BG40145A3 - Метод за получаване на 3-(3-пиридил)-1н,3н- пирило (1,2-с)тиазол-7-карбонитрил - Google Patents

Метод за получаване на 3-(3-пиридил)-1н,3н- пирило (1,2-с)тиазол-7-карбонитрил

Info

Publication number
BG40145A3
BG40145A3 BG065204A BG6520484A BG40145A3 BG 40145 A3 BG40145 A3 BG 40145A3 BG 065204 A BG065204 A BG 065204A BG 6520484 A BG6520484 A BG 6520484A BG 40145 A3 BG40145 A3 BG 40145A3
Authority
BG
Bulgaria
Prior art keywords
pyridyl
carbonitrile
thiazole
preparation
pyrilo
Prior art date
Application number
BG065204A
Other languages
Bulgarian (bg)
English (en)
Inventor
Jean-Louis Fabre
Daniel Farge
Claude James
Daniel Lave
Original Assignee
Rhone- Poulenc Sante Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone- Poulenc Sante Sa filed Critical Rhone- Poulenc Sante Sa
Publication of BG40145A3 publication Critical patent/BG40145A3/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyrrole Compounds (AREA)
BG065204A 1983-01-13 1984-01-10 Метод за получаване на 3-(3-пиридил)-1н,3н- пирило (1,2-с)тиазол-7-карбонитрил BG40145A3 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8300453A FR2541280B1 (fr) 1983-01-13 1983-01-13 Nouveaux derives du 1h, 3h-pyrrolo (1,2c) thiazolecarboxamide-7, leur preparation et les medicaments qui les contiennent

Publications (1)

Publication Number Publication Date
BG40145A3 true BG40145A3 (bg) 1986-10-15

Family

ID=9284898

Family Applications (3)

Application Number Title Priority Date Filing Date
BG065204A BG40145A3 (bg) 1983-01-13 1984-01-10 Метод за получаване на 3-(3-пиридил)-1н,3н- пирило (1,2-с)тиазол-7-карбонитрил
BG063835A BG39639A3 (bg) 1983-01-13 1984-01-10 Метод за получаване на 1н, 3н- пироло/1,2-с/ тиазолови производни
BG065203A BG40144A3 (bg) 1983-01-13 1984-01-10 Метод за получаване на 7-(1-имидазолилкарбонил)-3-(3-пиридил)- -1н,3н-пироло/1,2-с/тиазол

Family Applications After (2)

Application Number Title Priority Date Filing Date
BG063835A BG39639A3 (bg) 1983-01-13 1984-01-10 Метод за получаване на 1н, 3н- пироло/1,2-с/ тиазолови производни
BG065203A BG40144A3 (bg) 1983-01-13 1984-01-10 Метод за получаване на 7-(1-имидазолилкарбонил)-3-(3-пиридил)- -1н,3н-пироло/1,2-с/тиазол

Country Status (28)

