BG38939A3 - Method for preparing 1, 1- dioxopenicillanoyloxymethyl ester of 6- (2- amino- 2- phenylacetamido)- penicillanic acid - Google Patents

Method for preparing 1, 1- dioxopenicillanoyloxymethyl ester of 6- (2- amino- 2- phenylacetamido)- penicillanic acid

Info

Publication number
BG38939A3
BG38939A3 BG067396A BG6739682A BG38939A3 BG 38939 A3 BG38939 A3 BG 38939A3 BG 067396 A BG067396 A BG 067396A BG 6739682 A BG6739682 A BG 6739682A BG 38939 A3 BG38939 A3 BG 38939A3
Authority
BG
Bulgaria
Prior art keywords
phenylacetamido
ester
amino
preparing
dioxopenicillanoyloxymethyl
Prior art date
Application number
BG067396A
Other languages
Bulgarian (bg)
English (en)
Inventor
Vytautas Jasys
Original Assignee
Pfizer Inc., a corporation organized аnd existing under the laws of the State of Delaware
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc., a corporation organized аnd existing under the laws of the State of Delaware filed Critical Pfizer Inc., a corporation organized аnd existing under the laws of the State of Delaware
Publication of BG38939A3 publication Critical patent/BG38939A3/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32—Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Cephalosporin Compounds (AREA)
BG067396A 1981-03-23 1982-03-15 Method for preparing 1, 1- dioxopenicillanoyloxymethyl ester of 6- (2- amino- 2- phenylacetamido)- penicillanic acid BG38939A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24645681A 1981-03-23 1981-03-23

Publications (1)

Publication Number Publication Date
BG38939A3 true BG38939A3 (en) 1986-03-14

Family

ID=22930766

Family Applications (2)

Application Number Title Priority Date Filing Date
BG055782A BG37380A3 (en) 1981-03-23 1982-03-15 Method for preparing 1, 1- dioxo- 6- halo (or 6, 6- dihalo)- penicillanoyloxymethylic ester of 6- (2- amino- 2- phenylacetamido) penicillanic acid
BG067396A BG38939A3 (en) 1981-03-23 1982-03-15 Method for preparing 1, 1- dioxopenicillanoyloxymethyl ester of 6- (2- amino- 2- phenylacetamido)- penicillanic acid

Family Applications Before (1)

Application Number Title Priority Date Filing Date
BG055782A BG37380A3 (en) 1981-03-23 1982-03-15 Method for preparing 1, 1- dioxo- 6- halo (or 6, 6- dihalo)- penicillanoyloxymethylic ester of 6- (2- amino- 2- phenylacetamido) penicillanic acid

Country Status (32)

Country Link
EP (1) EP0061274B1 (fr)
JP (3) JPS57169493A (fr)
KR (1) KR860001368B1 (fr)
AU (1) AU531892B2 (fr)
BG (2) BG37380A3 (fr)
CA (1) CA1213581A (fr)
CS (1) CS227345B2 (fr)
DD (1) DD202163A5 (fr)
DE (1) DE3267505D1 (fr)
DK (3) DK162392C (fr)
EG (1) EG15803A (fr)
ES (2) ES510655A0 (fr)
FI (1) FI74284C (fr)
GB (1) GB2095250A (fr)
GR (1) GR75935B (fr)
GT (1) GT198274393A (fr)
HK (1) HK52487A (fr)
HU (2) HU187667B (fr)
IE (1) IE52835B1 (fr)
IL (1) IL65308A (fr)
IN (1) IN159362B (fr)
MY (1) MY8700499A (fr)
NO (1) NO159658C (fr)
NZ (1) NZ200066A (fr)
PH (1) PH17602A (fr)
PL (3) PL138851B1 (fr)
PT (1) PT74621B (fr)
RO (2) RO87946A (fr)
SG (1) SG23387G (fr)
SU (2) SU1277897A3 (fr)
YU (2) YU42761B (fr)
ZA (1) ZA821899B (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0084730A1 (fr) * 1982-01-22 1983-08-03 Beecham Group Plc Esters de dérivés de pénicilline avec des inhibiteurs de bêta-lactamase, leur préparation et leur application
PH20068A (en) * 1982-12-06 1986-09-18 Pfizer Process and intermediates for sultamicillin and analogs
GB8808701D0 (en) * 1988-04-13 1988-05-18 Erba Carlo Spa Beta-lactam derivatives
ES2039299B1 (es) * 1991-10-04 1994-05-16 Asturpharma S A Procedimiento de obtencion de esteres de acido 1,1-dioxopenicilanico y sus sales.
ES2100125B1 (es) * 1995-06-02 1998-04-01 Asturpharma S A Procedimiento de preparacion de esteres de metanodiol de acido dioxopenicilanico.
CN112724162B (zh) * 2020-12-28 2022-06-10 华南农业大学 一种阿莫西林-舒巴坦杂合分子的合成方法及应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR830001903B1 (ko) * 1979-02-13 1983-09-19 레오 파마슈티칼 프로덕츠 리미티드 페니실란산유도체의 제조방법
IE49881B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates
SE449103B (sv) * 1979-03-05 1987-04-06 Pfizer Sett att framstella penicillansyra-1,1-dioxid samt estrar derav
ZA80646B (en) * 1979-03-05 1981-02-25 Pfizer Process and intermediates for penicillanic acid,1,1-dioxide and esters thereof
IE50650B1 (en) * 1979-10-11 1986-06-11 Leo Pharm Prod Ltd Method for producing penicillanic acid derivatives

