ATE79620T1 - N-heterozyklische-4-piperidinamine enthaltende anti-histaminische zusammensetzungen. - Google Patents
N-heterozyklische-4-piperidinamine enthaltende anti-histaminische zusammensetzungen.Info
- Publication number
- ATE79620T1 ATE79620T1 AT87200128T AT87200128T ATE79620T1 AT E79620 T1 ATE79620 T1 AT E79620T1 AT 87200128 T AT87200128 T AT 87200128T AT 87200128 T AT87200128 T AT 87200128T AT E79620 T1 ATE79620 T1 AT E79620T1
- Authority
- AT
- Austria
- Prior art keywords
- alkyl
- substd
- alkoxy
- furanyl
- opt
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Hydrogenated Pyridines (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US82549186A | 1986-02-03 | 1986-02-03 | |
EP87200128A EP0232937B1 (fr) | 1986-02-03 | 1987-01-28 | Compositions anti-histaminiques contenant des N-hétérocyclyl-4-pipéridinamines |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE79620T1 true ATE79620T1 (de) | 1992-09-15 |
Family
ID=25244134
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT87200128T ATE79620T1 (de) | 1986-02-03 | 1987-01-28 | N-heterozyklische-4-piperidinamine enthaltende anti-histaminische zusammensetzungen. |
Country Status (26)
Country | Link |
---|---|
EP (1) | EP0232937B1 (fr) |
JP (2) | JPH0794393B2 (fr) |
CN (1) | CN1018614B (fr) |
AT (1) | ATE79620T1 (fr) |
AU (1) | AU583706B2 (fr) |
CA (1) | CA1327579C (fr) |
CY (1) | CY1865A (fr) |
DE (1) | DE3781173T2 (fr) |
DK (1) | DK173674B1 (fr) |
EG (1) | EG17993A (fr) |
ES (1) | ES2052544T3 (fr) |
FI (1) | FI870448A (fr) |
GR (1) | GR3006158T3 (fr) |
HK (1) | HK114695A (fr) |
HU (1) | HU201067B (fr) |
IE (1) | IE60885B1 (fr) |
IL (1) | IL81448A (fr) |
MA (1) | MA20868A1 (fr) |
NO (1) | NO870407L (fr) |
NZ (1) | NZ219165A (fr) |
PH (1) | PH24738A (fr) |
PT (1) | PT84234B (fr) |
TN (1) | TNSN87015A1 (fr) |
ZA (1) | ZA87744B (fr) |
ZM (1) | ZM1287A1 (fr) |
ZW (1) | ZW2087A1 (fr) |
Families Citing this family (26)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NZ223654A (en) * | 1987-03-09 | 1990-03-27 | Janssen Pharmaceutica Nv | 1-alkyl-substituted-benzimidazole-4-piperidinamines and pharmaceutical compositions |
US4897401A (en) * | 1987-06-19 | 1990-01-30 | Janssen Pharmaceutical N.V. | N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives useful in treating allergic diseases |
US4988689A (en) * | 1987-07-01 | 1991-01-29 | Janssen Pharmaceutica N.V. | ((Pharmacologically active bicyclic heterocyclic)methyl and -heteroatom) substituted hexahydro-1H-azepines and pyrrolidines |
CA1317939C (fr) * | 1987-07-01 | 1993-05-18 | Janssen Pharmaceutica Naamloze Vennootschap | Hexahydro-1h-azepines et pyrrolidines a substitution par des ((heterocyclyle bicyclique) methyle et -hetero |
PH30434A (en) * | 1989-04-07 | 1997-05-09 | Janssen Pharmaceutica Nv | Hydroxyalkylfuranyl derivatives |
IT1229231B (it) * | 1989-05-08 | 1991-07-26 | Dompe Farmaceutici Spa | Aminoimidazopiridine farmacologicamente attive |
CA2043564A1 (fr) * | 1990-07-06 | 1992-01-07 | Alfons G. M. De Knaep | 3-[(5-methyl-2-furyl)methyl]-n-(4-piperidyl)-3h-imidazo[4,5-b]pyridin-2-amine 2-hydroxypropane-1,2,3-tricarboxylate |
NZ239540A (en) * | 1990-09-24 | 1993-11-25 | Neurosearch As | 1-phenyl benzimidazole derivatives and medicaments |
AU730229B2 (en) * | 1992-09-03 | 2001-03-01 | Sepracor, Inc. | Use of norastemizole for the treatment of allergic disorders |
CA2143610C (fr) * | 1992-09-03 | 2004-08-24 | Raymond L. Woosley | Utilisation de norastemizole pour le traitement de troubles allergiques |
