GB1323277A - Triazolobenzodiazepines - Google Patents
TriazolobenzodiazepinesInfo
- Publication number
- GB1323277A GB1323277A GB1667072A GB1667072A GB1323277A GB 1323277 A GB1323277 A GB 1323277A GB 1667072 A GB1667072 A GB 1667072A GB 1667072 A GB1667072 A GB 1667072A GB 1323277 A GB1323277 A GB 1323277A
- Authority
- GB
- United Kingdom
- Prior art keywords
- alkyl
- compounds
- oxides
- triazolobenzodiazepines
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
1323277 Triazolobenzodiazepines UPJOHN CO 11 April 1972 [10 May 1971] 16670/72 Heading C2C Compounds of the general formula (R = 5-6 membered heteroaromatic radical; A=R, C 5-7 cycloalkyl, R 4 R 5 Ph; R 4,5 =H, C 1-3 alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl or alkanoylamino, halogen, NO 2 , CN, CF 3 , NH 2 , di-(C 1-3 alkyl) amino; R 1 =H, C 1-3 alkyl), their 5-oxides and acid addition salts of the compounds and 5-oxides are prepared by reacting a compound of the formula with RCONHNH 2 , optionally followed by oxidation and/or salt formation. The above compounds are sedatives, hypnotics, anticonvulsants, tranquillizers and muscle relaxants, and increase growth rate and feed efficiency of livestock. They may be administered in the form of pharmaceutical or veterinary preparations or food premixes containing them in association with a carrier.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US14206871A | 1971-05-10 | 1971-05-10 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1323277A true GB1323277A (en) | 1973-07-11 |
Family
ID=22498436
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB1667072A Expired GB1323277A (en) | 1971-05-10 | 1972-04-11 | Triazolobenzodiazepines |
Country Status (9)
| Country | Link |
|---|---|
| JP (1) | JPS554109B1 (en) |
| AU (1) | AU456535B2 (en) |
| BE (1) | BE783274A (en) |
| CH (1) | CH573432A5 (en) |
| DE (1) | DE2222068C2 (en) |
| FR (1) | FR2137685B1 (en) |
| GB (1) | GB1323277A (en) |
| NL (1) | NL7206300A (en) |
| ZA (1) | ZA722628B (en) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4455307A (en) * | 1982-01-04 | 1984-06-19 | The Upjohn Company | Antihypertensive use of triazolobenzodiazepines |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AT338799B (en) * | 1974-03-02 | 1977-09-12 | Boehringer Sohn Ingelheim | PROCESS FOR PREPARING NEW SUBSTITUTED 6-ARYL-4H-S-TRIAZOLO- (3,4C) -THIENO- (2,3E) -1,4-DIAZEPINE AND THEIR SALTS |
| US3894025A (en) * | 1974-03-21 | 1975-07-08 | Upjohn Co | 1-Piperazino-6-phenyl-4H-s-triazolo{8 4,3-a{9 {8 1,4{9 -benzodiazepine compounds |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3987052A (en) * | 1969-03-17 | 1976-10-19 | The Upjohn Company | 6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines |
| DE1955349C2 (en) * | 1969-11-04 | 1982-01-28 | Takeda Chemical Industries, Ltd., Osaka | s-Triazolo [4,3-a] [1,4] benzodiazepines |
-
1972
- 1972-04-11 GB GB1667072A patent/GB1323277A/en not_active Expired
- 1972-04-18 ZA ZA722628A patent/ZA722628B/en unknown
- 1972-04-18 AU AU41282/72A patent/AU456535B2/en not_active Expired
- 1972-05-02 JP JP4340572A patent/JPS554109B1/ja active Pending
- 1972-05-05 DE DE2222068A patent/DE2222068C2/en not_active Expired
- 1972-05-09 FR FR7216572A patent/FR2137685B1/fr not_active Expired
- 1972-05-10 CH CH698972A patent/CH573432A5/xx not_active IP Right Cessation
- 1972-05-10 BE BE783274A patent/BE783274A/en not_active IP Right Cessation
- 1972-05-10 NL NL7206300A patent/NL7206300A/xx unknown
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4455307A (en) * | 1982-01-04 | 1984-06-19 | The Upjohn Company | Antihypertensive use of triazolobenzodiazepines |
Also Published As
| Publication number | Publication date |
|---|---|
| AU456535B2 (en) | 1974-12-04 |
| FR2137685A1 (en) | 1972-12-29 |
| AU4128272A (en) | 1973-10-25 |
| FR2137685B1 (en) | 1976-04-16 |
| DE2222068C2 (en) | 1984-06-14 |
| ZA722628B (en) | 1973-01-31 |
| NL7206300A (en) | 1972-11-14 |
| CH573432A5 (en) | 1976-03-15 |
| BE783274A (en) | 1972-11-10 |
| JPS554109B1 (en) | 1980-01-29 |
| DE2222068A1 (en) | 1972-11-23 |
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| GB1225677A (en) | ||
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed | ||
| PCNP | Patent ceased through non-payment of renewal fee |