BG60067B2 - МЕТОД ЗА ПОЛУЧАВАНЕ НА 3-/(5-МЕТИЛ-2-ФУРАНИЛ)МЕТИЛ/-N- (4-ПИПЕРИДИНИЛ)-3Н-ИМИДАЗО/4,5-b/-ПИРИДИН-2-АМИН 2-ХИДРОКСИ-1,2,3-ПРОПАНТРИКАРБОНАТ - Google Patents

МЕТОД ЗА ПОЛУЧАВАНЕ НА 3-/(5-МЕТИЛ-2-ФУРАНИЛ)МЕТИЛ/-N- (4-ПИПЕРИДИНИЛ)-3Н-ИМИДАЗО/4,5-b/-ПИРИДИН-2-АМИН 2-ХИДРОКСИ-1,2,3-ПРОПАНТРИКАРБОНАТ

Info

Publication number
BG60067B2
BG60067B2 BG094757A BG9475791A BG60067B2 BG 60067 B2 BG60067 B2 BG 60067B2 BG 094757 A BG094757 A BG 094757A BG 9475791 A BG9475791 A BG 9475791A BG 60067 B2 BG60067 B2 BG 60067B2
Authority
BG
Bulgaria
Prior art keywords
methyl
tricarbonate
imidazo
furanyl
piperidinyl
Prior art date
Application number
BG094757A
Other languages
Bulgarian (bg)
English (en)
Inventor
Alfons Gaston Maria Knaep
Tonny Nelen
Frans Janssens
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of BG60067B2 publication Critical patent/BG60067B2/bg

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pulmonology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Furan Compounds (AREA)
  • Medicinal Preparation (AREA)
BG094757A 1990-07-06 1991-07-04 МЕТОД ЗА ПОЛУЧАВАНЕ НА 3-/(5-МЕТИЛ-2-ФУРАНИЛ)МЕТИЛ/-N- (4-ПИПЕРИДИНИЛ)-3Н-ИМИДАЗО/4,5-b/-ПИРИДИН-2-АМИН 2-ХИДРОКСИ-1,2,3-ПРОПАНТРИКАРБОНАТ BG60067B2 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US54935090A 1990-07-06 1990-07-06

Publications (1)

Publication Number Publication Date
BG60067B2 true BG60067B2 (bg) 1993-09-30

Family

ID=24192647

Family Applications (1)

Application Number Title Priority Date Filing Date
BG094757A BG60067B2 (bg) 1990-07-06 1991-07-04 МЕТОД ЗА ПОЛУЧАВАНЕ НА 3-/(5-МЕТИЛ-2-ФУРАНИЛ)МЕТИЛ/-N- (4-ПИПЕРИДИНИЛ)-3Н-ИМИДАЗО/4,5-b/-ПИРИДИН-2-АМИН 2-ХИДРОКСИ-1,2,3-ПРОПАНТРИКАРБОНАТ

Country Status (25)

