AU2001270932A1 - Particulate composition of eletriptan showing a sigmoidal pattern of controlled release - Google Patents

Particulate composition of eletriptan showing a sigmoidal pattern of controlled release

Info

Publication number
AU2001270932A1
AU2001270932A1 AU2001270932A AU7093201A AU2001270932A1 AU 2001270932 A1 AU2001270932 A1 AU 2001270932A1 AU 2001270932 A AU2001270932 A AU 2001270932A AU 7093201 A AU7093201 A AU 7093201A AU 2001270932 A1 AU2001270932 A1 AU 2001270932A1
Authority
AU
Australia
Prior art keywords
composition
eletriptan
pharmaceutically acceptable
core
drug
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001270932A
Other languages
English (en)
Inventor
Manaud Pierre Frederick De Raspide
Ross James Macrae
Mathias Walther
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Ltd
Original Assignee
Pfizer Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ltd filed Critical Pfizer Ltd
Publication of AU2001270932A1 publication Critical patent/AU2001270932A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5021—Organic macromolecular compounds
    • A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Electroluminescent Light Sources (AREA)
  • Luminescent Compositions (AREA)
AU2001270932A 2000-08-02 2001-07-18 Particulate composition of eletriptan showing a sigmoidal pattern of controlled release Abandoned AU2001270932A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0018968.8A GB0018968D0 (en) 2000-08-02 2000-08-02 Particulate composition
GB0018968.8 2000-08-02
PCT/IB2001/001279 WO2002009675A1 (en) 2000-08-02 2001-07-18 Particulate composition of eletriptan showing a sigmoidal pattern of controlled release

Publications (1)

Publication Number Publication Date
AU2001270932A1 true AU2001270932A1 (en) 2002-02-13

Family

ID=9896843

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001270932A Abandoned AU2001270932A1 (en) 2000-08-02 2001-07-18 Particulate composition of eletriptan showing a sigmoidal pattern of controlled release

Country Status (38)

Country Link
US (1) US20020034545A1 (de)
EP (1) EP1365748B1 (de)
JP (1) JP2004505034A (de)
KR (1) KR20030024820A (de)
CN (1) CN1630511A (de)
AP (1) AP2001002233A0 (de)
AR (1) AR030099A1 (de)
AT (1) ATE308978T1 (de)
AU (1) AU2001270932A1 (de)
BG (1) BG107361A (de)
BR (1) BR0112839A (de)
CA (1) CA2417887C (de)
CZ (1) CZ2003241A3 (de)
DE (1) DE60114887T2 (de)
EA (1) EA200300110A1 (de)
EC (1) ECSP034451A (de)
EE (1) EE200300051A (de)
ES (1) ES2250429T3 (de)
GB (1) GB0018968D0 (de)
GT (1) GT200100149A (de)
HR (1) HRP20030036A2 (de)
HU (1) HUP0301453A2 (de)
IL (1) IL153494A0 (de)
IS (1) IS6649A (de)
MA (1) MA26934A1 (de)
MX (1) MXPA03000999A (de)
NO (1) NO20030498L (de)
NZ (1) NZ522976A (de)
OA (1) OA12348A (de)
PA (1) PA8523101A1 (de)
PE (1) PE20020385A1 (de)
PL (1) PL359847A1 (de)
SK (1) SK1082003A3 (de)
SV (1) SV2002000574A (de)
TN (1) TNSN01115A1 (de)
UY (1) UY26861A1 (de)
WO (1) WO2002009675A1 (de)
ZA (1) ZA200300868B (de)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20040022853A1 (en) * 2001-04-26 2004-02-05 Control Delivery Systems, Inc. Polymer-based, sustained release drug delivery system
EP1572107A1 (de) * 2002-12-16 2005-09-14 CHX Technologies Inc. Temporärer, pharmazeutisch inaktiver zahnüberzug für in situ schutz von therapeutischen dentalen wirkstoffen vor saliva und abrasion durch kauen
JP2006522790A (ja) * 2003-04-11 2006-10-05 ファイザー・インク エレトリプタンと重炭酸ナトリウムを含む医薬組み合わせ物
GB2407498B (en) * 2003-10-30 2008-06-11 Cipla Ltd Oral formulations for 5-HT receptor agonists with reduced degradation of active ingredient
WO2005120456A2 (en) * 2004-06-09 2005-12-22 Pfizer Limited Formulation of eletriptan
WO2006013431A1 (en) * 2004-07-29 2006-02-09 Pfizer Limited Stable controlled-release pharmaceutical formulation of eletriptan
US20080107727A1 (en) * 2005-01-31 2008-05-08 Katashi Nakashima Multiple Unit Oral Sustained Release Preparation and Production Method Thereof
DK1915137T3 (da) 2005-08-10 2013-11-04 Add Advanced Drug Delivery Technologies Ltd Oralt præparat med kontrolleret frisætning
US20070134322A1 (en) * 2005-12-14 2007-06-14 Forest Laboratories, Inc. Modified and pulsatile release pharmaceutical formulations of escitalopram
DE602007012236D1 (de) 2006-04-26 2011-03-10 Supernus Pharmaceuticals Inc Oxcarbazepin-zubereitungen für kontrollierte freisetzung mit sigmoidalem freisetzungsprofil
US20080226715A1 (en) * 2007-03-16 2008-09-18 Albert Cha Therapeutic compositions and methods
CA2694440A1 (en) 2007-07-25 2009-01-29 Biolex Therapeutics, Inc. Controlled release interferon drug products and treatment of hcv infection using same
KR20120110098A (ko) 2009-11-16 2012-10-09 에보니크 룀 게엠베하 고형 (메트)아크릴레이트 공중합체를 분산제에 의해 분산된 형태로 전환시키는 방법
KR20170054446A (ko) * 2014-09-09 2017-05-17 찰스톤 래보라토리즈, 인크. 약학적 조성물
GB201716716D0 (en) * 2017-10-12 2017-11-29 Univ Of Hertfordshire Higher Education Corporation Method for coating particles

