AU777097B2 - Process for preparing cyclic thioamides - Google Patents

Process for preparing cyclic thioamides Download PDF

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Publication number
AU777097B2
AU777097B2 AU22635/00A AU2263500A AU777097B2 AU 777097 B2 AU777097 B2 AU 777097B2 AU 22635/00 A AU22635/00 A AU 22635/00A AU 2263500 A AU2263500 A AU 2263500A AU 777097 B2 AU777097 B2 AU 777097B2
Authority
AU
Australia
Prior art keywords
compound
formula
acid
reacting
preparing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU22635/00A
Other languages
English (en)
Other versions
AU2263500A (en
Inventor
Paul David Hill
George Joseph Quallich
Jeffrey William Raggon
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Products Inc
Original Assignee
Pfizer Products Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc filed Critical Pfizer Products Inc
Publication of AU2263500A publication Critical patent/AU2263500A/en
Application granted granted Critical
Publication of AU777097B2 publication Critical patent/AU777097B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/23—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
    • C07C323/24—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/25—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/52—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/60—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/12—1,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
AU22635/00A 1999-03-30 2000-03-28 Process for preparing cyclic thioamides Ceased AU777097B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US12683199P 1999-03-30 1999-03-30
US60/126831 1999-03-30

Publications (2)

Publication Number Publication Date
AU2263500A AU2263500A (en) 2000-10-05
AU777097B2 true AU777097B2 (en) 2004-09-30

Family

ID=22426907

Family Applications (1)

Application Number Title Priority Date Filing Date
AU22635/00A Ceased AU777097B2 (en) 1999-03-30 2000-03-28 Process for preparing cyclic thioamides

Country Status (25)

Country Link
US (1) US6388127B1 (enrdf_load_stackoverflow)
EP (1) EP1041070B1 (enrdf_load_stackoverflow)
JP (1) JP3566175B2 (enrdf_load_stackoverflow)
KR (1) KR100386524B1 (enrdf_load_stackoverflow)
CN (2) CN1290829C (enrdf_load_stackoverflow)
AR (1) AR029744A1 (enrdf_load_stackoverflow)
AT (1) ATE277025T1 (enrdf_load_stackoverflow)
AU (1) AU777097B2 (enrdf_load_stackoverflow)
BR (1) BR0001492A (enrdf_load_stackoverflow)
CA (1) CA2302727C (enrdf_load_stackoverflow)
CZ (1) CZ298140B6 (enrdf_load_stackoverflow)
DE (1) DE60013942T2 (enrdf_load_stackoverflow)
DK (1) DK1041070T3 (enrdf_load_stackoverflow)
ES (1) ES2226715T3 (enrdf_load_stackoverflow)
HU (1) HUP0001327A3 (enrdf_load_stackoverflow)
ID (1) ID25428A (enrdf_load_stackoverflow)
IL (1) IL135243A (enrdf_load_stackoverflow)
IN (1) IN188844B (enrdf_load_stackoverflow)
PL (1) PL196446B1 (enrdf_load_stackoverflow)
PT (1) PT1041070E (enrdf_load_stackoverflow)
RU (1) RU2219173C2 (enrdf_load_stackoverflow)
TR (1) TR200000834A2 (enrdf_load_stackoverflow)
TW (1) TW460472B (enrdf_load_stackoverflow)
YU (1) YU15500A (enrdf_load_stackoverflow)
ZA (1) ZA200001536B (enrdf_load_stackoverflow)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE277025T1 (de) * 1999-03-30 2004-10-15 Pfizer Prod Inc Verfahren zur herstellung von cyclischen thioamiden
WO2014039715A1 (en) 2012-09-07 2014-03-13 University Of Rochester Methods and compositions for site-specific labeling of peptides and proteins
US9999921B2 (en) 2015-06-15 2018-06-19 Gm Global Technology Operatioins Llc Method of making aluminum or magnesium based composite engine blocks or other parts with in-situ formed reinforced phases through squeeze casting or semi-solid metal forming and post heat treatment

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2755278A (en) * 1956-07-17 Thiamori
GB8412862D0 (en) * 1984-05-19 1984-06-27 Beecham Group Plc Compounds
DE3581641D1 (de) * 1984-10-04 1991-03-07 Zenyaku Kogyo Kk 1,4-thiazinabkoemmlinge, deren herstellung und diese enthaltende kardiotonische mittel.
IL106142A (en) * 1992-06-29 1997-03-18 Merck & Co Inc Morpholine and thiomorpholine tachykinin receptor antagonists, their preparation and pharmaceutical compositions containing them
WO1994003652A1 (en) 1992-07-31 1994-02-17 Yokota Corporation Co., Ltd. Method of making metal of high purity from scrap of worked metal
GB9225377D0 (en) * 1992-12-04 1993-01-27 Ici Plc Herbicides
TW280812B (enrdf_load_stackoverflow) * 1993-07-02 1996-07-11 Bayer Ag
FR2715933B1 (fr) * 1994-02-07 1996-04-12 Oreal Nouveaux N-(hydroxyalkyl) carbamates d'alkyle et leurs applications en cosmétique, plus particulièrement dans des compositions capillaires.
US5663409A (en) * 1995-06-07 1997-09-02 Novus International, Inc. Process for the preparation of 3-(methylthio) propanal and 2-hydroxy-4-(methylthio) butanenitrile
UA56185C2 (uk) * 1996-09-30 2003-05-15 Пфайзер Інк. Аралкіл- та аралкіліденгетероциклічні лактами та іміди, фармацевтична композиція та спосіб лікування
ATE277025T1 (de) * 1999-03-30 2004-10-15 Pfizer Prod Inc Verfahren zur herstellung von cyclischen thioamiden

Also Published As

Publication number Publication date
CN1273244A (zh) 2000-11-15
IL135243A (en) 2005-09-25
RU2219173C2 (ru) 2003-12-20
EP1041070B1 (en) 2004-09-22
IN188844B (enrdf_load_stackoverflow) 2002-11-09
BR0001492A (pt) 2000-10-17
YU15500A (sh) 2002-03-18
ZA200001536B (en) 2001-09-27
AR029744A1 (es) 2003-07-16
EP1041070A1 (en) 2000-10-04
HK1064364A1 (en) 2005-01-28
ID25428A (id) 2000-10-05
DK1041070T3 (da) 2005-01-24
TR200000834A2 (tr) 2000-11-21
DE60013942D1 (de) 2004-10-28
CN1163490C (zh) 2004-08-25
ES2226715T3 (es) 2005-04-01
HU0001327D0 (en) 2000-06-28
DE60013942T2 (de) 2006-02-23
TW460472B (en) 2001-10-21
HUP0001327A3 (en) 2003-06-30
CZ20001142A3 (cs) 2000-12-13
CA2302727A1 (en) 2000-09-30
PL196446B1 (pl) 2008-01-31
CN1290829C (zh) 2006-12-20
PT1041070E (pt) 2004-12-31
AU2263500A (en) 2000-10-05
KR20010014647A (ko) 2001-02-26
CZ298140B6 (cs) 2007-07-04
ATE277025T1 (de) 2004-10-15
HUP0001327A2 (hu) 2001-04-28
CA2302727C (en) 2004-02-24
KR100386524B1 (ko) 2003-06-02
PL339287A1 (en) 2000-10-09
CN1519230A (zh) 2004-08-11
US6388127B1 (en) 2002-05-14
JP3566175B2 (ja) 2004-09-15
JP2000309581A (ja) 2000-11-07
HK1032053A1 (en) 2001-07-06
IL135243A0 (en) 2001-05-20

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