ATE300522T1 - Cyclisierungsverfahrensschritt bei der herstellung von chinolonen und naphthyridinen - Google Patents
Cyclisierungsverfahrensschritt bei der herstellung von chinolonen und naphthyridinenInfo
- Publication number
- ATE300522T1 ATE300522T1 AT01990192T AT01990192T ATE300522T1 AT E300522 T1 ATE300522 T1 AT E300522T1 AT 01990192 T AT01990192 T AT 01990192T AT 01990192 T AT01990192 T AT 01990192T AT E300522 T1 ATE300522 T1 AT E300522T1
- Authority
- AT
- Austria
- Prior art keywords
- naphthyridines
- quinolones
- production
- process step
- cyclization process
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 3
- 150000005054 naphthyridines Chemical class 0.000 title 1
- LISFMEBWQUVKPJ-UHFFFAOYSA-N quinolin-2-ol Chemical compound C1=CC=C2NC(=O)C=CC2=C1 LISFMEBWQUVKPJ-UHFFFAOYSA-N 0.000 title 1
- 238000007363 ring formation reaction Methods 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000003153 chemical reaction reagent Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- Virology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Molecular Biology (AREA)
- AIDS & HIV (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Quinoline Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US25563300P | 2000-12-14 | 2000-12-14 | |
| PCT/US2001/048536 WO2002048113A1 (en) | 2000-12-14 | 2001-12-07 | Cyclization process step in the making of quinolones and naphthyridines |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE300522T1 true ATE300522T1 (de) | 2005-08-15 |
Family
ID=22969207
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT01990192T ATE300522T1 (de) | 2000-12-14 | 2001-12-07 | Cyclisierungsverfahrensschritt bei der herstellung von chinolonen und naphthyridinen |
Country Status (19)
| Country | Link |
|---|---|
| EP (1) | EP1343766B1 (de) |
| JP (2) | JP4417007B2 (de) |
| KR (1) | KR100603163B1 (de) |
| CN (1) | CN1232508C (de) |
| AT (1) | ATE300522T1 (de) |
| AU (2) | AU2905702A (de) |
| BR (1) | BR0116229A (de) |
| CA (1) | CA2427831C (de) |
| CZ (1) | CZ20031379A3 (de) |
| DE (1) | DE60112325T2 (de) |
| DK (1) | DK1343766T3 (de) |
| ES (1) | ES2247190T3 (de) |
| HU (1) | HUP0303991A3 (de) |
| IL (2) | IL155677A0 (de) |
| MX (1) | MXPA03005338A (de) |
| NO (1) | NO325236B1 (de) |
| NZ (1) | NZ525569A (de) |
| PL (1) | PL207394B1 (de) |
| WO (1) | WO2002048113A1 (de) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR100735587B1 (ko) * | 2002-08-05 | 2007-07-04 | 더 프록터 앤드 갬블 캄파니 | 퀴놀론계 항생제 중간체의 제조 방법 |
| US6803469B2 (en) * | 2002-08-05 | 2004-10-12 | The Procter & Gamble Company | Process for preparing quinolone antibiotic intermediates |
| US7176220B2 (en) * | 2002-11-20 | 2007-02-13 | Japan Tobacco Inc. | 4-oxoquinoline compound and use thereof as pharmaceutical agent |
| US7402674B2 (en) | 2004-01-31 | 2008-07-22 | Sanofi-Aventis Deutschland Gmbh, | 7-Phenylamino-4-quinolone-3-carboxylic acid derivatives, process for their preparation and their use as medicaments |
| JP4669040B2 (ja) | 2006-03-06 | 2011-04-13 | 日本たばこ産業株式会社 | ４−オキソキノリン化合物の製造方法 |
| WO2007102499A1 (ja) | 2006-03-06 | 2007-09-13 | Japan Tobacco Inc. | ４－オキソキノリン化合物の製造方法 |
| AU2007296555B2 (en) | 2006-09-12 | 2012-07-12 | Gilead Sciences, Inc. | Process and intermediates for preparing integrase inhibitors |
| US8658183B2 (en) | 2007-08-09 | 2014-02-25 | Taigen Biotechnology Company, Ltd. | Antimicrobial parenteral formulation |
| AR068403A1 (es) | 2007-09-11 | 2009-11-18 | Gilead Sciences Inc | Proceso e intermediarios para la preparacion de inhibidores de integrasa |
