BE2011C004I2 - - Google Patents
Info
- Publication number
- BE2011C004I2 BE2011C004I2 BE2011C004C BE2011C004C BE2011C004I2 BE 2011C004 I2 BE2011C004 I2 BE 2011C004I2 BE 2011C004 C BE2011C004 C BE 2011C004C BE 2011C004 C BE2011C004 C BE 2011C004C BE 2011C004 I2 BE2011C004 I2 BE 2011C004I2
- Authority
- BE
- Belgium
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/16—Purine radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
- C07D473/32—Nitrogen atom
- C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/338,185 US6403567B1 (en) | 1999-06-22 | 1999-06-22 | N-pyrazole A2A adenosine receptor agonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BE2011C004I2 true BE2011C004I2 (US07585860-20090908-C00083.png) | 2019-05-21 |
Family
ID=23323763
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BE2011C004C BE2011C004I2 (US07585860-20090908-C00083.png) | 1999-06-22 | 2011-02-03 |
Country Status (27)
Families Citing this family (69)
| Publication number | Priority date | Publication date | Assignee | Title |
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| CZ308577B6 (cs) | 2011-08-18 | 2020-12-16 | Farmak, A. S. | Způsob přípravy 2-(4-methoxykarbonylpyrazol-1-yl)adenosinu a 2-(4-ethoxykarbonylpyrazol-1-yl)adenosinu |
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| CZ305213B6 (cs) * | 2013-04-29 | 2015-06-10 | Farmak, A. S. | Polymorf E 2-[4-[(methylamino)karbonyl]-1H-pyrazol-1-yl]adenosinu a způsob jeho přípravy |
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| CN104513241B (zh) * | 2013-09-30 | 2017-02-08 | 浙江海正药业股份有限公司 | 瑞加德松新中间体及其制备方法和应用 |
| CN104744540A (zh) * | 2013-12-26 | 2015-07-01 | 上海紫源制药有限公司 | 一种制备瑞加德松的方法 |
| CN105085593A (zh) * | 2014-04-21 | 2015-11-25 | 上海紫源制药有限公司 | 瑞加德松的晶型及其制备方法 |
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| US9809617B2 (en) | 2015-07-03 | 2017-11-07 | Shanghai Ziyuan Pharmaceutical Co., Ltd. | Crystal form of regadenoson and preparation method thereof |
| CN106397442B (zh) * | 2015-07-28 | 2020-03-27 | 国药集团国瑞药业有限公司 | 一种瑞加德松的纯化方法 |
| RU2742417C1 (ru) | 2017-01-13 | 2021-02-05 | Тобиси Фармасьютикал Ко., Лтд. | Регулятор активации нейтрофилов |
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| US10815265B2 (en) | 2018-06-29 | 2020-10-27 | Usv Private Limited | Process for preparation of regadenoson and polymorphs thereof |
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