Also Published As

Publication number Publication date
SU1277897A3 (ru) 1986-12-15
SU1277898A3 (ru) 1986-12-15
GT198274393A (es) 1983-09-08
DK165746B (da) 1993-01-11
AU8176482A (en) 1982-11-04
DK162392C (da) 1992-03-09
IL65308A0 (en) 1982-05-31
CA1213581A (fr) 1986-11-04
KR830009113A (ko) 1983-12-17
DK165746C (da) 1993-06-07
IE52835B1 (en) 1988-03-16
EP0061274B1 (fr) 1985-11-21
DD202163A5 (de) 1983-08-31
JPS6345287A (ja) 1988-02-26
PT74621A (en) 1982-04-01
PL235578A1 (en) 1983-06-20
FI820991L (fi) 1982-09-24
NO159658B (no) 1988-10-17
RO87946A (fr) 1985-12-20
JPS63146886A (ja) 1988-06-18
FI74284B (fi) 1987-09-30
SG23387G (en) 1987-07-10
YU61982A (en) 1985-03-20
PL240664A1 (en) 1983-09-12
PL139261B1 (en) 1987-01-31
EP0061274A1 (fr) 1982-09-29
DE3267505D1 (en) 1986-01-02
DK127182A (da) 1982-09-24
DK121491D0 (da) 1991-06-21
GB2095250A (en) 1982-09-29
HU189917B (en) 1986-08-28
DK162392B (da) 1991-10-21
PL240663A1 (en) 1983-09-12
PH17602A (en) 1984-10-05
JPS57169493A (en) 1982-10-19
YU43585B (en) 1989-08-31
NO159658C (no) 1989-01-25
ES8403132A1 (es) 1984-03-01
YU42761B (en) 1988-12-31
HUT34985A (en) 1985-05-28
FI74284C (fi) 1988-01-11
ES8305768A1 (es) 1983-04-16
YU181084A (en) 1987-06-30
IL65308A (en) 1985-03-31
RO84278B (ro) 1984-07-30
MY8700499A (en) 1987-12-31
EG15803A (en) 1990-08-30
ZA821899B (en) 1983-01-26
PL138851B1 (en) 1986-11-29
NZ200066A (en) 1985-08-16
DK21892D0 (da) 1992-02-20
RO87946B (ro) 1985-12-02
IE820659L (en) 1982-09-23
DK21892A (da) 1992-02-20
PT74621B (en) 1984-11-26
HU187667B (en) 1986-02-28
NO820898L (no) 1982-09-24
HK52487A (en) 1987-07-17
KR860001368B1 (ko) 1986-09-17
PL134250B1 (en) 1985-08-31
JPH0331717B2 (fr) 1991-05-08
DK121491A (da) 1991-06-21
DK167119B1 (da) 1993-08-30
RO84278A (fr) 1984-05-23
ES518970A0 (es) 1984-03-01
CS227345B2 (en) 1984-04-16
BG37380A3 (en) 1985-05-15
IN159362B (fr) 1987-05-09
AU531892B2 (en) 1983-09-08
ES510655A0 (es) 1983-04-16
GR75935B (fr) 1984-08-02

Similar Documents

Publication Publication Date Title
BG40654A3 (en) Method for preparing cycloalkyltriazoles
BG40652A3 (en) Method for preparing (1- arylcyclobutyl) alkylamines
BG37526A3 (en) Method for preparing esters of malonic acid
BG40142A3 (en) Method for preparing piperazine derivatives
BG40481A3 (en) Method for preparing phenetanolamines
BG42185A3 (en) Method for preparing pyridylic compounds
BG39976A3 (en) Method for preparing benzamides
BG28568A3 (bg) Метод за получаване на естери на оксаловата киселина
BG42355A3 (en) Method for preparing aminoguanidinic derivatives
BG38489A3 (en) Method for preparing oxazophosphorine- 6, 4- thiolcalsulphonic acids and their neutral salts
BG40650A3 (en) Method for preparing ester of treo- 2- hydroxy- 3- (4- metoxyphenyl)- 3- (2- nitrophenylthio)- propionic acid
BG40807A3 (en) Method for preparing n- phenylcarbamates
BG35746A3 (en) Method for preparing 1- cyclohexenylmethylpyrolidines
BG40803A3 (en) Method for preparing arylcyclobutylalkylaminic derivatives
BG40147A3 (en) Method for preparing heterocyclic compounds
BG39639A3 (bg) Метод за получаване на 1н, 3н- пироло/1,2-с/ тиазолови производни
BG42352A3 (en) Method for preparing derivatives of cyclopropane- carbonic acid esters
BG38637A3 (en) Method for preparing 2- exo- hydroxy- 7- oxabicyclo [2, 2, 1] heptanes
BG38939A3 (en) Method for preparing 1, 1- dioxopenicillanoyloxymethyl ester of 6- (2- amino- 2- phenylacetamido)- penicillanic acid
BG38938A3 (en) Method for preparing chlormethylester of penicillanic acid derivatives
BG36935A3 (en) Method for preparing benzodiazepine compounds
BG35749A3 (en) Method for preparing 20- dihydro- 20, 23- dideoxytilonolide
BG41129A3 (en) Method for preparing acetamide derivatives
BG38338A3 (en) Method for preparing 6 alpha- methylhydrocortisonic derivatives
BG39977A3 (en) Method for preparing derivatives of furyloxazolylacetic acid