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2624732B1 (fr) * 1987-12-21 1991-02-15 Synthelabo Formulation pharmaceutique a liberation prolongee
US5411745A (en) * 1994-05-25 1995-05-02 Euro-Celtique, S.A. Powder-layered morphine sulfate formulations
GB9417310D0 (en) * 1994-08-27 1994-10-19 Pfizer Ltd Therapeutic agents
GB9825988D0 (en) * 1998-11-27 1999-01-20 Pfizer Ltd Indole derivatives
GB9922963D0 (en) * 1999-09-28 1999-12-01 Pfizer Ltd Polymorphic salt
FR2795962B1 (fr) * 1999-07-08 2003-05-09 Prographarm Laboratoires Procede de fabrication de granules enrobes a gout masque et liberation immediate du principe actif
US20020044962A1 (en) * 2000-06-06 2002-04-18 Cherukuri S. Rao Encapsulation products for controlled or extended release

Also Published As

Publication number Publication date
IL153494A0 (en) 2003-07-06
HRP20030036A2 (en) 2003-04-30
JP2004505034A (ja) 2004-02-19
GT200100149A (es) 2002-06-25
EE200300051A (et) 2004-10-15
DE60114887D1 (de) 2005-12-15
AP2001002233A0 (en) 2001-09-30
BR0112839A (pt) 2003-06-24
CA2417887C (en) 2006-11-14
ZA200300868B (en) 2004-04-16
WO2002009675A9 (en) 2003-07-10
HUP0301453A2 (hu) 2003-08-28
AR030099A1 (es) 2003-08-13
NO20030498D0 (no) 2003-01-31
OA12348A (en) 2004-03-19
CA2417887A1 (en) 2002-02-07
DE60114887T2 (de) 2006-07-20
ATE308978T1 (de) 2005-11-15
MA26934A1 (fr) 2004-12-20
ES2250429T3 (es) 2006-04-16
MXPA03000999A (es) 2003-06-09
UY26861A1 (es) 2002-02-28
CN1630511A (zh) 2005-06-22
PL359847A1 (en) 2004-09-06
PA8523101A1 (es) 2002-08-26
EP1365748B1 (de) 2005-11-09
EA200300110A1 (ru) 2003-06-26
SK1082003A3 (en) 2004-09-08
ECSP034451A (es) 2003-03-10
WO2002009675A1 (en) 2002-02-07
KR20030024820A (ko) 2003-03-26
CZ2003241A3 (cs) 2004-02-18
PE20020385A1 (es) 2002-05-11
GB0018968D0 (en) 2000-09-20
IS6649A (is) 2002-12-05
US20020034545A1 (en) 2002-03-21
EP1365748A2 (de) 2003-12-03
NZ522976A (en) 2004-11-26
NO20030498L (no) 2003-01-31
SV2002000574A (es) 2002-12-02
TNSN01115A1 (fr) 2005-11-10
BG107361A (bg) 2003-06-30

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Legal Events

Date Code Title Description
MK4 Application lapsed section 142(2)(d) - no continuation fee paid for the application