US5624948A (en) * | 1993-05-20 | 1997-04-29 | Kissei Pharmaceutical Co., Ltd. | 1-(2-benzimidazolyl)-1,5-diazacyclooctane compounds |
TW429256B (en) * | 1995-12-27 | 2001-04-11 | Janssen Pharmaceutica Nv | 1-(1,2-disubstituted piperidinyl)-4-(benzimidazolyl- and imidazopyridinyl)-piperidine derivatives |
NZ527200A (en) * | 1997-03-26 | 2004-12-24 | Sepracor Inc | Stable norastemizole formulations including a super disintegrant |
US5817823A (en) * | 1997-04-17 | 1998-10-06 | Sepracor Inc. | Method for synthesizing 2-substituted imidazoles |
AP1552A (en) | 1999-06-28 | 2006-01-17 | Janssen Pharmaceutica Nv | Respiratory syncytial virus replication inhibitors. |
ATE258928T1 (de) | 1999-06-28 | 2004-02-15 | Janssen Pharmaceutica Nv | Respiratorisches syncytialvirus replikation inhibitoren |
DE60033859T2 (de) * | 1999-06-28 | 2007-11-08 | Janssen Pharmaceutica N.V. | Hemmer des Respiratorischen Syncytial Virus |
GB0215293D0 (en) | 2002-07-03 | 2002-08-14 | Rega Foundation | Viral inhibitors |
US20070021404A1 (en) * | 2003-06-24 | 2007-01-25 | Dan Peters | Novel aza-ring derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
EP1706403B9 (fr) | 2003-12-22 | 2012-07-25 | K.U.Leuven Research & Development | Composes d'imidazo[4,5-c]pyridine et methodes de traitement antiviral |
SI1841765T1 (sl) | 2004-12-21 | 2009-08-31 | Gilead Sciences Inc | Imidazo(4,5-c)piridinska spojina in postopek za antivirusno zdravljenje |
JP5065908B2 (ja) * | 2004-12-24 | 2012-11-07 | プロシディオン・リミテッド | Gタンパク質結合受容体作動薬 |
JP5078869B2 (ja) | 2005-03-08 | 2012-11-21 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | ニューロキニン(nk1)拮抗物質としてのジアザ−スピロ−[4.4]−ノナン誘導体 |
PL2038275T3 (pl) | 2006-07-07 | 2010-08-31 | Gilead Sciences Inc | Nowe pochodne pirydazyny i ich zastosowanie |
UA99466C2 (en) | 2007-07-06 | 2012-08-27 | Гилиад Сайенсиз, Инк. | Crystalline pyridazine compound |
AU2009296820B2 (en) * | 2008-09-26 | 2014-03-20 | Merck Sharp & Dohme Llc | Novel cyclic benzimidazole derivatives useful anti-diabetic agents |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4219559A (en) | 1979-01-10 | 1980-08-26 | Janssen Pharmaceutica N.V. | N-Heterocyclyl-4-piperidinamines |
CA1140119A (fr) * | 1978-04-03 | 1983-01-25 | Joseph Torremans | Nouvelles n-heterocycle-4-piperidinamines |
IN156065B (fr) * | 1982-07-12 | 1985-05-04 | Janssen Pharmaceutica Nv | |
US4556660A (en) * | 1982-07-12 | 1985-12-03 | Janssen Pharmaceutica N.V. | N-(Bicyclic heterocyclyl)-4-piperidinamines |
US4634704A (en) * | 1983-10-06 | 1987-01-06 | Janssen Pharmaceutica, N.V. | Anti-allergic five membered heterocyclic ring containing N-(bicyclic heterocycyl)-4-piperidinamines |
DE3484096D1 (de) * | 1983-11-30 | 1991-03-14 | Janssen Pharmaceutica Nv | Bizyklisches heterozyklyl aufveisende n-(bizyklisches heterozyklyl-4-piperidinamine. |
PH23995A (en) * | 1984-01-09 | 1990-02-09 | Janssen Pharmaceutica Nv | 4((bicycle heterocyclyl)-methyl and hetero)piperidines |
PL144514B1 (en) * | 1984-01-09 | 1988-06-30 | Janssen Pharmaceutica Nv | Method of obtaining novel derivatives of n-/4-piperidinolo/-2-imidazoloamine |
US4588722A (en) * | 1984-01-09 | 1986-05-13 | Janssen Pharmaceutica N.V. | N-(4-piperidinyl) bicyclic condensed 2-imidazolamine derivatives |
-
1987
- 1987-01-28 EP EP87200128A patent/EP0232937B1/fr not_active Expired - Lifetime
- 1987-01-28 ES ES87200128T patent/ES2052544T3/es not_active Expired - Lifetime
- 1987-01-28 AT AT87200128T patent/ATE79620T1/de not_active IP Right Cessation