Country Link
US (1) US4529728A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
EP (1) EP0115979B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
JP (2) JPS59137490A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
KR (1) KR910001482B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AR (1) AR240828A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AT (1) ATE21248T1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AU (1) AU562795B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BG (3) BG40145A3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (1) CA1229603A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CS (1) CS262417B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DD (1) DD218362A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DE (1) DE3460401D1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DK (1) DK13984A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ES (2) ES8407058A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FI (1) FI76577C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FR (1) FR2541280B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GR (1) GR81679B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
HU (1) HU193277B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IE (1) IE56839B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IL (1) IL70664A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
MA (1) MA20001A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
MX (5) MX160610A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NO (1) NO167031C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NZ (1) NZ206807A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PL (2) PL140595B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PT (1) PT77952B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
SU (3) SU1245263A3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ZA (2) ZA84235B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2557111B1 (fr) * 1983-12-21 1986-04-11 Rhone Poulenc Sante Nouveaux derives ortho-condenses du pyrrole, leur preparation et les medicaments qui les contiennent
FR2601016B1 (fr) * 1986-07-04 1988-10-07 Rhone Poulenc Sante Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2601015B1 (fr) * 1986-07-04 1988-08-05 Rhone Poulenc Sante Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent
CN1030415A (zh) 1987-02-20 1989-01-18 山之内制药株式会社 饱和的杂环碳酰胺衍生物和它的制备方法
FR2617484B1 (fr) * 1987-07-02 1989-10-20 Rhone Poulenc Sante Procede de preparation de l'acide (pyridyl-3)-3 1h-3h-pyrrolo (1,2-c) thiazolecarboxylique-7 dextrogyre
FR2626004B1 (fr) * 1988-01-20 1991-08-02 Rhone Poulenc Sante Procede de preparation du (pyridyl-3)-3 1h, 3h-pyrrolo (1,2-c) thiazolecarbonitrile-7
FR2644456B1 (fr) * 1989-03-17 1991-07-05 Rhone Poulenc Sante Nouveaux derives du 1h, 3h-pyrrolo(1,2-c)thiazolecarboxamide-7, leur preparation et les compositions pharmaceutiques qui les contiennent
JPH05501103A (ja) * 1989-06-26 1993-03-04 ザ・リサーチ・ファウンデーション・オヴ・ステイト・ユニヴァーシティ・オヴ・ニューヨーク ビス―アシルオキシメチル誘導体
FR2678834A1 (fr) * 1991-07-09 1993-01-15 Rhone Poulenc Rorer Sa Nouvelle application therapeutique du pyridylpyrrolothiazole carboxamide.
IL102494A0 (en) * 1991-07-17 1993-01-14 Abbott Lab Platelet activating factor antagonists
HU230518B1 (hu) * 2005-12-20 2016-10-28 Richter Gedeon Nyrt. Bradykinin B1 receptor szelektív antagonista hatással rendelkező új fenatridin származékok, eljárás előállításukra, és az ezeket tartalmazó gyógyszerkészítmények

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3544590A (en) * 1967-04-28 1970-12-01 Exxon Research Engineering Co Cyclic amines and the process for their formation
US3865839A (en) * 1973-03-01 1975-02-11 Hoechst Co American Thiopyranopyrrolylsalicyclic acids and derivatives thereof

Also Published As

Publication number Publication date
BG40144A3 (bg) 1986-10-15
DK13984D0 (da) 1984-01-12
SU1266472A3 (ru) 1986-10-23
DK13984A (da) 1984-07-14
MA20001A1 (fr) 1984-10-01
JPS59134798A (ja) 1984-08-02
MX13291A (es) 1993-11-01
AR240828A1 (es) 1991-02-28
CA1229603A (fr) 1987-11-24
FI840106A0 (fi) 1984-01-12
FR2541280B1 (fr) 1985-06-21
FI840106A7 (fi) 1984-07-14
IL70664A (en) 1986-10-31
AU562795B2 (en) 1987-06-18
PT77952A (fr) 1984-02-01
FI76577C (fi) 1988-11-10
ES528873A0 (es) 1984-08-16
ES8407058A1 (es) 1984-08-16
ES8502123A1 (es) 1984-12-16
NO840106L (no) 1984-07-16
PL251304A1 (en) 1985-09-24
PT77952B (fr) 1986-07-14
JPH0547548B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1993-07-19
NO167031B (no) 1991-06-17
EP0115979A1 (fr) 1984-08-15
SU1245263A3 (ru) 1986-07-15
DD218362A5 (de) 1985-02-06
FR2541280A1 (fr) 1984-08-24
MX13462A (es) 1993-08-01
MX13292A (es) 1993-11-01
IL70664A0 (en) 1984-04-30
ATE21248T1 (de) 1986-08-15
NZ206807A (en) 1985-12-13
FI76577B (fi) 1988-07-29
AU2320284A (en) 1984-07-19
PL141846B1 (en) 1987-08-31
ZA84233B (en) 1984-09-26
BG39639A3 (bg) 1986-07-15
PL245701A1 (en) 1985-05-07
JPH0653748B2 (ja) 1994-07-20
US4529728A (en) 1985-07-16
ES531518A0 (es) 1984-12-16
CS19784A2 (en) 1988-08-16
KR840007419A (ko) 1984-12-07
MX13463A (es) 1993-10-01
HU193277B (en) 1987-09-28
NO167031C (no) 1991-09-25
EP0115979B1 (fr) 1986-08-06
DE3460401D1 (en) 1986-09-11
HUT34986A (en) 1985-05-28
SU1284459A3 (ru) 1987-01-15
ZA84235B (en) 1984-09-26
IE56839B1 (en) 1992-01-01
AR240828A2 (es) 1991-02-28
KR910001482B1 (ko) 1991-03-09
IE840064L (en) 1984-07-13
JPS59137490A (ja) 1984-08-07
GR81679B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1984-12-12
PL140595B1 (en) 1987-05-30
CS262417B2 (en) 1989-03-14
MX160610A (es) 1990-03-28

