AU503212B2 - 1-(3,5-dihydroxyphenyl)-2[hydroxyalkyl)amino] ethanols and their esters - Google Patents
1-(3,5-dihydroxyphenyl)-2[hydroxyalkyl)amino] ethanols and their estersInfo
- Publication number
- AU503212B2 AU503212B2 AU18122/76A AU1812276A AU503212B2 AU 503212 B2 AU503212 B2 AU 503212B2 AU 18122/76 A AU18122/76 A AU 18122/76A AU 1812276 A AU1812276 A AU 1812276A AU 503212 B2 AU503212 B2 AU 503212B2
- Authority
- AU
- Australia
- Prior art keywords
- ethanols
- dihydroxyphenyl
- hydroxyalkyl
- esters
- amino
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical class CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 title 1
- 150000002148 esters Chemical class 0.000 title 1
- 235000019441 ethanol Nutrition 0.000 title 1
- 125000002768 hydroxyalkyl group Chemical group 0.000 title 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
- C07C213/04—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reaction of ammonia or amines with olefin oxides or halohydrins
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
- C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
- C07C45/70—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form
- C07C45/71—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form being hydroxy groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
- C07D265/32—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings with oxygen atoms directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pulmonology (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Immunology (AREA)
- Emergency Medicine (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SESE7510988/ | 1975-10-01 | ||
| SE7510988A SE7510988L (sv) | 1975-10-01 | 1975-10-01 | Nya farmaceutiskt aktiva foreningar |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU1812276A AU1812276A (en) | 1978-04-06 |
| AU503212B2 true AU503212B2 (en) | 1979-08-30 |
Family
ID=20325688
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU18122/76A Expired AU503212B2 (en) | 1975-10-01 | 1976-09-27 | 1-(3,5-dihydroxyphenyl)-2[hydroxyalkyl)amino] ethanols and their esters |
Country Status (19)
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3163871D1 (en) | 1980-07-09 | 1984-07-05 | Draco Ab | 1-(dihydroxyphenyl)-2-amino-ethanol derivatives; preparation, compositions and intermediates |
| EP0103830A3 (de) * | 1982-09-22 | 1985-07-31 | Bayer Ag | Wachstumsfördernde Phenylethylamin-Derivate |
| AU705320B2 (en) * | 1995-12-28 | 1999-05-20 | Welfide Corporation | 2-amino-2-(2-(4-octylphenyl)ethyl)propane-1,3-diol or a pharmaceutically acceptable acid addition salt thereof for use in the preparation of a non-oral medicament, and for treatment of diseases and disorders |
| EA016485B1 (ru) | 2003-06-17 | 2012-05-30 | Арена Фармасьютикалз, Инк. | Способы получения 3-бензазепинов |
| EP2471779A1 (en) | 2006-04-03 | 2012-07-04 | Arena Pharmaceuticals, Inc. | Process for the resolution of a mixture of (R)- and (S)-8-chloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine |
| JP5404414B2 (ja) | 2006-12-05 | 2014-01-29 | アリーナ ファーマシューティカルズ， インコーポレイテッド | （ｒ）−８−クロロ−１−メチル−２，３，４，５−テトラヒドロ−１ｈ−３−ベンゾアゼピンおよびその中間体を調製するための方法 |
| RU2361604C1 (ru) * | 2007-10-29 | 2009-07-20 | Федеральное агентство по высокотехнологичной медицинской помощи Федеральное государственное учреждение "Уральский научно-исследовательский институт дерматовенерологии и иммунопатологии" (ФГУ УрНИИДВиИ Росмедтехнологий) | Способ лечения атопического дерматита |
