ATE37373T1 - Synergistinderivate, ihre herstellung und diese enthaltende pharmazeutische zubereitungen. - Google Patents

Synergistinderivate, ihre herstellung und diese enthaltende pharmazeutische zubereitungen.

Info

Publication number
ATE37373T1
ATE37373T1 AT84401480T AT84401480T ATE37373T1 AT E37373 T1 ATE37373 T1 AT E37373T1 AT 84401480 T AT84401480 T AT 84401480T AT 84401480 T AT84401480 T AT 84401480T AT E37373 T1 ATE37373 T1 AT E37373T1
Authority
AT
Austria
Prior art keywords
azepin
azetidin
pyrrolidin
piperidin
alkyl
Prior art date
Application number
AT84401480T
Other languages
English (en)
Inventor
Jean-Pierre Corbet
Claude Cotrel
Daniel Farge
Jean-Marc Paris
Original Assignee
Rhone Poulenc Sante
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Sante filed Critical Rhone Poulenc Sante
Application granted granted Critical
Publication of ATE37373T1 publication Critical patent/ATE37373T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • C07K5/06182—Dipeptides with the first amino acid being heterocyclic and Pristinamycin II; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00—Peptide or protein sequence
    • Y10S930/01—Peptide or protein sequence
    • Y10S930/19—Antibiotic
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00—Peptide or protein sequence
    • Y10S930/01—Peptide or protein sequence
    • Y10S930/27—Cyclic peptide or cyclic protein

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Public Health (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Saccharide Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Lubricants (AREA)
  • Orthopedics, Nursing, And Contraception (AREA)
  • Fixed Capacitors And Capacitor Manufacturing Machines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT84401480T 1983-07-13 1984-07-12 Synergistinderivate, ihre herstellung und diese enthaltende pharmazeutische zubereitungen. ATE37373T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8311707A FR2549065B1 (fr) 1983-07-13 1983-07-13 Nouveaux derives de synergistines, leur preparation et les compositions pharmaceutiques qui les contiennent
EP84401480A EP0135410B1 (de) 1983-07-13 1984-07-12 Synergistinderivate, ihre Herstellung und diese enthaltende pharmazeutische Zubereitungen

Publications (1)

Publication Number Publication Date
ATE37373T1 true ATE37373T1 (de) 1988-10-15

Family

ID=9290814

Family Applications (1)

Application Number Title Priority Date Filing Date
AT84401480T ATE37373T1 (de) 1983-07-13 1984-07-12 Synergistinderivate, ihre herstellung und diese enthaltende pharmazeutische zubereitungen.

Country Status (18)

