ATE481403T1 - Substituierte 1-phenyl-1,5-dihydro-pyridoä3,2- büindol-2-on-derivate verwendbar als pharmazeutische antiinfektiva - Google Patents

Substituierte 1-phenyl-1,5-dihydro-pyridoä3,2- büindol-2-on-derivate verwendbar als pharmazeutische antiinfektiva

Info

Publication number
ATE481403T1
ATE481403T1 AT05747918T AT05747918T ATE481403T1 AT E481403 T1 ATE481403 T1 AT E481403T1 AT 05747918 T AT05747918 T AT 05747918T AT 05747918 T AT05747918 T AT 05747918T AT E481403 T1 ATE481403 T1 AT E481403T1
Authority
AT
Austria
Prior art keywords
pyridoä3
büindol
antiinfectives
dihydro
phenyl
Prior art date
Application number
AT05747918T
Other languages
English (en)
Inventor
Bart Kesteleyn
Sandrine Vendeville
Natalie Kindermans
Dominique Surleraux
Pierre Jean-Marie Raboisson
Piet Wigerinck
Annick Ann Peeters
Original Assignee
Tibotec Pharm Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tibotec Pharm Ltd filed Critical Tibotec Pharm Ltd
Application granted granted Critical
Publication of ATE481403T1 publication Critical patent/ATE481403T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/16Antivirals for RNA viruses for influenza or rhinoviruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
AT05747918T 2004-05-17 2005-05-17 Substituierte 1-phenyl-1,5-dihydro-pyridoä3,2- büindol-2-on-derivate verwendbar als pharmazeutische antiinfektiva ATE481403T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP04102170 2004-05-17
PCT/EP2005/052263 WO2005111035A1 (en) 2004-05-17 2005-05-17 6,7,8,9-substituted 1-phenyl-1,5-dihydro-pyrido[3,2-b]indol-2-ones useful as anti-infective pharmaceutical agents

Publications (1)

Publication Number Publication Date
ATE481403T1 true ATE481403T1 (de) 2010-10-15

Family

ID=34929105

Family Applications (1)

Application Number Title Priority Date Filing Date
AT05747918T ATE481403T1 (de) 2004-05-17 2005-05-17 Substituierte 1-phenyl-1,5-dihydro-pyridoä3,2- büindol-2-on-derivate verwendbar als pharmazeutische antiinfektiva

Country Status (14)

Country Link
US (2) US7622581B2 (de)
EP (1) EP1751156B1 (de)
JP (1) JP2007538050A (de)
CN (1) CN1976930B (de)
AR (1) AR049637A1 (de)
AT (1) ATE481403T1 (de)
BR (1) BRPI0511173A (de)
DE (1) DE602005023600D1 (de)
ES (1) ES2351702T3 (de)
MX (1) MXPA06013313A (de)
PL (1) PL1751156T3 (de)
RU (1) RU2377243C2 (de)
TW (1) TW200607502A (de)
WO (1) WO2005111035A1 (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2004647A1 (de) 2006-04-03 2008-12-24 Tibotec Pharmaceuticals Ltd. Hiv-inhibierende 3,4-dihydroimidazo[4,5-b]pyridin-5-one
WO2008037783A1 (en) * 2006-09-29 2008-04-03 Tibotec Pharmaceuticals Ltd. Process for preparing 2-oxo-2,5-dihydro-1h-pyrido[3,2-b]indole-3-carbonitriles
EA201101397A1 (ru) 2009-04-09 2012-05-30 Бёрингер Ингельхайм Интернациональ Гмбх Ингибиторы репликации вируса иммунодефицита человека
AU2011252351A1 (en) * 2010-05-14 2012-10-11 Affectis Pharmaceuticals Ag Novel methods for the preparation of P2X7R antagonists
RU2451680C1 (ru) 2011-02-21 2012-05-27 Общество С Ограниченной Ответственностью "Научно-Исследовательская Компания "Медбиофарм" Клатратный комплекс циклодекстрина или арабиногалактана с 9-фенил-симм-октагидроселеноксантеном, способ его получения (варианты), фармацевтическая композиция и лекарственное средство
RU2464042C1 (ru) * 2011-03-31 2012-10-20 Общество С Ограниченной Ответственностью "Научно-Исследовательская Компания "Медбиофарм" КЛАТРАТНЫЙ КОМПЛЕКС β-ЦИКЛОДЕКСТРИНА С ПРОИЗВОДНЫМ 5-ГИДРОКСИ-4-АМИНОМЕТИЛ-1-ЦИКЛОГЕКСИЛ(ИЛИ ЦИКЛОГЕПТИЛ)-3-АЛКОКСИКАРБОНИЛИНДОЛА, СПОСОБ ЕГО ПОЛУЧЕНИЯ (ВАРИАНТЫ), ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ И ЛЕКАРСТВЕННОЕ СРЕДСТВО
BR112014005935A2 (pt) 2011-09-16 2017-03-28 Fovea Pharmaceuticals derivados de anilina, sua preparação e sua aplicação terapêutica
RU2640081C1 (ru) * 2016-07-11 2017-12-26 Общество с ограниченной ответственностью "ЛАЙФ САЙНСЕС ОХФК" Фармацевтическая композиция и лекарственное средство на основе клатратного комплекса N-карбамоилметил-4-фенил-2-пирролидон или 4-фенилпирацетам с циклодекстрином, способы его получения (варианты)
JP7374916B2 (ja) * 2018-03-20 2023-11-07 コンパニー ゼネラール デ エタブリッスマン ミシュラン 少なくとも3重撚りを有する改善されたアラミド繊維コード
CN108530381B (zh) * 2018-05-07 2021-09-21 上海科技大学 一种由酰胺酯制备二胺衍生物的方法
WO2022212471A1 (en) * 2021-03-31 2022-10-06 Virginia Commonwealth University Bivalent ligands to understand dimerization of the mu opioid receptor and the chemokine receptor ccr5 in neurological disorders

