AU2002248339B2 - Substituted Arylamine Derivatives and Methods of Use - Google Patents

Substituted Arylamine Derivatives and Methods of Use Download PDF

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Publication number
AU2002248339B2
AU2002248339B2 AU2002248339A AU2002248339A AU2002248339B2 AU 2002248339 B2 AU2002248339 B2 AU 2002248339B2 AU 2002248339 A AU2002248339 A AU 2002248339A AU 2002248339 A AU2002248339 A AU 2002248339A AU 2002248339 B2 AU2002248339 B2 AU 2002248339B2
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AU
Australia
Prior art keywords
phenyl
optionally substituted
methyl
trifluoromethyl
amino
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Ceased
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AU2002248339A
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AU2002248339A1 (en
Inventor
Shon Booker
Guolin Cai
Guoqing Chen
Michael Croghan
Lucian Dipietro
Celia Dominguez
Daniel Elbaum
Julie Germain
Qi Huang
Joseph L. Kim
Tae-Seong Kim
Vinod F. Patel
Leon M. Smith
Andrew Tasker
Ning Xi
Shimin Xu
Chester Chenguang Yuan
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Amgen Inc
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Amgen Inc
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Publication of AU2002248339B2 publication Critical patent/AU2002248339B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
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  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • General Health & Medical Sciences (AREA)
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AU2002248339A 2001-01-12 2002-01-11 Substituted Arylamine Derivatives and Methods of Use Ceased AU2002248339B2 (en)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US26136001P 2001-01-12 2001-01-12
US60/261,360 2001-01-12
US32368601P 2001-09-19 2001-09-19
US60/323,686 2001-09-19
US10/046,526 US20020147198A1 (en) 2001-01-12 2002-01-10 Substituted arylamine derivatives and methods of use
US10/046,526 2002-01-10
PCT/US2002/000742 WO2002055501A2 (en) 2001-01-12 2002-01-11 N-pyridyl carboxamide derivatives and pharmaceutical compositions containing them

Publications (2)

Publication Number Publication Date
AU2002248339A1 AU2002248339A1 (en) 2003-02-06
AU2002248339B2 true AU2002248339B2 (en) 2005-07-28

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AU2002248339A Ceased AU2002248339B2 (en) 2001-01-12 2002-01-11 Substituted Arylamine Derivatives and Methods of Use

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US (1) US20020147198A1 (enExample)
EP (1) EP1358161A2 (enExample)
JP (1) JP2004531473A (enExample)
AU (1) AU2002248339B2 (enExample)
CA (1) CA2434274A1 (enExample)
MX (1) MXPA03006010A (enExample)
WO (1) WO2002055501A2 (enExample)

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US6995162B2 (en) 2001-01-12 2006-02-07 Amgen Inc. Substituted alkylamine derivatives and methods of use
US6878714B2 (en) * 2001-01-12 2005-04-12 Amgen Inc. Substituted alkylamine derivatives and methods of use
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US7148357B2 (en) * 2002-07-31 2006-12-12 Schering Ag VEGFR-2 and VEGFR-3 inhibitory anthranilamide pyridines
CA2493026C (en) * 2002-07-31 2011-05-24 Bayer Schering Pharma Aktiengesellschaft Vegfr-2 and vegfr-3 inhibitory anthranilamide pyridines
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