Country Link
US (1) US4590004A (de)
EP (1) EP0135410B1 (de)
JP (1) JPH0631252B2 (de)
KR (1) KR910002842B1 (de)
AT (1) ATE37373T1 (de)
AU (1) AU567951B2 (de)
CA (1) CA1222513A (de)
DE (1) DE3474146D1 (de)
DK (1) DK170421B1 (de)
ES (1) ES534314A0 (de)
FI (1) FI78106C (de)
FR (1) FR2549065B1 (de)
GR (1) GR82382B (de)
IE (1) IE57550B1 (de)
IL (1) IL72398A (de)
PT (1) PT78895B (de)
SU (1) SU1396968A3 (de)
ZA (1) ZA845315B (de)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2576022B1 (fr) * 1985-01-11 1987-09-11 Rhone Poulenc Sante Nouveaux derives de la pristinamycine ii b, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2599036B1 (fr) * 1986-05-22 1988-09-09 Rhone Poulenc Sante Nouveaux derives de synergistines, leur preparation et les compositions pharmaceutiques qui les contiennent
GB8616768D0 (en) * 1986-07-09 1986-08-13 May & Baker Ltd Process
US4859690A (en) * 1986-11-21 1989-08-22 Merck & Co., Inc. Therapeutic virginiamycin M1 analogs
US4772595A (en) * 1986-11-21 1988-09-20 Merck & Co., Inc. Synthetic virginiamycin M1 analogs
US4762923A (en) * 1986-11-21 1988-08-09 Merck & Co. Inc. Fermentation analogs of virginiamycin M1
ES2033335T3 (es) * 1987-07-07 1993-03-16 Rhone-Poulenc Sante Nuevo procedimiento para la preparacion de derivados de la pristinamicina ii b.
FR2655343B1 (fr) * 1989-12-05 1992-05-07 Rhone Poulenc Sante Procede de preparation de synergistine.
FR2664599B1 (fr) * 1990-07-16 1993-06-18 Rhone Poulenc Sante Vinylsulfonyl pristinamycine et sa preparation.
US5242938A (en) * 1992-08-27 1993-09-07 Merck & Co., Inc. Derivatives of virginiamycin M1
FR2701709B1 (fr) * 1993-02-17 1995-04-07 Rhone Poulenc Rorer Sa Forme purifiée de streptograminés, sa préparation et les compositions pharmaceutiques qui la contiennent.
FR2755857B1 (fr) * 1996-11-19 1998-12-24 Rhone Poulenc Rorer Sa Compositions pharmaceutiques stabilisees, a base de quinupristine et de dalfopristine et leur preparation
FR2766489B1 (fr) * 1997-07-28 1999-08-27 Rhone Poulenc Rorer Sa Derives de streptogramines, leur preparation et les compositions qui les contiennent
FR2795733B1 (fr) * 1999-06-30 2001-09-07 Aventis Pharma Sa Derives de streptogramines, leur preparation et les compositions qui les contiennent
FR2818644B1 (fr) * 2000-12-21 2004-10-22 Aventis Pharma Sa Derives de streptogramines, leur preparation et les compositions qui les contiennent
CN103360463B (zh) * 2012-04-08 2016-06-08 浙江海正药业股份有限公司 一种达福普汀及其中间体的分离纯化方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2549063B1 (fr) * 1983-07-13 1985-10-25 Rhone Poulenc Sante Nouveaux derives de synergistines, leur preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
FI842813A0 (fi) 1984-07-12
FI78106C (fi) 1989-06-12
ZA845315B (en) 1985-02-27
US4590004A (en) 1986-05-20
KR910002842B1 (ko) 1991-05-06
AU567951B2 (en) 1987-12-10
IL72398A (en) 1987-10-30
FR2549065A1 (fr) 1985-01-18
DK342484A (da) 1985-01-14
AU3047184A (en) 1986-01-16
PT78895A (fr) 1984-08-01
DK170421B1 (da) 1995-08-28
JPS6075483A (ja) 1985-04-27
FR2549065B1 (fr) 1985-10-25
ES8504202A1 (es) 1985-04-01
DK342484D0 (da) 1984-07-12
IE57550B1 (en) 1992-11-18
IL72398A0 (en) 1984-11-30
ES534314A0 (es) 1985-04-01
SU1396968A3 (ru) 1988-05-15
DE3474146D1 (en) 1988-10-27
KR850001216A (ko) 1985-03-16
FI78106B (fi) 1989-02-28
EP0135410A1 (de) 1985-03-27
FI842813A (fi) 1985-01-14
IE841788L (en) 1985-01-13
PT78895B (fr) 1986-08-14
CA1222513A (fr) 1987-06-02
EP0135410B1 (de) 1988-09-21
JPH0631252B2 (ja) 1994-04-27
GR82382B (de) 1984-12-13

Similar Documents

Publication Publication Date Title
ATE37373T1 (de) Synergistinderivate, ihre herstellung und diese enthaltende pharmazeutische zubereitungen.
DK0582788T3 (da) 7-(Substituerede)-9-[(substitueret glycyl)-amido]-demethyl-6-deoxytetracycliner
TW289757B (de)
TR200000197T2 (tr) Yeni bileşimler
ATE242783T1 (de) Glycopeptid-derivate und pharmazeutische zusammensetzungen, die sie enthalten
AU5670690A (en) Lysolecithin derivatives for treating autoimmune diseases
ATE212629T1 (de) Diaminopyrimidine, diese enthaltende pharmazeutische zusammensetzungen und ihre verwendung als antibakterielle mittel
DE69502587D1 (de) 2-heteroaryl-5,11-dihydro-6h-dipyrido[3,2-b:2',3'-e] [1,4]diazepine und ihre verwendung zur vorbeugung und behandlung von hiv-infektion
DE69118064D1 (de) Diamino-s-Triazinonderivate und diese enthaltende selbstlöschende polymere Zusammensetzungen
AU567570B2 (en) Synergistine derivatives
IL97913A0 (en) Heterocyclic compounds,their preparation and pharmaceutical compositions containing them
DE69011781D1 (de) 1-acyl-2-pyrrolidinone zur Verbesserung der Lernfähigkeit und des Gedächtnisses und diese enthaltende pharmazeutische Zubereitungen.
DE69115135D1 (de) 1-Alkyl-3-(Acylamino)-Epsilon-Caprolactame zur Verbesserung der Lernfähigkeit und des Gedächtnisses und diese enthaltende pharmazeutische Zubereitungen.
NZ222078A (en) 1,2,4-triazole derivatives and pharmaceutical compositions
ATE2786T1 (de) 1-(2-propynyloxy)-2-amino-3-propanol-aether, ihre herstellung und sie enthaltende pharmazeutische zusammensetzung.

Legal Events

Date Code Title Description
EELA Cancelled due to lapse of time