Similar Documents

Publication Publication Date Title
IE790676L (en) N-heterocyclyl-4-piperidinamines
BG36199A3 (en) Method for preparing derivatives of 3- (1- piperidinylalkyl)- 4h- pyrido (1, 2- a) pyrimidin- 4- on
ATE39928T1 (de) 4-dimethylamino-1-hydroxybutan-1,1diphosphons|ure, deren wasserloesliche salze, verfahren zu ihrer herstellung sowie ihre verwendung.
BG37526A3 (bg) Метод за получаване на естери на малоновата киселина
BG37528A3 (bg) Метод за получаване на 4- аминофенил-амониев-тридецил- фосфонат
BG35327A3 (bg) Метод за получаване на пиридоксинови производни
BG40145A3 (bg) Метод за получаване на 3-(3-пиридил)-1н,3н- пирило (1,2-с)тиазол-7-карбонитрил
YU43032B (en) Process for obtaining 2,5-diketo-d-gluconic acid
BG29722A3 (bg) Метод за получаване на 2,5-дисубституирани пиримидин-4-они
BG42004A3 (en) Method for preparing pyridyl compounds
RO86850A (ro) Procedeu pentru prepararea unor 2-fenilimidazo/4,5c/-piridine
BG38489A3 (en) Method for preparing oxazophosphorine- 6, 4- thiolcalsulphonic acids and their neutral salts
BG38940A3 (en) Method for preparing penicillanoyloxymethyl penicillanate- 1, 1- dioxide
DE3374695D1 (en) L-2-hydroxy-4-methylpentanoic acid dehydrogenase, process for its production and its use
TR23890A (tr) Saf asit borik üretimine mahsus usul.
BG41129A3 (en) Method for preparing acetamide derivatives
BG38939A3 (en) Method for preparing 1, 1- dioxopenicillanoyloxymethyl ester of 6- (2- amino- 2- phenylacetamido)- penicillanic acid
FI883167L (fi) Menetelmä 3-(3-pyridyyli)-1H,3H-pyrrolo/1,2-c/tiatsoli-7-karboksyylihapon oikealle kiertävän muodon valmistamiseksi
BG39977A3 (en) Method for preparing derivatives of furyloxazolylacetic acid
ATE12772T1 (de) Verfahren zur herstellung von 5,6,7,7a-tetrahydro-4h-tieno (3,2-c) pyridin-2-onderivaten.
BG36937A3 (bg) Метод за получаване на производни на 5,6,7,7а-тетрахидро- 4н-тиен(3,2-с)пиридин-2-они
BG40653A3 (en) Method for preparing amidothiocarbamate derivatives of carbon acid
BG36346A3 (bg) Метод за получаване на имидазо/4,5,-в/-пиридини и -пиримидини
BG35041A3 (bg) Метод за получаване на заместени 2-пиперидин-4-амино-6,7- диметоксихиназолини
DK146181C (da) Fremgangsmaade til fremstilling af 4-amino-5-chlor-1-phenyl-pyridazon-6