- 1987-01-28 CA CA000528342A patent/CA1327579C/fr not_active Expired - Lifetime
- 1987-01-28 DE DE8787200128T patent/DE3781173T2/de not_active Expired - Lifetime
- 1987-01-28 EG EG48/87A patent/EG17993A/xx active
- 1987-01-30 PH PH34794A patent/PH24738A/en unknown
- 1987-02-02 NO NO870407A patent/NO870407L/no unknown
- 1987-02-02 PT PT84234A patent/PT84234B/pt unknown
- 1987-02-02 FI FI870448A patent/FI870448A/fi not_active Application Discontinuation
- 1987-02-02 ZM ZM12/87A patent/ZM1287A1/xx unknown
- 1987-02-02 AU AU68218/87A patent/AU583706B2/en not_active Expired
- 1987-02-02 ZA ZA87744A patent/ZA87744B/xx unknown
- 1987-02-02 IL IL81448A patent/IL81448A/xx not_active IP Right Cessation
- 1987-02-02 MA MA21102A patent/MA20868A1/fr unknown
- 1987-02-02 JP JP62020600A patent/JPH0794393B2/ja not_active Expired - Lifetime
- 1987-02-02 ZW ZW20/87A patent/ZW2087A1/xx unknown
- 1987-02-02 HU HU87354A patent/HU201067B/hu unknown
- 1987-02-02 DK DK198700541A patent/DK173674B1/da not_active IP Right Cessation
- 1987-02-02 IE IE25887A patent/IE60885B1/en not_active IP Right Cessation
- 1987-02-03 CN CN87100563A patent/CN1018614B/zh not_active Expired
- 1987-02-03 TN TNTNSN87015A patent/TNSN87015A1/fr unknown
- 1987-02-04 NZ NZ219165A patent/NZ219165A/en unknown
-
1992
- 1992-11-05 GR GR920402478T patent/GR3006158T3/el unknown
-
1994
- 1994-10-03 JP JP6260917A patent/JPH0819126B2/ja not_active Expired - Lifetime
-
1995
- 1995-07-13 HK HK114695A patent/HK114695A/xx not_active IP Right Cessation
-
1996
- 1996-04-05 CY CY186596A patent/CY1865A/xx unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EG17993A (en) | Anti-histaminic compositions containing n-heterocyclyl-4-piperidinanines | |
CA2498143A1 (fr) | Composition antimicrobienne et sa methode d'utilisation | |
DE60123277D1 (de) | Makrolidantibiotika | |
UY25459A1 (es) | Procedimiento para preparar una forma cristalina del acido 7 -([1a, 5a, 6a]-6-amino-3-azabiciclo [3, 1, 0] hex-3-il)-6-fl uor-1-(2,4-difluorofenil)-1, 4-dihidro-4-oxo-1, 8-naftiridin -3-carboxilico anhidro, sal del acido metanosulfonico | |
SE0002476D0 (sv) | New compounds | |
NO912414D0 (no) | Forbindelse med mavesyreinhiberende effekt og fremgangsmaate for dens fremstilling. | |
DK1340757T3 (da) | 1-methylcarbapenemderivater | |
UY26459A1 (es) | 3,4-dihidroquinazolinas 5,6-disustituidas | |
FI872930A0 (fi) | Analogiamenetelmä ripulinvastaisten 4-(bentsoyyliamino)piperidiinibutaaniamidijohdannaisten valmistamiseksi | |
CA2425319A1 (fr) | Traitement et prophylaxie de maladies et d'infections des porcs et de la volaille | |
RU2003104017A (ru) | Ингибиторы тромбина, содержащие аминоизохинолиновую группу | |
HUT56549A (en) | Process for producing new imidazole derivatives and pharmaceutical compositions comprising such imidazole derivatives as active ingredient | |
RU2021128535A (ru) | Синергетическая композиция, содержащая четвертичное аммониевое соединение и карнозиновую кислоту для применения в качестве антибактериального, антигрибкового средства | |
SE0301904D0 (sv) | Novel imidazopyridine compound II with therapeutic effect | |
JP2023075371A (ja) | 新型コロナウイルス感染症(covid-19)の予防または治療剤および医薬組成物 | |
WO2023154804A3 (fr) | Méthode de traitement d'une lésion de la moelle épinière et composition correspondante | |
TH58970B (th) | สูตรผสมสำหรับใช้กับตา |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
UEP | Publication of translation of european patent specification | ||
EELA | Cancelled due to lapse of time |