AU2002217356A1 - Novel 2,3-benzodiazepine derivatives and pharmaceutical compositions containing the same as the active ingredient - Google Patents
Novel 2,3-benzodiazepine derivatives and pharmaceutical compositions containing the same as the active ingredientInfo
- Publication number
- AU2002217356A1 AU2002217356A1 AU2002217356A AU1735602A AU2002217356A1 AU 2002217356 A1 AU2002217356 A1 AU 2002217356A1 AU 2002217356 A AU2002217356 A AU 2002217356A AU 1735602 A AU1735602 A AU 1735602A AU 2002217356 A1 AU2002217356 A1 AU 2002217356A1
- Authority
- AU
- Australia
- Prior art keywords
- sup
- sub
- novel
- group
- active ingredient
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- RPBDCDQMCRHNLM-UHFFFAOYSA-N C1=NNC=C2C=CC=CC2=C1 Chemical class C1=NNC=C2C=CC=CC2=C1 RPBDCDQMCRHNLM-UHFFFAOYSA-N 0.000 title abstract 2
- 239000004480 active ingredient Substances 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 3
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 125000001309 chloro group Chemical group Cl* 0.000 abstract 2
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 abstract 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
- 239000003158 myorelaxant agent Substances 0.000 abstract 1
- 230000000324 neuroprotective effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/02—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Addiction (AREA)
- Psychology (AREA)
- Otolaryngology (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HU0004994 | 2000-12-21 | ||
| HU0004994A HU225100B1 (hu) | 2000-12-21 | 2000-12-21 | 2,3-Benzodiazepinszármazékok, ilyen hatóanyagot tartalmazó gyógyászati készítmények és alkalmazásuk |
| PCT/HU2001/000151 WO2002050044A1 (en) | 2000-12-21 | 2001-12-19 | Novel 2,3-benzodiazepine derivatives and pharmaceutical compositions containing the same as the active ingredient |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2002217356A1 true AU2002217356A1 (en) | 2002-07-01 |
Family
ID=89978876
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2002217356A Abandoned AU2002217356A1 (en) | 2000-12-21 | 2001-12-19 | Novel 2,3-benzodiazepine derivatives and pharmaceutical compositions containing the same as the active ingredient |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US7189711B2 (hu) |
| EP (1) | EP1351942B1 (hu) |
| JP (1) | JP4201252B2 (hu) |
| AT (1) | ATE271548T1 (hu) |
| AU (1) | AU2002217356A1 (hu) |
| BG (1) | BG66199B1 (hu) |
| CA (1) | CA2431761C (hu) |
| CZ (1) | CZ301371B6 (hu) |
| DE (1) | DE60104448T2 (hu) |
| DK (1) | DK1351942T3 (hu) |
| EA (1) | EA005867B1 (hu) |
| ES (1) | ES2225412T3 (hu) |
| HU (1) | HU225100B1 (hu) |
| PL (1) | PL211495B1 (hu) |
| PT (1) | PT1351942E (hu) |
| RO (1) | RO121268B1 (hu) |
| SK (1) | SK286620B6 (hu) |
| TR (1) | TR200402493T4 (hu) |
| UA (1) | UA74615C2 (hu) |
| WO (1) | WO2002050044A1 (hu) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HUP0302449A3 (en) * | 2003-08-04 | 2005-06-28 | Egis Gyogyszergyar Nyilvanosan | 8-chloro-2,3-benzodiazepine derivatives, pharmaceutical compositions containing them and process for producing them |
| CA2633804A1 (en) * | 2005-12-30 | 2007-07-12 | Egis Gyogyszergyar Nyilvanosan Mukodo Reszvenytarsasag | Optical isomers of dihydro-2,3-benzodiazepines and their stereoselective synthesis |
| US9890147B2 (en) * | 2012-08-16 | 2018-02-13 | Bayer Pharma Aktiengesellshaft | 2,3-benzodiazepines |
| WO2014202578A1 (de) * | 2013-06-17 | 2014-12-24 | Bayer Pharma Aktiengesellschaft | Substituierte phenyl-2,3-benzodiazepine |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU191698B (en) * | 1984-07-27 | 1987-03-30 | Gyogyszerkutato Intezet | Process for producing new 1-aryl-5h-2beta-benzodiazepines |