Country Link
EP (1) EP0464927B1 (de)
JP (1) JPH04230382A (de)
KR (1) KR0165894B1 (de)
CN (1) CN1026790C (de)
AT (1) ATE142207T1 (de)
AU (1) AU632949B2 (de)
BG (1) BG60067B2 (de)
CA (1) CA2043564A1 (de)
CZ (1) CZ279435B6 (de)
DE (1) DE69121807T2 (de)
ES (1) ES2091285T3 (de)
FI (1) FI94132C (de)
GR (1) GR3020951T3 (de)
HU (1) HUT58333A (de)
IE (1) IE75695B1 (de)
IL (1) IL98725A (de)
MX (1) MX9100102A (de)
NO (1) NO177854C (de)
NZ (1) NZ238369A (de)
PL (1) PL168719B1 (de)
PT (1) PT98215B (de)
RU (1) RU2047615C1 (de)
SG (1) SG48825A1 (de)
SK (1) SK278127B6 (de)
ZA (1) ZA915241B (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6211199B1 (en) 1995-11-17 2001-04-03 Aventis Pharmaceuticals Inc. Substituted 4-(1H-benzimidazol-2-yl-amino)piperidines useful for the treatment of allergic diseases
US6194406B1 (en) 1995-12-20 2001-02-27 Aventis Pharmaceuticals Inc. Substituted 4-(1H-benzimidazol-2-yl)[1,4]diazepanes useful for the treatment of allergic disease
US6423704B2 (en) 1995-12-20 2002-07-23 Aventis Pharmaceuticals Inc. Substituted 4-(1H-benzimidazol-2-yl)[1,4]diazepanes useful for the treatment of allergic diseases
US5922737A (en) * 1996-02-21 1999-07-13 Hoechst Marion Roussel, Inc. Substituted N-methyl-N-(4-(4-(1H-Benzimidazol-2-YL-amino) piperidin-1-YL)-2-(arlyl) butyl) benzamides useful for the treatment of allergic diseases
US5998439A (en) 1996-02-21 1999-12-07 Hoescht Marion Roussel, Inc. Substituted N-methyl-N-(4-(piperidin-1-yl)-2-(aryl)butyl)benzamides useful for the treatment of allergic diseases
US5932571A (en) * 1996-02-21 1999-08-03 Hoechst Marion Roussel, Inc. Substituted N-methyl-N-(4-(4-(1H-benzimidazol-2-yl) {1,4}diazepan-1-yl)-2-(aryl) butyl) benzamides useful for the treatment of allergic diseases
KR100289063B1 (ko) * 1997-12-17 2001-05-02 정선종 누름스윗치에의한휴대전화기용자동안테나
RU2139872C1 (ru) * 1998-12-22 1999-10-20 Кубанский государственный технологический университет 2,4-диметил-3-(5-нитрофурфурил)-пиразол, обладающий способностью активировать прорастание семян пшеницы
US7235567B2 (en) * 2000-06-15 2007-06-26 Schering Corporation Crystalline polymorph of a bisulfate salt of a thrombin receptor antagonist
RU2177782C1 (ru) * 2000-12-06 2002-01-10 Научный Центр Здоровья детей РАМН Суппозитории ректальные, содержащие витаминный комплекс

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3484096D1 (de) * 1983-11-30 1991-03-14 Janssen Pharmaceutica Nv Bizyklisches heterozyklyl aufveisende n-(bizyklisches heterozyklyl-4-piperidinamine.
CA1327579C (en) * 1986-02-03 1994-03-08 Frans Eduard Janssens Anti-histaminic compositions containing n-heterocyclyl-4-piperidinamines
GB8900380D0 (en) * 1989-01-09 1989-03-08 Janssen Pharmaceutica Nv 2-aminopyrimidinone derivatives
PH30434A (en) * 1989-04-07 1997-05-09 Janssen Pharmaceutica Nv Hydroxyalkylfuranyl derivatives

Also Published As

Publication number Publication date
ES2091285T3 (es) 1996-11-01
EP0464927A3 (en) 1992-04-08
KR920002597A (ko) 1992-02-28
CZ279435B6 (cs) 1995-04-12
AU8020691A (en) 1992-01-09
FI94132C (fi) 1995-07-25
ATE142207T1 (de) 1996-09-15
HUT58333A (en) 1992-02-28
RU2047615C1 (ru) 1995-11-10
ZA915241B (en) 1993-03-31
EP0464927B1 (de) 1996-09-04
HU912284D0 (en) 1991-12-30
KR0165894B1 (ko) 1999-01-15
IL98725A0 (en) 1992-07-15
MX9100102A (es) 1992-02-28
NO912650L (no) 1992-01-07
FI94132B (fi) 1995-04-13
IL98725A (en) 1995-07-31
PL168719B1 (pl) 1996-03-29
CN1026790C (zh) 1994-11-30
CS198791A3 (en) 1992-03-18
SG48825A1 (en) 1998-05-18
DE69121807T2 (de) 1997-01-23
AU632949B2 (en) 1993-01-14
PT98215A (pt) 1992-06-30
SK278127B6 (en) 1996-02-07
FI913281A0 (fi) 1991-07-05
EP0464927A2 (de) 1992-01-08
FI913281L (fi) 1992-01-07
PT98215B (pt) 1999-01-29
IE75695B1 (en) 1997-09-10
NO912650D0 (no) 1991-07-05
CN1058020A (zh) 1992-01-22
NZ238369A (en) 1993-07-27
NO177854C (no) 1995-12-06
CA2043564A1 (en) 1992-01-07
IE912362A1 (en) 1992-01-15
GR3020951T3 (en) 1996-12-31
PL290956A1 (en) 1992-06-26
JPH04230382A (ja) 1992-08-19
DE69121807D1 (de) 1996-10-10
NO177854B (no) 1995-08-28

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