AU2008317400B2 - Methods of using (+)-1,4-dihydro-7-[(3S,4S)-3-methoxy-4-(methylamino) -1-pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3- carboxylic acid in combination therapy - Google Patents
Methods of using (+)-1,4-dihydro-7-[(3S,4S)-3-methoxy-4-(methylamino) -1-pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3- carboxylic acid in combination therapy Download PDFInfo
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- AU2008317400B2 AU2008317400B2 AU2008317400A AU2008317400A AU2008317400B2 AU 2008317400 B2 AU2008317400 B2 AU 2008317400B2 AU 2008317400 A AU2008317400 A AU 2008317400A AU 2008317400 A AU2008317400 A AU 2008317400A AU 2008317400 B2 AU2008317400 B2 AU 2008317400B2
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- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
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- A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
- A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
- A61K31/7068—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid
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Landscapes
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- General Health & Medical Sciences (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AU2014277779A AU2014277779B2 (en) | 2007-10-22 | 2014-12-18 | METHODS OF USING (+)-1,4-DIHYDRO-7-[(3s,4s)-3-METHOXY-4-(METHYLAMINO)-1-PYRROLIDINYL]-4-OXO-1-(2-THIAZOLYL)-1,8-NAPHTHYRIDINE-3-CARBOXYLIC ACID IN COMBINATION THERAPY |
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| US98176607P | 2007-10-22 | 2007-10-22 | |
| US60/981,766 | 2007-10-22 | ||
| PCT/US2008/011960 WO2009054935A1 (en) | 2007-10-22 | 2008-10-21 | Methods of using (+)-1,4-dihydro-7-[(3s,4s)-3-methoxy-4-(methylamino)-1-pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3-carboxylic acid in combination therapy |
Related Child Applications (1)
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| AU2014277779A Division AU2014277779B2 (en) | 2007-10-22 | 2014-12-18 | METHODS OF USING (+)-1,4-DIHYDRO-7-[(3s,4s)-3-METHOXY-4-(METHYLAMINO)-1-PYRROLIDINYL]-4-OXO-1-(2-THIAZOLYL)-1,8-NAPHTHYRIDINE-3-CARBOXYLIC ACID IN COMBINATION THERAPY |
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| AU2008317400A1 AU2008317400A1 (en) | 2009-04-30 |
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| AU2008317400A Ceased AU2008317400B2 (en) | 2007-10-22 | 2008-10-21 | Methods of using (+)-1,4-dihydro-7-[(3S,4S)-3-methoxy-4-(methylamino) -1-pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3- carboxylic acid in combination therapy |
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| JP (3) | JP6029808B2 (enExample) |
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| CA (1) | CA2703044C (enExample) |
| MX (1) | MX2010004350A (enExample) |
| WO (1) | WO2009054935A1 (enExample) |
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|---|---|---|---|---|
| WO2005089757A1 (en) | 2004-03-15 | 2005-09-29 | Sunesis Pharmaceuticals, Inc. | Sns-595 and methods of using the same |
| US8580814B2 (en) | 2006-04-03 | 2013-11-12 | Sunesis Pharmaceuticals, Inc. | Methods of using (+)-1,4-dihydro-7-[(3S,4S)-3-methoxy-4-(methylamino)-1-pyrrolidinyl]-4- oxo-1-(2-thiazolyl)-1,8-naphthyridine-3-carboxylic acid for treatment of cancer |
| CA2654876A1 (en) | 2006-06-12 | 2007-12-21 | Sunesis Pharmaceuticals, Inc. | 1-8-naphthyridine compounds for the treatment of cancer |
