BE862608A - Nouvelles imidazo (1,2-a)quinoxalines substitu2es en position 4, leur procede de preparation et medicament les contenant - Google Patents

Nouvelles imidazo (1,2-a)quinoxalines substitu2es en position 4, leur procede de preparation et medicament les contenant

Info

Publication number
BE862608A
BE862608A BE184085A BE184085A BE862608A BE 862608 A BE862608 A BE 862608A BE 184085 A BE184085 A BE 184085A BE 184085 A BE184085 A BE 184085A BE 862608 A BE862608 A BE 862608A
Authority
BE
Belgium
Prior art keywords
quinoxalines
substituted
preparation
product containing
medicinal product
Prior art date
Application number
BE184085A
Other languages
English (en)
French (fr)
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of BE862608A publication Critical patent/BE862608A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Transplantation (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
BE184085A 1977-01-07 1978-01-03 Nouvelles imidazo (1,2-a)quinoxalines substitu2es en position 4, leur procede de preparation et medicament les contenant BE862608A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US75764077A 1977-01-07 1977-01-07

Publications (1)

Publication Number Publication Date
BE862608A true BE862608A (fr) 1978-07-03

Family

ID=25048641

Family Applications (1)

Application Number Title Priority Date Filing Date
BE184085A BE862608A (fr) 1977-01-07 1978-01-03 Nouvelles imidazo (1,2-a)quinoxalines substitu2es en position 4, leur procede de preparation et medicament les contenant

Country Status (19)

Country Link
US (1) US4160097A (enExample)
JP (2) JPS5387398A (enExample)
AU (1) AU521807B2 (enExample)
BE (1) BE862608A (enExample)
CA (1) CA1149385A (enExample)
CH (2) CH636102A5 (enExample)
CS (1) CS200232B2 (enExample)
DE (2) DE2800480A1 (enExample)
DK (1) DK157024C (enExample)
FI (1) FI64374C (enExample)
FR (1) FR2376858A1 (enExample)
GB (2) GB1579498A (enExample)
GR (1) GR73168B (enExample)
IE (1) IE46191B1 (enExample)
LU (1) LU78813A1 (enExample)
NL (1) NL7800114A (enExample)
SE (2) SE436359B (enExample)
YU (1) YU44663B (enExample)
ZA (1) ZA7827B (enExample)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE439308B (sv) * 1978-08-02 1985-06-10 Roussel Uclaf Imidazo(1,2-a)kinoxaliner och farmaceutiska kompositioner derav
JPS5569567A (en) * 1978-11-21 1980-05-26 Eisai Co Ltd Novel imidazole compound, and antidepressant containing the same
IT1209431B (it) * 1980-11-28 1989-07-16 Angeli Inst Spa Imidazolilfenil amidine, processi per la loro preparazione e loro impiego farmaceutico, ed intermedi di preparazione.
DE3830054A1 (de) * 1988-09-03 1990-03-15 Boehringer Mannheim Gmbh Phenylamide - verfahren zu ihrer herstellung sowie diese verbindungen enthaltende arzneimittel
JPH0349309U (enExample) * 1989-09-21 1991-05-14
US6635626B1 (en) 1997-08-25 2003-10-21 Bristol-Myers Squibb Co. Imidazoquinoxaline protein tyrosine kinase inhibitors
US6235740B1 (en) 1997-08-25 2001-05-22 Bristol-Myers Squibb Co. Imidazoquinoxaline protein tyrosine kinase inhibitors
CA2310072A1 (en) 1997-11-11 1999-05-20 Hiroyuki Ohno Fused pyrazine compounds
DE69940808D1 (de) * 1998-03-04 2009-06-10 Bristol Myers Squibb Co Heterocyclen substituierte imidazopyrazine als protein- tyrosin-kinase-inhibitoren
AU1182702A (en) 2000-10-03 2002-04-15 Bristol Myers Squibb Co Amino-substituted tetracyclic compounds useful as anti-inflammatory agents and pharmaceutical compositions comprising same
US6869956B2 (en) * 2000-10-03 2005-03-22 Bristol-Myers Squibb Company Methods of treating inflammatory and immune diseases using inhibitors of IκB kinase (IKK)
CZ20032287A3 (cs) * 2001-02-01 2004-02-18 Bristol-Myers Squibb Company Způsoby léčení zánětlivých a imunitních nemocí za použití inhibitorů IkB kinázy (IKK)
EP2066642A1 (en) * 2006-09-25 2009-06-10 Arete Therapeutics, INC. Soluble epoxide hydrolase inhibitors
WO2024169848A1 (zh) * 2023-02-17 2024-08-22 南京同诺康医药科技有限公司 miR-124诱导剂及其制备方法和用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3541109A (en) * 1968-06-25 1970-11-17 Du Pont 1-substituted imidazoles useful in acth reserve assay
US4011236A (en) * 1968-09-09 1977-03-08 Merck & Co., Inc. N-(benzimidazol-2-yl)arylcarboxamides as ultraviolet (uv) light absorbers
GB1347493A (en) * 1971-02-11 1974-02-27 Aspro Nicholas Ltd Benzazine derivatives
US3994893A (en) 1975-11-03 1976-11-30 E. R. Squibb & Sons, Inc. 4-Amino derivatives of pyrozolo[1,5-a]quinoxaline-3-carboxylic acid and esters

Also Published As

Publication number Publication date
SE460477B (sv) 1989-10-16
US4160097A (en) 1979-07-03
FI780023A7 (fi) 1978-07-08
SE8300945L (sv) 1983-02-21
SE8300945D0 (sv) 1983-02-21
FR2376858A1 (fr) 1978-08-04
YU2178A (en) 1990-04-30
FI64374C (fi) 1983-11-10
CH640229A5 (fr) 1983-12-30
CA1149385A (en) 1983-07-05
JPS61171470A (ja) 1986-08-02
DE2858766C2 (enExample) 1990-04-05
DK157024C (da) 1990-04-02
CH636102A5 (fr) 1983-05-13
DK4278A (da) 1978-07-08
DE2800480A1 (de) 1978-07-13
DK157024B (da) 1989-10-30
JPS5387398A (en) 1978-08-01
JPH0130825B2 (enExample) 1989-06-22
SE436359B (sv) 1984-12-03
SE7800138L (sv) 1978-07-08
FI64374B (fi) 1983-07-29
FR2376858B1 (enExample) 1980-10-24
CS200232B2 (en) 1980-08-29
LU78813A1 (fr) 1978-09-18
ZA7827B (en) 1979-01-31
IE780037L (en) 1978-07-07
AU3233178A (en) 1979-07-19
DE2800480C2 (enExample) 1990-04-12
NL7800114A (nl) 1978-07-11
GR73168B (enExample) 1984-02-14
YU44663B (en) 1990-12-31
JPS6259110B2 (enExample) 1987-12-09
IE46191B1 (en) 1983-03-23
GB1579499A (en) 1980-11-19
AU521807B2 (en) 1982-04-29
GB1579498A (en) 1980-11-19

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: BRISTOL-MYERS CY

Effective date: 19920131