| HU219778B (hu) * | 1990-12-21 | 2001-07-30 | Gyógyszerkutató Intézet Közös Vállalat | Eljárás N-acil-2,3-benzodiazepin-származékok, savaddíciós sóik és az ezeket tartalmazó gyógyászati készítmények előállítására, valamint a vegyületek egy csoportja, és az ezeket tartalmazó gyógyászati készítmények |
| DE19604920A1 (de) | 1996-02-01 | 1997-08-07 | Schering Ag | Neue 2,3-Benzodiazepinderivate, deren Herstellung und Verwendung als Arzneimittel |
| US5891871A (en) * | 1996-03-21 | 1999-04-06 | Cocensys, Inc. | Substituted 2,3-benzodiazepin-4-ones and the use thereof |
| HU9600871D0 (en) * | 1996-04-04 | 1996-05-28 | Gyogyszerkutato Intezet | New 2,3-benzodiazepine derivatives |
| HU227128B1 (en) | 1999-07-07 | 2010-07-28 | Egyt Gyogyszervegyeszeti Gyar | New 2,3-benzodiazepine derivatives |
| RU2325811C2 (ru) | 2006-06-28 | 2008-06-10 | Общество С Ограниченной Ответственностью "Фито-Маг" | Способ хранения плодоовощной и растениеводческой продукции |
-
2000
- 2000-12-21 HU HU0004994A patent/HU225100B1/hu not_active IP Right Cessation
-
2001
- 2001-12-19 DK DK01271364T patent/DK1351942T3/da active
- 2001-12-19 PL PL362029A patent/PL211495B1/pl unknown
- 2001-12-19 RO ROA200300539A patent/RO121268B1/ro unknown
- 2001-12-19 DE DE60104448T patent/DE60104448T2/de not_active Expired - Lifetime
- 2001-12-19 AT AT01271364T patent/ATE271548T1/de not_active IP Right Cessation
- 2001-12-19 US US10/450,898 patent/US7189711B2/en not_active Expired - Fee Related
- 2001-12-19 UA UA2003076874A patent/UA74615C2/uk unknown
- 2001-12-19 CZ CZ20031680A patent/CZ301371B6/cs not_active IP Right Cessation
- 2001-12-19 ES ES01271364T patent/ES2225412T3/es not_active Expired - Lifetime
- 2001-12-19 PT PT01271364T patent/PT1351942E/pt unknown
- 2001-12-19 CA CA2431761A patent/CA2431761C/en not_active Expired - Fee Related
- 2001-12-19 AU AU2002217356A patent/AU2002217356A1/en not_active Abandoned
- 2001-12-19 SK SK788-2003A patent/SK286620B6/sk not_active IP Right Cessation
- 2001-12-19 EP EP01271364A patent/EP1351942B1/en not_active Expired - Lifetime
- 2001-12-19 TR TR2004/02493T patent/TR200402493T4/xx unknown
- 2001-12-19 EA EA200300691A patent/EA005867B1/ru not_active IP Right Cessation
- 2001-12-19 WO PCT/HU2001/000151 patent/WO2002050044A1/en active IP Right Grant
- 2001-12-19 JP JP2002551541A patent/JP4201252B2/ja not_active Expired - Fee Related
-
2003
- 2003-06-20 BG BG107932A patent/BG66199B1/bg unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2431761A1 (en) | 2002-06-27 |
| TR200402493T4 (tr) | 2004-12-21 |
| RO121268B1 (ro) | 2007-02-28 |
| SK286620B6 (sk) | 2009-02-05 |
| PT1351942E (pt) | 2004-11-30 |
| SK7882003A3 (en) | 2003-11-04 |
| US7189711B2 (en) | 2007-03-13 |
| ES2225412T3 (es) | 2005-03-16 |
| DK1351942T3 (da) | 2004-11-22 |
| EP1351942B1 (en) | 2004-07-21 |
| EP1351942A1 (en) | 2003-10-15 |
| JP4201252B2 (ja) | 2008-12-24 |
| WO2002050044A1 (en) | 2002-06-27 |
| HU225100B1 (hu) | 2006-06-28 |
| CA2431761C (en) | 2010-05-25 |
| CZ20031680A3 (cs) | 2003-11-12 |
| BG107932A (bg) | 2004-02-27 |
| PL211495B1 (pl) | 2012-05-31 |
| JP2004516284A (ja) | 2004-06-03 |
| HU0004994D0 (en) | 2001-03-28 |
| PL362029A1 (en) | 2004-10-18 |
| CZ301371B6 (cs) | 2010-02-03 |
| US20040092510A1 (en) | 2004-05-13 |
| ATE271548T1 (de) | 2004-08-15 |
| BG66199B1 (bg) | 2012-01-31 |
| DE60104448T2 (de) | 2005-07-28 |
| UA74615C2 (en) | 2006-01-16 |
| EA200300691A1 (ru) | 2003-12-25 |
| DE60104448D1 (de) | 2004-08-26 |
| HUP0004994A2 (hu) | 2002-11-28 |
| EA005867B1 (ru) | 2005-06-30 |
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