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB427857A (en) 1934-08-02 1935-05-01 Newsum Sons & Company Ltd H A new or improved system of construction for skeleton structures, particularly vehicle body frames and door frames
US5145684A (en) 1991-01-25 1992-09-08 Sterling Drug Inc. Surface modified drug nanoparticles
PH30929A (en) 1992-09-03 1997-12-23 Janssen Pharmaceutica Nv Beads having a core coated with an antifungal and a polymer.
CN1110300C (zh) 1993-10-01 2003-06-04 阿斯特拉公司 工艺技术ⅰ
KR19990044257A (ko) 1996-05-20 1999-06-25 디르크 반테 생체이용율이 개선된 항진균성 조성물
SI0969821T1 (en) 1997-03-26 2003-10-31 Janssen Pharmaceutica N.V. Pellets having a core coated with an antifungal and a polymer
AU2002246659A1 (en) * 2000-12-18 2002-08-06 The Government Of The United States Of America, As Represented By The Secretary, Department Of Healt Benzoylalkylindolepyridinium compounds and pharmaceutical compositions comprising such compounds
WO2002055520A2 (en) * 2000-12-18 2002-07-18 Us Health Benzoylalkylindolepyridinium compounds and pharmaceutical compositions comprising such compounds
US6933303B2 (en) * 2001-10-19 2005-08-23 Transtech Pharma, Inc. Heteroaryl-fused nitrogen heterocycles as therapeutic agents
AP1927A (en) * 2002-11-15 2008-12-10 Tibotec Pharm Ltd Substituted indolepyridinium as anti-infective compounds

Also Published As

Publication number Publication date
US20070167434A1 (en) 2007-07-19
BRPI0511173A (pt) 2007-12-04
RU2377243C2 (ru) 2009-12-27
US20100029635A1 (en) 2010-02-04
PL1751156T3 (pl) 2011-03-31
CN1976930B (zh) 2011-01-19
WO2005111035A1 (en) 2005-11-24
MXPA06013313A (es) 2007-02-02
US7622581B2 (en) 2009-11-24
EP1751156B1 (de) 2010-09-15
JP2007538050A (ja) 2007-12-27
EP1751156A1 (de) 2007-02-14
DE602005023600D1 (de) 2010-10-28
TW200607502A (en) 2006-03-01
AR049637A1 (es) 2006-08-23
ES2351702T3 (es) 2011-02-09
CN1976930A (zh) 2007-06-06
RU2006144852A (ru) 2008-06-27

Similar Documents

Publication Publication Date Title
ATE481403T1 (de) Substituierte 1-phenyl-1,5-dihydro-pyridoä3,2- büindol-2-on-derivate verwendbar als pharmazeutische antiinfektiva
BRPI0618904A2 (pt) composto, composição farmacêutica, e, uso do composto
BRPI0614205A2 (pt) composto, composição farmacêutica, e, uso de composto
ATE415400T1 (de) Pyrazolopyridinderivate
NO20075628L (no) Farmasøytiske formuleringer
IS8578A (is) 3- karbamoýl - 2- pýridón afleiður
DK1725553T3 (da) Tetrahydropyridoindolderivater
ATE383361T1 (de) Pyrrazolopyrimidinderivate
ATE540935T1 (de) Chinazolinderivate
DK1753764T3 (da) Pyrrolopyridin-derivater
DK2033629T3 (da) Fast farmaceutisk sammensætning omfattende valsartan
ATE483702T1 (de) Neue pharmazeutische verbindungen
NL2000336A1 (nl) Spirocyclische derivaten.
ATE430142T1 (de) Phenylpiperazin-methanon-derivate
ATE404542T1 (de) 4-phenylpyrimidin-2-carbonitrilderivate
DE602005018177D1 (de) Drehzerstäubungskopf-lackiervorrichtung
DE602006018645D1 (de) 3-monosubstituiertes tropan-derivat als nociceptinrezeptor-ligand
DK1740574T3 (da) 4-amino-5-cyanopyrimidinderivater
ATE369347T1 (de) Trimere makrocyclisch substituierte halogen- benzolderivate
ITMI20051155A1 (it) Nuovi composti fluorurati, loro sintesi e uso.
ATE489943T1 (de) Pharmazeutische zusammensetzung mit 2,3-dihydro-6-nitroimidazoä2,1-büoxazolderivate
DE602005005033D1 (de) Sprühgetrocknete pharmazeutische zusammensetzungen
DK1720557T3 (da) Hurtig-opløselig, smagsmaskeret tablet
ITMI20041447A1 (it) Composizione farmaceutica comprendente gabapentina
ITMI20040943A1 (it) Composizione farmaceutica cicatrizzante

Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties