A IT4861886A IT1214735B IT 1214735 B IT1214735 B IT 1214735B IT 8648618 A IT8648618 A IT 8648618A IT 4861886 A IT4861886 A IT 4861886A IT 1214735 B IT1214735 B IT 1214735B
Authority
IT
Italy
Prior art keywords
dione
prostate
hormone
treatment
nitrofenil
Prior art date
Application number
IT8648618A
Other languages
English (en)
Other versions
IT8648618A0 (it
Inventor
Martine Moguilewski
Marie-Madeleine Bouton
Original Assignee
Roussel Maestretti Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Maestretti Spa filed Critical Roussel Maestretti Spa
Priority to IT8648618A priority Critical patent/IT1214735B/it
Publication of IT8648618A0 publication Critical patent/IT8648618A0/it
Priority to PCT/FR1987/000435 priority patent/WO1988003404A1/fr
Priority to AT87907513T priority patent/ATE116852T1/de
Priority to EP87907513A priority patent/EP0301034B1/fr
Priority to JP62506989A priority patent/JP2777888B2/ja
Priority to DE3750984T priority patent/DE3750984T2/de
Application granted granted Critical
Publication of IT1214735B publication Critical patent/IT1214735B/it
Priority to US07/529,948 priority patent/US5084472A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT8648618A 1986-11-04 1986-11-04 Impiego di 1-(3'-trifluorometil 4'nitrofenil) 4,4-dimetilimidazolin2,5-dione per il trattamento di cancri ormonodipendenti diverso da quello della prostata IT1214735B (it)

Priority Applications (7)

Application Number Priority Date Filing Date Title
IT8648618A IT1214735B (it) 1986-11-04 1986-11-04 Impiego di 1-(3'-trifluorometil 4'nitrofenil) 4,4-dimetilimidazolin2,5-dione per il trattamento di cancri ormonodipendenti diverso da quello della prostata
PCT/FR1987/000435 WO1988003404A1 (fr) 1986-11-04 1987-11-03 Application de la 1-(3'trifluoromethyl 4'-nitrophenyl) 4,4-dimethyl imidazoline 2,5-dione au traitement des cancers hormonodependants autres que celui de la prostate
AT87907513T ATE116852T1 (de) 1986-11-04 1987-11-03 Verwendung von 1-(3'-trifluormethyl-4'- nitrophenyl)-4,4- dimethylimidazolin-2,5-dion zur herstellung eines medikaments zur behandlung von hormonabhängigen krebserkrankungen ausser denen der prostata, der haut und des grimmdarms.
EP87907513A EP0301034B1 (fr) 1986-11-04 1987-11-03 Utilisation de la 1-(3'trifluoromethyl 4'-nitrophenyl) 4,4-dimethyl imidazoline 2,5-dione pour la fabrication d'un medicament destine au traitement des cancers hormonodependants autres que ceux de la prostate, de la peau et du colon
JP62506989A JP2777888B2 (ja) 1986-11-04 1987-11-03 前立腺癌以外のホルモン依存性癌の治療への1―(3′―トリフルオルメチル―4′―ニトロフエニル)―4,4―ジメチルイミダゾリン―2,5―ジオンの使用
DE3750984T DE3750984T2 (de) 1986-11-04 1987-11-03 Verwendung von 1-(3'-trifluormethyl-4'-nitrophenyl)-4,4- dimethylimidazolin-2,5-dion zur herstellung eines medikaments zur behandlung von hormonabhängigen krebserkrankungen ausser denen der prostata, der haut und des grimmdarms.
US07/529,948 US5084472A (en) 1986-11-04 1990-05-29 Application of 1-(3'-trifluoromethyl-4'-nitrophenyl)-4,4'-dimethylimidazoline 2,5-dione in the treatment of hormone-dependent cancers other than that of the prostate

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT8648618A IT1214735B (it) 1986-11-04 1986-11-04 Impiego di 1-(3'-trifluorometil 4'nitrofenil) 4,4-dimetilimidazolin2,5-dione per il trattamento di cancri ormonodipendenti diverso da quello della prostata

Publications (2)

Publication Number Publication Date
IT8648618A0 IT8648618A0 (it) 1986-11-04
IT1214735B true IT1214735B (it) 1990-01-18

Family

ID=11267665

Family Applications (1)

Application Number Title Priority Date Filing Date
IT8648618A IT1214735B (it) 1986-11-04 1986-11-04 Impiego di 1-(3'-trifluorometil 4'nitrofenil) 4,4-dimetilimidazolin2,5-dione per il trattamento di cancri ormonodipendenti diverso da quello della prostata

Country Status (6)

Country Link
EP (1) EP0301034B1 (it)
JP (1) JP2777888B2 (it)
AT (1) ATE116852T1 (it)
DE (1) DE3750984T2 (it)
IT (1) IT1214735B (it)
WO (1) WO1988003404A1 (it)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2329276A1 (fr) * 1975-10-29 1977-05-27 Roussel Uclaf Nouvelles imidazolidines substituees, procede de preparation, application comme medicament et compositions les renfermant
FR2465486A1 (fr) * 1979-09-21 1981-03-27 Roussel Uclaf Nouvelle application utilisant la lh-rh ou des agonistes

Also Published As

Publication number Publication date
JP2777888B2 (ja) 1998-07-23
ATE116852T1 (de) 1995-01-15
IT8648618A0 (it) 1986-11-04
JPH01501230A (ja) 1989-04-27
EP0301034A1 (fr) 1989-02-01
WO1988003404A1 (fr) 1988-05-19
DE3750984T2 (de) 1995-05-18
EP0301034B1 (fr) 1995-01-11
DE3750984D1 (de) 1995-02-23

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Legal Events

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TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19961105