| JP5491421B2 (ja) | 2008-03-04 | 2014-05-14 | アリーナ ファーマシューティカルズ， インコーポレイテッド | ５−ｈｔ２ｃアゴニストである（ｒ）−８−クロロ−１−メチル−２，３，４，５−テトラヒドロ−１ｈ−３−ベンゾアゼピンに関連する中間体の調製のためのプロセス |
| EP2443080A2 (en) | 2009-06-18 | 2012-04-25 | Arena Pharmaceuticals, Inc. | Process for the preparation of 5-ht2c receptor agonists |
| KR20130112848A (ko) | 2010-06-02 | 2013-10-14 | 아레나 파마슈티칼스, 인크. | 5-ｈｔ2ｃ 수용체 아고니스트의 제조 방법 |
| CA2808912C (en) | 2010-09-01 | 2019-09-17 | Zezhi Jesse Shao | Modified-release dosage forms of 5-ht2c agonists useful for weight management |
| MX2013002418A (es) | 2010-09-01 | 2013-08-01 | Arena Pharm Inc | Administracion de lorcaserina a individuos con daño renal. |
| SG10201506865WA (en) | 2010-09-01 | 2015-10-29 | Arena Pharm Inc | Non-hygroscopic salts of 5-ht2c agonists |
| WO2012030938A1 (en) | 2010-09-01 | 2012-03-08 | Arena Pharmaceuticals, Inc. | Salts of lorcaserin with optically active acids |
| AR088670A1 (es) | 2012-10-09 | 2014-06-25 | Arena Pharm Inc | Metodo de control del peso |
-
1975
- 1975-10-01 SE SE7510988A patent/SE7510988L/xx unknown
-
1976
- 1976-09-07 ZA ZA765331A patent/ZA765331B/xx unknown
- 1976-09-11 DE DE19762640972 patent/DE2640972A1/de not_active Withdrawn
- 1976-09-15 AT AT682376A patent/AT347427B/de not_active IP Right Cessation
- 1976-09-16 FI FI762660A patent/FI762660A7/fi not_active Application Discontinuation
- 1976-09-22 SU SU762402852A patent/SU638252A3/ru active
- 1976-09-27 AU AU18122/76A patent/AU503212B2/en not_active Expired
- 1976-09-27 NZ NZ182165A patent/NZ182165A/xx unknown
- 1976-09-28 DD DD195022A patent/DD126278A5/xx unknown
- 1976-09-30 ES ES451979A patent/ES451979A1/es not_active Expired
- 1976-09-30 LU LU75916A patent/LU75916A1/xx unknown
- 1976-09-30 NL NL7610845A patent/NL7610845A/xx not_active Application Discontinuation
- 1976-09-30 NO NO763345A patent/NO763345L/no unknown
- 1976-09-30 FR FR7629467A patent/FR2326183A1/fr not_active Withdrawn
- 1976-09-30 GB GB7640684A patent/GB1542317A/en not_active Expired
- 1976-09-30 DK DK439776AA patent/DK141622B/da unknown
- 1976-10-01 CS CS782253A patent/CS199644B2/cs unknown
- 1976-10-01 CS CS766357A patent/CS199643B2/cs unknown
- 1976-10-01 JP JP51118924A patent/JPS5242840A/ja active Pending
- 1976-10-01 BE BE171148A patent/BE846837A/xx unknown
-
1977
- 1977-10-13 SU SU772532454A patent/SU674669A3/ru active
Also Published As
| Publication number | Publication date |
|---|---|
| FR2326183A1 (fr) | 1977-04-29 |
| SU638252A3 (ru) | 1978-12-15 |
| DK439776A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1977-04-02 |
| DK141622B (da) | 1980-05-12 |
| ES451979A1 (es) | 1978-01-01 |
| GB1542317A (en) | 1979-03-14 |
| ATA682376A (de) | 1978-05-15 |
| SE7510988L (sv) | 1977-04-02 |
| CS199643B2 (en) | 1980-07-31 |
| AT347427B (de) | 1978-12-27 |
| FI762660A7 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1977-04-02 |
| JPS5242840A (en) | 1977-04-04 |
| AU1812276A (en) | 1978-04-06 |
| ZA765331B (en) | 1977-08-31 |
| NZ182165A (en) | 1978-07-10 |
| NO763345L (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1977-04-04 |
| BE846837A (fr) | 1977-04-01 |
| CS199644B2 (en) | 1980-07-31 |
| SU674669A3 (ru) | 1979-07-15 |
| LU75916A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1978-05-16 |
| DE2640972A1 (de) | 1977-04-14 |
| DD126278A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1977-07-06 |
| NL7610845A (nl) | 1977-04-05 |
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