| US20100048609A1 (en) * | 2006-08-01 | 2010-02-25 | Jacobs Jeffrey W | Pharmaceutical dosage forms for (+)-1,4-dihydro-7-[(3s,4s)-3-methoxy-4-(methylamino)-1-pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3-carboxylic acid |
| CA2708264C (en) | 2007-12-10 | 2018-07-03 | Sunesis Pharmaceuticals, Inc. | Methods of using (+)-1,4-dihydro-7-[(3s,4s)-3-methoxy-4-(methylamino)-1-pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3-carboxylic acid for treatment of antecedent hematologic disorders |
| KR20170090535A (ko) | 2008-12-31 | 2017-08-07 | 선에시스 파마슈티컬스 인코포레이티드 | (＋)-1,4-다이하이드로-7-［(3ｓ,4ｓ)-3-메톡시-4-(메틸아미노)-1-피롤리딘일］-4-옥소-1-(2-티아졸릴)-1,8-나프티리딘-3-카복실산의 제조 방법 |
| UA110465C2 (en) * | 2009-09-04 | 2016-01-12 | Sunesis Pharmaceutecals Inc | Stable sns-595 composition |
| TW201120037A (en) * | 2009-10-26 | 2011-06-16 | Sunesis Pharmaceuticals Inc | Compounds and methods for treatment of cancer |
| WO2025033367A1 (ja) * | 2023-08-04 | 2025-02-13 | 湧永製薬株式会社 | 抗腫瘍剤併用療法 |
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| WO2007028171A1 (en) * | 2005-09-02 | 2007-03-08 | Sunesis Pharmaceuticals, Inc. | Methods of using (+)-1,4-dihydro-7-[(3s,4s)-3-methoxy-4-(methylamino)-1-pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3-carboxylic acid for treatment of cancer |
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| KR20170090535A (ko) | 2008-12-31 | 2017-08-07 | 선에시스 파마슈티컬스 인코포레이티드 | (＋)-1,4-다이하이드로-7-［(3ｓ,4ｓ)-3-메톡시-4-(메틸아미노)-1-피롤리딘일］-4-옥소-1-(2-티아졸릴)-1,8-나프티리딘-3-카복실산의 제조 방법 |
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- 2008-10-21 JP JP2010531016A patent/JP6029808B2/ja not_active Expired - Fee Related
- 2008-10-21 AU AU2008317400A patent/AU2008317400B2/en not_active Ceased
- 2008-10-21 CN CN201310524590.3A patent/CN103720701A/zh active Pending
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- 2008-10-21 EP EP08843165.5A patent/EP2214662B1/en not_active Not-in-force
- 2008-10-21 MX MX2010004350A patent/MX2010004350A/es active IP Right Grant
- 2008-10-21 WO PCT/US2008/011960 patent/WO2009054935A1/en not_active Ceased
- 2008-10-21 EP EP16177763.6A patent/EP3141250A1/en not_active Withdrawn
- 2008-10-21 CN CN2008801223989A patent/CN101909613A/zh active Pending
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2013
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Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005089756A1 (en) * | 2004-03-15 | 2005-09-29 | Sunesis Pharmaceuticals, Inc. | Sns-595 and methods of using the same |
| WO2007028171A1 (en) * | 2005-09-02 | 2007-03-08 | Sunesis Pharmaceuticals, Inc. | Methods of using (+)-1,4-dihydro-7-[(3s,4s)-3-methoxy-4-(methylamino)-1-pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3-carboxylic acid for treatment of cancer |
Also Published As
| Publication number | Publication date |
|---|---|
| JP6029808B2 (ja) | 2016-11-24 |
| AU2008317400A1 (en) | 2009-04-30 |
| CN101909613A (zh) | 2010-12-08 |
| US20160317510A1 (en) | 2016-11-03 |
| JP2015057397A (ja) | 2015-03-26 |
| MX2010004350A (es) | 2010-05-19 |
| EP2214662A1 (en) | 2010-08-11 |
| EP2214662B1 (en) | 2016-07-13 |
| WO2009054935A1 (en) | 2009-04-30 |
| US20140205679A1 (en) | 2014-07-24 |
| US8518872B2 (en) | 2013-08-27 |
| JP2011500805A (ja) | 2011-01-06 |
| JP2017031197A (ja) | 2017-02-09 |
| EP3141250A1 (en) | 2017-03-15 |
| CA2703044C (en) | 2016-05-10 |
| CA2703044A1 (en) | 2009-04-30 |
| US20100297142A1 (en) | 2010-11-25 |
| CN103720701A (zh) | 2014-04-16 |
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