| EA018653B1 (ru) | 2008-07-01 | 2013-09-30 | Тайджен Байотекнолоджи Ко., Лтд. | Лечение инфекций, вызванных антибиотикоустойчивыми бактериями |
| AU2013296289B2 (en) | 2012-08-03 | 2017-10-05 | Gilead Sciences, Inc. | Process and intermediates for preparing integrase inhibitors |
| CN112969965A (zh) | 2018-07-19 | 2021-06-15 | 林特弗德有限公司 | 噻吨酮衍生物、包含其的组合物和包含所述组合物的图案形成方法 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0775145A1 (de) * | 1994-08-02 | 1997-05-28 | The Procter & Gamble Company | Verfahren zur herstellung von quinolonyl laktam antimikorbielle verbindungen und zwischenprodukte |
| EP0775114B1 (de) * | 1994-08-02 | 2000-03-22 | The Procter & Gamble Company | Verfahren zur herstellung von antimikrobiellen verbindungen |
-
2001
- 2001-12-07 BR BR0116229-2A patent/BR0116229A/pt not_active IP Right Cessation
- 2001-12-07 MX MXPA03005338A patent/MXPA03005338A/es active IP Right Grant
- 2001-12-07 IL IL15567701A patent/IL155677A0/xx active IP Right Grant
- 2001-12-07 CN CNB018207146A patent/CN1232508C/zh not_active Expired - Lifetime
- 2001-12-07 HU HU0303991A patent/HUP0303991A3/hu unknown
- 2001-12-07 AU AU2905702A patent/AU2905702A/xx active Pending
- 2001-12-07 ES ES01990192T patent/ES2247190T3/es not_active Expired - Lifetime
- 2001-12-07 JP JP2002549644A patent/JP4417007B2/ja not_active Expired - Fee Related
- 2001-12-07 CZ CZ20031379A patent/CZ20031379A3/cs unknown
- 2001-12-07 AU AU2002229057A patent/AU2002229057B2/en not_active Ceased
- 2001-12-07 DK DK01990192T patent/DK1343766T3/da active
- 2001-12-07 KR KR1020037007905A patent/KR100603163B1/ko not_active Expired - Fee Related
- 2001-12-07 DE DE60112325T patent/DE60112325T2/de not_active Expired - Lifetime
- 2001-12-07 AT AT01990192T patent/ATE300522T1/de active
- 2001-12-07 EP EP01990192A patent/EP1343766B1/de not_active Expired - Lifetime
- 2001-12-07 PL PL363355A patent/PL207394B1/pl not_active IP Right Cessation
- 2001-12-07 CA CA002427831A patent/CA2427831C/en not_active Expired - Fee Related
- 2001-12-07 NZ NZ525569A patent/NZ525569A/en not_active IP Right Cessation
- 2001-12-07 WO PCT/US2001/048536 patent/WO2002048113A1/en not_active Ceased
-
2003
- 2003-04-30 IL IL155677A patent/IL155677A/en not_active IP Right Cessation
- 2003-06-12 NO NO20032667A patent/NO325236B1/no not_active IP Right Cessation
-
2009
- 2009-10-05 JP JP2009231801A patent/JP2010001315A/ja not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| IL155677A0 (en) | 2003-11-23 |
| BR0116229A (pt) | 2003-11-04 |
| EP1343766A1 (de) | 2003-09-17 |
| IL155677A (en) | 2009-02-11 |
| KR100603163B1 (ko) | 2006-07-24 |
| CN1481365A (zh) | 2004-03-10 |
| CZ20031379A3 (cs) | 2003-11-12 |
| AU2905702A (en) | 2002-06-24 |
| HUP0303991A3 (en) | 2012-09-28 |
| PL363355A1 (en) | 2004-11-15 |
| NZ525569A (en) | 2004-09-24 |
| DE60112325D1 (de) | 2005-09-01 |
| NO325236B1 (no) | 2008-03-03 |
| KR20030063420A (ko) | 2003-07-28 |
| NO20032667L (no) | 2003-08-14 |
| ES2247190T3 (es) | 2006-03-01 |
| NO20032667D0 (no) | 2003-06-12 |
| HUP0303991A2 (hu) | 2004-04-28 |
| JP2004515542A (ja) | 2004-05-27 |
| PL207394B1 (pl) | 2010-12-31 |
| AU2002229057B2 (en) | 2005-04-21 |
| CA2427831C (en) | 2009-08-18 |
| WO2002048113A1 (en) | 2002-06-20 |
| EP1343766B1 (de) | 2005-07-27 |
| JP4417007B2 (ja) | 2010-02-17 |
| JP2010001315A (ja) | 2010-01-07 |
| CA2427831A1 (en) | 2002-06-20 |
| DK1343766T3 (da) | 2005-10-31 |
| DE60112325T2 (de) | 2006-05-24 |
| CN1232508C (zh) | 2005-12-21 |
| MXPA03005338A (es) | 2003-10-06 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification |
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