AU556754B2 - Microencapsulation of water soluble polypeptides - Google Patents

Microencapsulation of water soluble polypeptides

Info

Publication number
AU556754B2
AU556754B2 AU77560/81A AU7756081A AU556754B2 AU 556754 B2 AU556754 B2 AU 556754B2 AU 77560/81 A AU77560/81 A AU 77560/81A AU 7756081 A AU7756081 A AU 7756081A AU 556754 B2 AU556754 B2 AU 556754B2
Authority
AU
Australia
Prior art keywords
microencapsulation
water soluble
soluble polypeptides
water
biocompatable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired, expires
Application number
AU77560/81A
Other languages
English (en)
Other versions
AU7756081A (en
Inventor
John S. Kent
Danny H. Lewis
Lynda M. Sanders
Thomas R. Tice
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Syntex USA LLC
Original Assignee
Syntex USA LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22772297&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU556754(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Syntex USA LLC filed Critical Syntex USA LLC
Publication of AU7756081A publication Critical patent/AU7756081A/en
Application granted granted Critical
Publication of AU556754B2 publication Critical patent/AU556754B2/en
Adjusted expiration legal-status Critical
Expired legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5021—Organic macromolecular compounds
    • A61K9/5031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poly(lactide-co-glycolide)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08—Peptides having 5 to 11 amino acids
    • A61K38/09—Luteinising hormone-releasing hormone [LHRH], i.e. Gonadotropin-releasing hormone [GnRH]; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
    • A61K9/1647—Polyesters, e.g. poly(lactide-co-glycolide)

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Endocrinology (AREA)
  • Immunology (AREA)
  • Reproductive Health (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Manufacturing Of Micro-Capsules (AREA)
  • Medicinal Preparation (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Immobilizing And Processing Of Enzymes And Microorganisms (AREA)
  • Peptides Or Proteins (AREA)
AU77560/81A 1980-11-18 1981-11-17 Microencapsulation of water soluble polypeptides Expired AU556754B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US20786480A 1980-11-18 1980-11-18
US207864 1980-11-18

Publications (2)

Publication Number Publication Date
AU7756081A AU7756081A (en) 1982-05-27
AU556754B2 true AU556754B2 (en) 1986-11-20

Family

ID=22772297

Family Applications (1)

Application Number Title Priority Date Filing Date
AU77560/81A Expired AU556754B2 (en) 1980-11-18 1981-11-17 Microencapsulation of water soluble polypeptides

Country Status (15)

Country Link
EP (1) EP0052510B2 (online.php)
JP (1) JPS57118512A (online.php)
AT (1) ATE21624T1 (online.php)
AU (1) AU556754B2 (online.php)
CA (1) CA1176565A (online.php)
DE (2) DE3175230D1 (online.php)
HK (1) HK20489A (online.php)
IE (1) IE52003B1 (online.php)
IL (1) IL64298A (online.php)
MY (1) MY8700835A (online.php)
NL (1) NL930001I2 (online.php)
NZ (1) NZ198982A (online.php)
PH (1) PH19942A (online.php)
SG (1) SG94487G (online.php)
ZA (1) ZA817973B (online.php)

Families Citing this family (184)

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EP0052510B2 (en) 1994-10-19
HK20489A (en) 1989-03-17
NL930001I1 (nl) 1993-02-16
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ZA817973B (en) 1983-07-27
EP0052510A3 (en) 1982-09-08
IL64298A0 (en) 1982-02-28
PH19942A (en) 1986-08-14
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IE52003B1 (en) 1987-05-13
EP0052510B1 (en) 1986-08-27
JPS57118512A (en) 1982-07-23
EP0052510A2 (en) 1982-05-26
DE52510T1 (de) 1986-03-20
CA1176565A (en) 1984-10-23
IL64298A (en) 1985-07-31
SG94487G (en) 1988-05-06
ATE21624T1 (de) 1986-09-15
JPH0440329B2 (online.php) 1992-07-02
IE812695L (en) 1982-05-18
DE3175230D1 (en) 1986-10-02

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