AU491139B2 - 2-(2-acylhydrazino)-5-phenyl-3h-1,4-benzodiazepines - Google Patents

2-(2-acylhydrazino)-5-phenyl-3h-1,4-benzodiazepines

Info

Publication number
AU491139B2
AU491139B2 AU85499/75A AU8549975A AU491139B2 AU 491139 B2 AU491139 B2 AU 491139B2 AU 85499/75 A AU85499/75 A AU 85499/75A AU 8549975 A AU8549975 A AU 8549975A AU 491139 B2 AU491139 B2 AU 491139B2
Authority
AU
Australia
Prior art keywords
acylhydrazino
benzodiazepines
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
AU85499/75A
Other languages
English (en)
Other versions
AU8549975A (en
Inventor
Boling Hester' Jackson Jr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharmacia and Upjohn Co
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27123060&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU491139(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Upjohn Co filed Critical Upjohn Co
Application granted granted Critical
Publication of AU491139B2 publication Critical patent/AU491139B2/en
Publication of AU8549975A publication Critical patent/AU8549975A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20—Nitrogen atoms
AU85499/75A 1969-03-17 1975-10-07 2-(2-acylhydrazino)-5-phenyl-3h-1,4-benzodiazepines Expired AU491139B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US80793369A 1969-03-17 1969-03-17
US04/872,394 US3987052A (en) 1969-03-17 1969-10-29 6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines

Related Child Applications (1)

Application Number Title Priority Date Filing Date
AU11085/70A Division AU462769B2 (en) 1969-03-17 1970-02-05 6-PHENYL-4H-s-TRIAZOLO [4,3-2] [1,4] BENZODIAZEPINES AND PROCESS

Publications (2)

Publication Number Publication Date
AU491139B2 true AU491139B2 (en) 1975-12-18
AU8549975A AU8549975A (en) 1975-12-18

Family

ID=27123060

Family Applications (2)

Application Number Title Priority Date Filing Date
AU85499/75A Expired AU491139B2 (en) 1969-03-17 1975-10-07 2-(2-acylhydrazino)-5-phenyl-3h-1,4-benzodiazepines
AU85500/75A Expired AU490626B2 (en) 1969-03-17 1975-10-07 Process for preparing 6-phenyl04h-s-triazolo-[4,3-1] [1,4] benzodiazepines

Family Applications After (1)

Application Number Title Priority Date Filing Date
AU85500/75A Expired AU490626B2 (en) 1969-03-17 1975-10-07 Process for preparing 6-phenyl04h-s-triazolo-[4,3-1] [1,4] benzodiazepines

Country Status (18)

Country Link
US (1) US3987052A (xx)
JP (1) JPS4940239B1 (xx)
AU (2) AU491139B2 (xx)
BE (1) BE747493A (xx)
BR (1) BR7017488D0 (xx)
CH (1) CH535788A (xx)
DE (1) DE2012190C3 (xx)
ES (1) ES376689A1 (xx)
FR (1) FR2034999A1 (xx)
GB (1) GB1291631A (xx)
HK (1) HK61677A (xx)
IL (1) IL33859A (xx)
NL (2) NL172510C (xx)
OA (1) OA03446A (xx)
PH (1) PH9329A (xx)
PL (1) PL80541B1 (xx)
SE (1) SE387641B (xx)
YU (1) YU35139B (xx)

