AU2015340305B2 - Diheteroaryl histone deacetylase inhibitors and their use in therapy - Google Patents

Diheteroaryl histone deacetylase inhibitors and their use in therapy Download PDF

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Publication number
AU2015340305B2
AU2015340305B2 AU2015340305A AU2015340305A AU2015340305B2 AU 2015340305 B2 AU2015340305 B2 AU 2015340305B2 AU 2015340305 A AU2015340305 A AU 2015340305A AU 2015340305 A AU2015340305 A AU 2015340305A AU 2015340305 B2 AU2015340305 B2 AU 2015340305B2
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alkyl
amino
pyrazin
compound according
heteroaryl
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AU2015340305A1 (en
Inventor
Alexander Richard Liam Cecil
Somhairle Maccormick
William John NODES
Stephen Joseph Shuttleworth
Franck Alexandre Silva
Cyrille Davy Tomassi
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Karus Therapeutics Ltd
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Karus Therapeutics Ltd
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    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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AU2015340305A 2014-10-29 2015-10-29 Diheteroaryl histone deacetylase inhibitors and their use in therapy Ceased AU2015340305B2 (en)

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GB1419228.0 2014-10-29
GBGB1419228.0A GB201419228D0 (en) 2014-10-29 2014-10-29 Compounds
PCT/GB2015/053260 WO2016067040A1 (en) 2014-10-29 2015-10-29 Diheteroaryl histone deacetylase inhibitors and their use in therapy

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AU2015340305A1 AU2015340305A1 (en) 2017-05-18
AU2015340305B2 true AU2015340305B2 (en) 2018-12-06

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US (1) US10407435B2 (enExample)
EP (1) EP3212625A1 (enExample)
JP (1) JP2017532357A (enExample)
KR (1) KR20170081194A (enExample)
CN (1) CN107001340A (enExample)
AU (1) AU2015340305B2 (enExample)
BR (1) BR112017008794A2 (enExample)
CA (1) CA2966072A1 (enExample)
GB (1) GB201419228D0 (enExample)
IL (1) IL251860A0 (enExample)
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IN2015DN03235A (enExample) 2012-11-07 2015-10-02 Karus Therapeutics Ltd
ES2688815T3 (es) 2013-05-10 2018-11-07 Karus Therapeutics Limited Inhibidores de histona desacetilasa novedosos
GB201419264D0 (en) 2014-10-29 2014-12-10 Karus Therapeutics Ltd Compounds
GB201419228D0 (en) 2014-10-29 2014-12-10 Karus Therapeutics Ltd Compounds
US20180141897A1 (en) 2014-12-08 2018-05-24 The Research Foundation For The State University Of New York Anti-fungals targeting the synthesis of fungal shingolipids
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