AU2007341937B2 - Polycyclic heteroaryl substituted triazoles useful as Axl inhibitors - Google Patents

Polycyclic heteroaryl substituted triazoles useful as Axl inhibitors Download PDF

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AU2007341937B2
AU2007341937B2 AU2007341937A AU2007341937A AU2007341937B2 AU 2007341937 B2 AU2007341937 B2 AU 2007341937B2 AU 2007341937 A AU2007341937 A AU 2007341937A AU 2007341937 A AU2007341937 A AU 2007341937A AU 2007341937 B2 AU2007341937 B2 AU 2007341937B2
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optionally substituted
benzo
group
dihydro
heteroaryl
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AU2007341937A1 (en
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Pingyu Ding
Dane Goff
Thilo Heckrodt
Sacha Holland
Joane Litvak
Rajinder Singh
Jiaxin Yu
Jing Zhang
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Rigel Pharmaceuticals Inc
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Rigel Pharmaceuticals Inc
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AU2007341937A 2006-12-29 2007-12-29 Polycyclic heteroaryl substituted triazoles useful as Axl inhibitors Active AU2007341937B2 (en)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US88285006P 2006-12-29 2006-12-29
US60/882,850 2006-12-29
US89540007P 2007-03-16 2007-03-16
US60/895,400 2007-03-16
US97093107P 2007-09-07 2007-09-07
US60/970,931 2007-09-07
PCT/US2007/089177 WO2008083367A2 (en) 2006-12-29 2007-12-29 Polycyclic heteroaryl substituted triazoles useful as axl inhibitors

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AU2007341937A1 AU2007341937A1 (en) 2008-07-10
AU2007341937B2 true AU2007341937B2 (en) 2013-07-11

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AU2007341937A Active AU2007341937B2 (en) 2006-12-29 2007-12-29 Polycyclic heteroaryl substituted triazoles useful as Axl inhibitors

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US (5) US7709482B2 (enExample)
EP (1) EP2078010B1 (enExample)
JP (2) JP5546250B2 (enExample)
CN (1) CN101622246B (enExample)
AU (1) AU2007341937B2 (enExample)
CA (1) CA2710234C (enExample)
CY (1) CY1115188T1 (enExample)
DK (1) DK2078010T3 (enExample)
ES (1) ES2460894T3 (enExample)
HR (1) HRP20140378T1 (enExample)
ME (1) ME01832B (enExample)
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PT (1) PT2078010E (enExample)
RS (1) RS53281B (enExample)
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JP2008543888A (ja) * 2005-06-24 2008-12-04 ギリアード サイエンシーズ， インコーポレイテッド ピリド（３，２−ｄ）ピリミジン、およびＣ型肝炎を治療するのに有用な医薬組成物
US7884119B2 (en) * 2005-09-07 2011-02-08 Rigel Pharmaceuticals, Inc. Triazole derivatives useful as Axl inhibitors
US8338435B2 (en) * 2006-07-20 2012-12-25 Gilead Sciences, Inc. Substituted pyrido(3,2-D) pyrimidines and pharmaceutical compositions for treating viral infections
TW200840584A (en) * 2006-12-26 2008-10-16 Gilead Sciences Inc Pyrido(3,2-d)pyrimidines useful for treating viral infections
EP2114954B1 (en) 2006-12-29 2013-02-13 Rigel Pharmaceuticals, Inc. Bicyclic aryl and bicyclic heteroaryl substituted triazoles useful as axl inhibitors
AU2007342005A1 (en) * 2006-12-29 2008-07-10 Rigel Pharmaceuticals, Inc. N3-heteroaryl substituted triazoles and N5-heteroaryl substituted triazoles useful as Axl inhibitors
ES2404668T3 (es) 2006-12-29 2013-05-28 Rigel Pharmaceuticals, Inc. Triazoles sustituidos con arilo bicíclico puenteado y heteroarilo bicíclico puenteado, útiles como agentes inhibidores del axl
PT2078010E (pt) * 2006-12-29 2014-05-07 Rigel Pharmaceuticals Inc Triazoles substituídos com heteroarilos policíclicos úteis como inibidores de axl
JP2010514810A (ja) 2006-12-29 2010-05-06 ライジェル ファーマシューティカルズ， インコーポレイテッド Ａｘｌインヒビターとして有用な置換トリアゾール
CA2704052C (en) * 2007-10-26 2015-04-21 Rigel Pharmaceuticals, Inc. Polycyclic aryl substituted triazoles and polycyclic heteroaryl substituted triazoles useful as axl inhibitors
HUE030912T2 (en) 2008-02-15 2017-06-28 Rigel Pharmaceuticals Inc Pyrimidine-2-amine compounds and their use as inhibitors of yak kinases
JP5592884B2 (ja) * 2008-07-09 2014-09-17 ライジェル ファーマシューティカルズ， インコーポレイテッド Ａｘｌ阻害剤として有用な多環式ヘテロアリール置換トリアゾール
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