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* Cited by examiner, † Cited by third party
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DE2164778C2 (de) * 1971-03-03 1984-07-05 The Upjohn Co., Kalamazoo, Mich. 6-(o-Chlorphenyl)-1-methyl-4H-s-triazolo[4,3-a][1,4]-benzodiazepin und dieses enthaltende pharmazeutische Präparat
DE2164777A1 (de) * 1971-03-03 1972-09-07 Upjohn Co 8-Nitro-6-(o-halogenphenyl)-l-methyl-4H-s-triazolo eckige Klammer auf 4,3-a eckige Klammer zu-eckige Klammer auf 1-4 eckige Klammer zu benzodiazepine und diese enthaltende pharmazeutische Präparate
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GB1331015A (en) * 1971-04-28 1973-09-19 Upjohn Co 1-substituted-6-phenyl-4h-s-triazolo-4,3-a-1,4-benzodiazepines
US3759943A (en) * 1971-04-28 1973-09-18 Upjohn Co Amido and amino triazolo benzodiazepines
US4141902A (en) 1971-04-28 1979-02-27 The Upjohn Company 1-Halomethyl-6-phenyl-4H-s-[4,3-a][1,4]benzodiazepines
US3709899A (en) 1971-04-28 1973-01-09 Upjohn Co 6-phenyl-4h-s-triazolo(4,3-a)(1,4)benzodiazepines and their production
GB1323277A (en) * 1971-05-10 1973-07-11 Upjohn Co Triazolobenzodiazepines
US3734922A (en) * 1971-05-11 1973-05-22 Upjohn Co Certain 4h-s-triazolo(4,3-a)(1,4)benzodiazepines
US4000289A (en) * 1971-07-08 1976-12-28 The Upjohn Company Animal feed and process
BE787251A (fr) * 1971-08-04 1973-02-05 Upjohn Co Nouvelles benzodiazepines et leur preparation
US3870793A (en) * 1971-08-09 1975-03-11 Upjohn Co Animal feed and process
GB1373300A (en) * 1971-09-08 1974-11-06 Upjohn Co Triazolobenzodiazepines and the manufacture thereof
GB1381158A (en) * 1971-09-13 1975-01-22 Upjohn Co Benzodiazepines and the manufacture thereof
US3767661A (en) * 1971-09-13 1973-10-23 Upjohn Co 4h-s-triazolo(4,3-a)(1,4)benzodiazepines
US3714178A (en) * 1971-09-30 1973-01-30 Upjohn Co 6,7-DIHYDRO-7-ALKYL-5H-1,2,4-TRIAZOLO[4,3-d][1,4]BENZODIAZEPINES AND THEIR PRODUCTION
BE790838A (fr) * 1971-11-02 1973-04-30 Upjohn Co Nouvelles 1-aminophenyl-6-phenyl-s-triazolo (4,3-a) (1,4)- benzodiazepines, leur procede de preparation et medicament les contenant
FI53821C (fi) * 1971-11-15 1978-08-10 Ciba Geigy Ag Foerfarande foer framstaellning av farmakologiskt vaerdefull 6-fenyl-8-klor-4h-s-triazolo(4 3-a)(1 4)bensodiazepin-1-metanol
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US4431589A (en) * 1980-12-11 1984-02-14 Lilly House Benzodiazepine compounds and their use as pharmaceuticals
US4375473A (en) * 1982-01-04 1983-03-01 The Upjohn Company Method
US4455307A (en) * 1982-01-04 1984-06-19 The Upjohn Company Antihypertensive use of triazolobenzodiazepines
US4508726A (en) * 1982-09-16 1985-04-02 The Upjohn Company Treatment of panic disorders with alprazolam
DE3332830A1 (de) * 1982-09-16 1984-03-22 The Upjohn Co., 49001 Kalamazoo, Mich. Verwendung von benzodiazepinen zur bekaempfung oder bei der behandlung von panikzustaenden
US4481208A (en) * 1983-06-06 1984-11-06 The Upjohn Company Treatment of panic disorders with estazolam
US4689413A (en) * 1983-03-17 1987-08-25 The Upjohn Company Triazolo-benzodiazepine-1-ethanamines as diuretics
US4514407A (en) * 1983-03-17 1985-04-30 The Upjohn Company 1-Ethanamine-triazolo-benzodiazepines as diuretics
US4474699A (en) * 1983-05-25 1984-10-02 The Upjohn Company Preparing 1-aminomethyl-6-substituted-4H-s-triazolo[4,3-a][1,4]benzodiazepines in improved procedures
US4588721A (en) * 1983-09-12 1986-05-13 The Upjohn Company Treatment of negative symptoms of schizophrenia
US4547499A (en) * 1984-05-10 1985-10-15 The Upjohn Company 2,4-Dihydro-2(omega-aminoalkyl)-1H-[1,2,4]triazolo[3,4-c]benzoxazin-1-one anti-allergy drug compounds, compositions and use
US4634703A (en) * 1985-10-25 1987-01-06 Bristol-Myers Company Method for alleviation of panic disorders
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CN109906220A (zh) 2016-11-01 2019-06-18 豪夫迈·罗氏有限公司 用于治疗cns相关疾病的1,3-二氢-1,4-苯并二氮杂*-2-硫酮化合物
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Also Published As

Publication number Publication date
JPS4940239B1 (xx) 1974-10-31
DE2012190C3 (de) 1980-11-13
NL8100081A (nl) 1981-04-29
NL172510B (nl) 1983-04-18
PH9329A (en) 1975-09-23
HK61677A (en) 1977-12-23
YU35139B (en) 1980-09-25
GB1291631A (en) 1972-10-04
SE387641B (sv) 1976-09-13
YU34570A (en) 1979-04-30
OA03446A (fr) 1971-03-30
NL170857B (nl) 1982-08-02
IL33859A (en) 1973-01-30
PL80541B1 (pl) 1975-08-30
BE747493A (fr) 1970-09-17
NL170857C (nl) 1983-01-03
BR7017488D0 (pt) 1973-02-13
AU8549975A (en) 1975-12-18
NL172510C (nl) 1983-09-16
US3987052A (en) 1976-10-19
FR2034999B1 (xx) 1973-07-13
CH535788A (de) 1973-04-15
AU490626B2 (en) 1975-12-18
ES376689A1 (es) 1972-05-01
DE2012190A1 (de) 1970-09-24
AU8550075A (en) 1975-12-18
DE2012190B2 (de) 1980-03-06
IL33859A0 (en) 1970-04-20
FR2034999A1 (fr) 1970-12-18
NL7003750A (nl) 1970-09-21

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